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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC11959 Naratriptan

    盐酸那拉曲坦,GR-85548A

     A potent 5-HT1B and 5-HT1D receptor agonist
  3. GC12443 Tranilast Sodium

    曲尼司特钠; MK-341 sodium; SB 252218 sodium

     An antiallergic agent
  4. GC17891 Tizanidine HCl

    盐酸替扎尼定

     An α2-adrenergic receptor agonist
  5. GC15629 Tizanidine

    替扎尼定

     An α2-adrenergic receptor agonist
  6. GC16785 Prazosin

    哌唑嗪

     Prazosin是一种特异性的α1-肾上腺素能受体（α1-AR）的拮抗剂，与人类重组α1A-AR、α1B-AR和α1D-AR的结合常数（Ki值）分别为0.2、0.25和0.32nM，与α2-AR的Ki值分别为340和3.7nM（在表达α2A-AR 的 HT-29 细胞和表达α2B-AR 的 NG108 细胞中）。
  7. GC16740 Alfuzosin

    阿夫唑嗪; SL 77499

     Alfuzosin (SL 77499-10) 是一种具有口服活性、选择性和竞争性的 α1-肾上腺素受体拮抗剂。
  8. GC12687 Bimatoprost

    比马前列素; AGN 192024

     The ocular hypotensive ingredient in Lumigan
  9. GC13428 Mosapride

    莫沙必利; TAK-370; AS-4370

     A 5-HT4 receptor agonist
  10. GC17081 Detomidine HCl

    盐酸地托咪定

     An α2-adrenoceptor agonist
  11. GC17197 Detomidine

    地托咪定

     Detomidine 是一种咪唑衍生物，是一种有效的 α2-肾上腺素能激动剂。
  12. GC10194 Ivabradine HCl

    盐酸伊伐布雷定

     An HCN channel blocker
  13. GC13371 Fluticasone propionate

    丙酸氟替卡松

     A synthetic corticosteroid and glucocorticoid receptor agonist
  14. GC16496 Ticlopidine

    盐酸噻氯匹定,PCR 5332

     A P2Y12 receptor antagonist with antiplatelet activity
  15. GC12920 Pregnenolone

    孕烯醇酮; 3β-Hydroxy-5-pregnen-20-one

     A natural steroid hormone
  16. GC17347 Alprostadil

    前列地尔; Alprostadil; PGE1;Prostaglandin E1

     前列地尔Alprostadil作为前列腺素受体配体,对小鼠EP3、EP4、EP2、IP和EP1的结合亲和Kis分别为1.1 nM、2.1 nM、10 nM、33 nM和36 nM。
  17. GC16871 Perindopril

    培哚普利; S-9490

     An orally active ACE inhibitor
  18. GC13478 Pizotifen Malate

    苯噻啶苹果酸盐,Pizotyline malate; BC-105 malate

     A triptan
  19. GC13053 Pizotifen

    苯噻啶; Pizotyline; BC-105

     A triptan
  20. GC13092 Fluvoxamine

    氟伏沙明; DU-23000

     Fluvoxamine是一种选择性血清素（5-HT）再摄取抑制剂（SSRI），具有抗抑郁活性。
  21. GC13447 Doxazosin

    多沙唑嗪; UK 33274

     An α1-AR antagonist
  22. GC17593 Lurasidone HCl

    盐酸鲁拉西酮; SM-13496 Hydrochloride

     An atypical antipsychotic
  23. GC16891 Quetiapine Fumarate

    富马酸喹硫平

     An antagonist of diverse neurological receptors
  24. GC15223 Tropisetron Hydrochloride

    盐酸托烷司琼

     A 5-HT3 receptor antagonist
  25. GC15918 Formoterol Hemifumarate

    富马酸福莫特罗,(±)Formoterol fumarate

     强效、选择性和长效 β2-肾上腺素能受体激动剂
  26. GC14769 Carvedilol

    卡维地洛; BM 14190

     Carvedilol是一种非选择性α1和β-肾上腺素能受体（Ars）的拮抗剂。
  27. GC11651 Ondansetron hydrochloride dihydrate

    盐酸昂丹司琼二水物; GR 38032 hydrochloride dihydrate; SN 307 hydrochloride dihydrate

     An Analytical Reference Material
  28. GC16087 Fesoterodine Fumarate

    富马酸非索罗定

     A muscarinic acetylcholine receptor antagonist
  29. GC14512 Fenspiride HCl

    盐酸芬司必利

     A histamine H1 receptor antagonist
  30. GC11219 (R)-(+)-Tolterodine

    托特罗定; (R)-(+)-Tolterodine; (+)-Tolterodine; (R)-Tolterodine; PNU-200583

     (R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂，在体内对膀胱的选择性优于唾液腺。
  31. GC17917 Palonosetron HCl

    盐酸帕洛诺司琼

     A 5-HT3 receptor antagonist
  32. GC11465 Bosentan Hydrate

    波生坦水合物

     An antagonist of endothelin receptors
  33. GC16269 Bosentan

    波生坦

     An antagonist of endothelin receptors
  34. GC15772 Darifenacin HBr

    氢溴酸达非那新; UK-88525 hydrobromide

     A muscarinic M3 receptor antagonist
  35. GC17053 Eletriptan HBr

    依来曲普坦氢溴酸盐; Eletriptan HBr; UK-116044 hydrobromide

     An agonist of 5-HT1B and 5-HT1D receptors
  36. GC17182 Solifenacin succinate

    索非那新琥珀酸盐; YM905

     A muscarinic M1, M2, and M3 receptor antagonist
  37. GC17954 Tolterodine tartrate

    酒石酸托特罗定,Kabi-2234; PNU-200583E

     A muscarinic acetylcholine receptor antagonist
  38. GC15317 SB408124 A potent orexin 1 receptor antagonist
  39. GC16708 Cinacalcet HCl

    盐酸西那卡塞; AMG-073 hydrochloride

     An allosteric agonist of the CaSR
  40. GC17949 Plerixafor 8HCl (AMD3100 8HCl)

    盐酸普乐沙福; AMD3100 octahydrochloride; JM3100 octahydrochloride; SID791 octahydrochloride

     An antagonist of CXCR4
  41. GC11182 LY404039

    (1R,4S,5S,6S)-4-氨基-2-硫杂双环[3.1.0]己烷-4,6-二甲酸2,2-二氧化物

     An agonist of mGluR2 and mGluR3
  42. GC10765 Valsartan

    缬沙坦; CGP 48933

     An AT1 receptor antagonist
  43. GC13911 S1RA hydrochloride

    4-[2-[[5-甲基-1-(2-萘基)-1H-吡唑-3-基]氧基]乙基]吗啉盐酸盐(1:1),E-52862 hydrochloride

     A σ1 receptor antagonist
  44. GC10407 S1RA

    E-52862

     A σ1 receptor antagonist
  45. GC10249 Losartan

    氯沙坦; DuP-753

     Losartan是一种血管紧张素II受体拮抗剂（IC50=20nM）。
  46. GC15839 Zafirlukast

    扎鲁司特; ICI 204219

     A selective CysLT1 receptor antagonist
  47. GC15029 Glycopyrrolate

    格隆溴铵; Glycopyrronium bromide; Glycopyrrolate bromide

     A muscarinic acetylcholine receptor antagonist
  48. GC15331 Prednisolone

    泼尼松龙

     The active metabolite of prednisone
  49. GC16772 Cortisone acetate

    醋酸可的松; Cortisone 21-acetate

     A synthetic glucocorticoid
  50. GC10642 Azilsartan medoxomil monopotassium

    阿齐沙坦酯衍生物,Azilsartan kamedoxomil; TAK 491 monopotassium

     Azilsartan medoxomil monopotassium 是一种口服血管紧张素 II 受体 1 型拮抗剂，IC50 为 0.62 nM，用于治疗成人原发性高血压。
  51. GC10799 Iloperidone hydrochloride

    盐酸伊潘立酮; HP 873 hydrochloride

     An atypical antipsychotic

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