Free Fatty Acid Receptors
Free Fatty Acid Receptors(游离脂肪酸受体)
FFAR1 (GPR40) is a G protein-coupled receptor for medium and long chain saturated and unsaturated fatty acids. It plays a role in glucose homeostasis, insulin secretion and bone homeostasis etc.
Free Fatty Acid Receptors 相关产品(16)
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10373 | MEDICA 16 | 87272-20-6 | - | |
A GPR40 agonist and GPR120 partial agonist | ||||
| GC10922 | TUG 424 | 1082058-99-8 | >98.00% | |
A selective FFAR1 (GPR40) agonist | ||||
| GC11467 | AS 2034178 | 1030846-42-4 | - | |
AS 2034178 是一种特异性的口服活性 GPR40 激动剂,具有葡萄糖依赖性胰岛素分泌增强作用。 | ||||
| GC16176 | GSK 137647 | 349085-82-1 | >99.50% | |
A selective GPR120 agonist | ||||
| GC17149 | 4-CMTB | 300851-67-6 | >99.00% | |
4-CMTB是一种选择性的游离脂肪酸受体2(FFA2/GPR43)激动剂和正变构调节剂。 | ||||
| GC17753 | AH 7614 | 6326-06-3 | >98.00% | |
A selective FFAR4 antagonist | ||||
| GC11434 | GSK1292263 | 1032823-75-8 | >99.00% | |
An agonist of GPR119 | ||||
| GC12401 | GW9508 | 885101-89-3 | >98.00% | |
An agonist of GPR40 | ||||
| GC14027 | GW-1100 | 306974-70-9 | - | |
A selective GPR40 antagonist | ||||
| GC16054 | TUG-770 | 1402601-82-4 | >99.50% | |
An agonist of FFA1/GPR40 | ||||
| GC16555 | TAK-875 | 1000413-72-8 | >98.50% | |
TAK-875是一种有效的,高选择性的口服生物利用的GPR40(G蛋白偶联受体40)激动剂,对人GPR40的EC 50 值为0.014μM。 | ||||
| GC50293 | CATPB | 1322598-09-3 | >98.00% | |
CATPB 是一种有效的选择性游离脂肪酸受体 2 (FFA2R/GPR43) 拮抗剂。 | ||||
| GC50313 | ZQ 16 | 376616-73-8 | - | |
Selective GPR84 agonist | ||||
| GC50333 | AMG 837 hemicalcium salt | 1291087-14-3 | - | |
An FFAR1 (GPR40) partial | ||||
| GC50578 | AZ 1729 | 2016864-46-1 | - | |
AZ 1729 是一种有效的游离脂肪酸 2 受体 (FFA2) 激活剂,可作为直接变构激动剂和正变构调节剂。 | ||||
| GC50662 | DL 175 | 2487253-25-6 | >98.00% | |
Potent and selective GPR84 biased agonist (EC50 = 33 nM) | ||||
