Adenosine Receptor(腺苷受体)

Cat.No. 产品名称 Information

GC17413 (±)-5'-Chloro-5'-deoxy-ENBA adenosine A1 receptor agonist, selective and high-affinity

GC10600 1,3-Dipropyl-8-phenylxanthine

A1 adenosine antagonist

GC11112 2'-MeCCPA An adenosine A₁ receptor agonist

GC10116 2-chloro-3-Deazaadenosine

6-Amino-2-chloropurine riboside,2-CADO,NSC 158900

Agonist of adenosine receptors

GC11665 2-Chloro-N6-cyclopentyladenosine

2-氯-N6-环戊基腺苷

An adenosine A₁ receptor antagonist

GC15111 2-Chloroadenosine

2-氯腺嘌呤核苷

An adenosine A receptor agonist

GC17503 2-Cl-IB-MECA

CF-102; 2-Cl-IB-MECA

An adenosine A₃ receptor agonist

GC11002 5'-(N-Cyclopropyl)carboxamidoadenosine

CPCA

A specific adenosine A₂ receptor agonist

GC13274 8-Aminoadenine

Adenine receptor agonist

GC50354 8-Cyclopentyl-1,3-dimethylxanthine

A1受体拮抗剂,CPT

An adenosine A₁ receptor antagonist

GC30918 A2A receptor antagonist 1

CPI-444 analog

A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。

GC30987 A2AR-agonist-1

JMF 1907

A2AR-agonist-1是腺苷A2A受体（A2AR）和平衡型核苷转运体1（ENT1）的强效激动剂，其Ki 值分别为 4.39 和 3.47。

GC38104 A2aR/A2bR antagonist-1

AB928

An adenosine A_2A and A_2B receptor dual antagonist

GC31974 A2B receptor antagonist 1

A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂，来自专利WO2009157938A1实例9B。

GC62820 A2B receptor antagonist 2

N-(4,6,7-三甲基喹唑啉-2-基)胍

A2B receptor antagonist 2 (compound 18) 是腺苷受体 A2B 的拮抗剂，其对rA1、rA2A 和 hA2BKi 值分别为2.30 μM、6.8 μM 和3.44 μM。

GC74081 A3AR antagonist 5 A3AR antagonist 5（化合物16）是人腺苷A3受体的选择性拮抗剂，亲和力pC为4.542μM。

GC30993 AB-MECA

1-[6-[[(4-氨基苯基)甲基]氨基]-9H-嘌呤-9-基]-1-脱氧-N-甲基-Β-D-呋喃脲酰胺

An adenosine A₃ receptor agonist

GC34143 Acefylline (Theophyllineacetic acid)

茶碱乙酸; Theophyllineacetic acid; Theophylline-7-acetic acid

An Analytical Reference Standard

GC19630 Adenosine 2′-monophosphate

腺苷-2'-一磷酸,2'-AMP; Adenosine 2'-phosphate; AMP 2'-phosphate

腺苷 &2#8242;-一磷酸 (2'-AMP) 被细胞外 2',3'-CAMP 转化。

GC35248 Adenosine 5'-monophosphate monohydrate

腺苷-5'-单磷酸一水合物,5'-AMP monohydrate

Adenosine 5'-monophosphate monohydrate (5'-Adenylic acid, 5'-AMP) is an activator of a class of protein kinases known as AMP-activated protein kinase (AMPK).

GC38733 Adenosine A1 receptor activator T62 Adenosine A1 receptor activator T62 是腺苷 A1 受体 (adenosine A1 receptor) 的变构增强剂。Adenosine A1 receptor activator T62 在急性疼痛的动物模型中产生抗伤害感受，并在炎性和神经损伤性疼痛的模型中降低超敏反应。

GC38884 Adenosine amine congener

ADAC

An adenosine A₁ receptor agonist

GC35249 Adenosine antagonist-1 Adenosine antagonist-1 是一个腺苷 A3 受体 (AA3R) 拮抗剂。

GC65901 Adenosine receptor antagonist 2 Adenosine receptor antagonist 2 是一种口服有效的 A2a/A2b 腺苷受体拮抗剂，IC50 分别为 1 nM 和 3 nM。Adenosine receptor antagonist 2 具有抗肿瘤活性。

GC66007 Adenosine receptor antagonist 3 Adenosine receptor antagonist 3 是一种有效的腺苷受体拮抗剂。Adenosine receptor antagonist 3 具有研究癌症疾病的潜力 (摘自专利 WO2019233994A1，化合物1)。

GC25051 Alloxazine

Isoalloxazine

Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.