Adenosine Receptor
Adenosine Receptor(腺苷受体)
Adenosine receptor (P1 receptors) is a class of purinergic receptors, G protein-coupled receptors with adenosine as endogenous ligand.
Adenosine Receptor 相关产品(130)
- GC17413(±)-5'-Chloro-5'-deoxy-ENBACAS: 103626-26-2
adenosine A1 receptor agonist, selective and high-affinity
- GC25051AlloxazineCAS: 490-59-5
Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
- GC30918A2A receptor antagonist 1CAS: 443103-97-7纯度: >99.50%
A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。
- GC30987A2AR-agonist-1CAS: 41552-95-8纯度: >98.00%
A2AR-agonist-1是腺苷A2A受体(A2AR)和平衡型核苷转运体1(ENT1)的强效激动剂,其Ki 值分别为 4.39 和 3.47。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15111 | 2-Chloroadenosine | 146-77-0 | >99.50% | |
An adenosine A receptor agonist | ||||
| GC15304 | NECA | 35920-39-9 | >99.50% | |
NECA是一种非选择性腺苷受体激动剂。 | ||||
| GC15689 | XCC | 96865-83-7 | - | |
Adenosine receptor antagonist | ||||
| GC15986 | LUF6000 | 890087-21-5 | >99.50% | |
A positive allosteric modulator of adenosine A 3 receptors | ||||
| GC16099 | DPCPX | 102146-07-6 | >98.00% / >99.00% | |
DPCPX 是一种高效、选择性强且具有高亲和力的 A 1 腺苷受体拮抗剂,对大鼠细胞膜腺苷酸环化酶的 K i 值为 0.45 nM。 | ||||
| GC16159 | ANR 94 | 634924-89-3 | - | |
ANR 94 是一种有效的选择性腺苷 A2A 受体 (AA2AR) 拮抗剂,对 hAA2AR 的 Ki 值为 46 nM。 | ||||
| GC17413 | (±)-5'-Chloro-5'-deoxy-ENBA | 103626-26-2 | - | |
adenosine A1 receptor agonist, selective and high-affinity | ||||
| GC17499 | Lu AA 47070 | 913842-25-8 | - | |
adenosine A2A receptor antagonist | ||||
| GC17503 | 2-Cl-IB-MECA | 163042-96-4 | >98.00% | |
An adenosine A 3 receptor agonist | ||||
| GC17756 | PSB 1115 | 152529-79-8 | - | |
PSB 1115是一种选择性A2B腺苷受体拮抗剂。 | ||||
| GC17844 | PSB 0788 | 1027513-54-7 | >98.00% | |
PSB 0788 是一种新型选择性高亲和力 A2B 拮抗剂,IC50 值为 3.64 nM,Ki 值为 0.393 nM。 | ||||
| GC18114 | BAY 60-6583 | 910487-58-0 | >99.50% | |
BAY 60-6583是一种高亲和力、高选择性腺苷A 2 B受体激动剂(EC 50 = 2.8nM)。 | ||||
| GC19049 | AZD4635 | 1321514-06-0 | >99.50% | |
AZD4635是一种强效、选择性的口服腺苷2A受体(A2AR)抑制剂,K i 值为1.7nM。 | ||||
| GC19197 | IB-MECA | 152918-18-8 | >98.00% | |
An adenosine A 3 receptor agonist | ||||
| GC19376 | Vipadenant | 442908-10-3 | >98.00% | |
A selective adenosine A 2A receptor antagonist | ||||
| GC19502 | BAY-545 | 1699717-32-2 | - | |
An adenosine A 2B receptor antagonist | ||||
| GC19630 | Adenosine 2′-monophosphate | 130-49-4 | - | |
腺苷 &2#8242;-一磷酸 (2'-AMP) 被细胞外 2',3'-CAMP 转化。 | ||||
| GC25051 | Alloxazine | 490-59-5 | - | |
Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor. | ||||
| GC30739 | N-0861 racemate | 121241-87-0 | - | |
N-0861racemate是N-0861的外消旋体。N-0861是一种选择性腺苷A1受体拮抗剂。 | ||||
| GC30851 | Tecadenoson (CVT-510) | 204512-90-3 | >99.50% | |
An adenosine A 1 receptor agonist | ||||
| GC30916 | PD 117519 (CI947) | 96392-15-3 | >99.50% | |
An adenosine receptor agonist | ||||
| GC30918 | A2A receptor antagonist 1 | 443103-97-7 | >99.50% | |
A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。 | ||||
| GC30987 | A2AR-agonist-1 | 41552-95-8 | >98.00% | |
A2AR-agonist-1是腺苷A2A受体(A2AR)和平衡型核苷转运体1(ENT1)的强效激动剂,其Ki 值分别为 4.39 和 3.47。 | ||||
| GC30993 | AB-MECA | 152918-26-8 | >99.00% | |
An adenosine A 3 receptor agonist | ||||
