5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(481)
- GC10769SB269970 HClCAS: 261901-57-9纯度: >98.50% / >98.00%
SB269970 HCl是一种强效且选择性的5-HT 7 受体拮抗剂，具有高亲和力 (pK i = 8.9)。
- GC10822Clozapine N-oxide (CNO)CAS: 34233-69-7纯度: >98.00%
Clozapine N-oxide（CNO）是一种强效的多巴胺拮抗剂，也是一种选择性肌动蛋白M4受体（EC50=11 nM）激动剂。
- GC10911Venlafaxine hydrochlorideCAS: 99300-78-4纯度: >99.50%
Venlafaxine hydrochloride是一种具有口服活性的5-羟色胺和去甲肾上腺素再摄取抑制剂 （SNRIs; Serotonin-norepinephrine reuptake inhibitors），对配体与人NE和5-HT转运蛋白结合的Ki值分别为2480nM和82nM。
- GC10945TandospironeCAS: 87760-53-0纯度: >99.00%
Tandospirone (SM-3997) 是一种有效的选择性 5-HT1A 受体部分激动剂，Ki 为 27 nM。
- GC11651Ondansetron hydrochloride dihydrateCAS: 103639-04-9纯度: >99.00%
An Analytical Reference Material
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10068 | CP 93129 dihydrochloride | 879089-64-2 | - | |
A 5-HT 1B receptor agonist | ||||
| GC10121 | Tianeptine sodium | 30123-17-2 | >99.50% | |
An atypical antidepressant | ||||
| GC10450 | PRX-08066 | 866206-54-4 | - | |
A 5-HT 2B receptor antagonist | ||||
| GC10460 | Rizatriptan Benzoate | 145202-66-0 | >99.50% | |
A 5-HT 1B and 5-HT 1D receptor agonist | ||||
| GC10614 | Rotigotine | 99755-59-6 | >99.50% | |
A non-selective dopamine receptor agonist | ||||
| GC10769 | SB269970 HCl | 261901-57-9 | >98.50% / >98.00% | |
SB269970 HCl是一种强效且选择性的5-HT 7 受体拮抗剂，具有高亲和力 (pK i = 8.9)。 | ||||
| GC10799 | Iloperidone hydrochloride | 1299470-39-5 | - | |
An atypical antipsychotic | ||||
| GC10822 | Clozapine N-oxide (CNO) | 34233-69-7 | >98.00% | |
Clozapine N-oxide（CNO）是一种强效的多巴胺拮抗剂，也是一种选择性肌动蛋白M4受体（EC50=11 nM）激动剂。 | ||||
| GC10848 | BMY 7378 | 21102-95-4 | - | |
BMY 7378是一种α 1D -肾上腺素能受体（α 1D -AR）的选择性拮抗剂，pk i 值为8.89，也是血清素1A受体（5-HT 1A R）的混合激动剂和拮抗剂。 | ||||
| GC10876 | Vilazodone Hydrochloride | 163521-08-2 | >98.00% | |
An SSRI and a partial agonist of 5-HT 1A | ||||
| GC10911 | Venlafaxine hydrochloride | 99300-78-4 | >99.50% | |
Venlafaxine hydrochloride是一种具有口服活性的5-羟色胺和去甲肾上腺素再摄取抑制剂 （SNRIs; Serotonin-norepinephrine reuptake inhibitors），对配体与人NE和5-HT转运蛋白结合的Ki值分别为2480nM和82nM。 | ||||
| GC10945 | Tandospirone | 87760-53-0 | >99.00% | |
Tandospirone (SM-3997) 是一种有效的选择性 5-HT1A 受体部分激动剂，Ki 为 27 nM。 | ||||
| GC11166 | Alosetron Hydrochloride | 122852-69-1 | >99.50% | |
A 5-HT 3 receptor antagonist | ||||
| GC11517 | SEA0400 | 223104-29-8 | >98.00% | |
A selective inhibitor of the Na + /Ca 2+ exchanger | ||||
| GC11521 | Ziprasidone HCl | 122883-93-6 | - | |
An atypical antipsychotic | ||||
| GC11570 | Desvenlafaxine | 93413-62-8 | - | |
An active metabolite of venlafaxine | ||||
| GC11651 | Ondansetron hydrochloride dihydrate | 103639-04-9 | >99.00% | |
An Analytical Reference Material | ||||
| GC11709 | Fluoxetine HCl | 56296-78-7 | >99.50% | |
An Analytical Reference Material | ||||
| GC11714 | Prucalopride | 179474-81-8 | >99.50% | |
A selective 5-HT 4 receptor agonist | ||||
| GC11824 | Asenapine | 65576-45-6 | >98.50% | |
An atypical antipsychotic | ||||
| GC11959 | Naratriptan | 143388-64-1 | >98.00% | |
A potent 5-HT 1B and 5-HT 1D receptor agonist | ||||
| GC11962 | Lu AE58054 Hydrochloride | 467458-02-2 | >99.50% | |
A 5-HT 6 receptor antagonist | ||||
| GC12091 | SB742457 | 607742-69-8 | >98.00% | |
A 5-HT 6 receptor antagonist | ||||
| GC12495 | Olanzapine | 132539-06-1 | >99.00% / >98.00% / >99.50% | |
Olanzapine是一种单胺拮抗剂。 | ||||