5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(481)
- GC10108WAY-100635CAS: 162760-96-5纯度: >98.00%
WAY-100635是一种具有高效性选择的5-hydroxytryptamine 1A（5-HT1A）受体拮抗剂，IC 50 值为0.91nM，K i 值为0.39nM。
- GC10679DR 4485 hydrochlorideCAS: 402942-53-4
DR4485 (hydrochloride) 是一种具有口服活性的选择性 5-HT7 拮抗剂 (pKi=8.14)。
- GC10698Cyproheptadine hydrochlorideCAS: 969-33-5纯度: >99.50%
An antihistamine with antiserotonergic and anticholinergic activities
- GC11100FlibanserinCAS: 167933-07-5纯度: >99.00%
A 5-HT 1A receptor agonist and 5-HT 2A receptor antagonist
- GC111762-Methyl-5-hydroxytryptamine hydrochlorideCAS: 845861-49-6
2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。
- GC11186BrexpiprazoleCAS: 913611-97-9纯度: >97.00%
Brexpiprazole是一种口服非典型抗精神病药物，是5-HT1A（K i =0.12nM）和dopamine D2L（K i =0.3nM）受体的强效部分激动剂，以及5-HT2A受体（K i =0.47nM）的拮抗剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10051 | MDL 100907 | 139290-65-6 | >98.00% | |
Selective antagonist of the serotonin receptor 5-HT 2A | ||||
| GC10108 | WAY-100635 | 162760-96-5 | >98.00% | |
WAY-100635是一种具有高效性选择的5-hydroxytryptamine 1A（5-HT1A）受体拮抗剂，IC 50 值为0.91nM，K i 值为0.39nM。 | ||||
| GC10117 | Aripiprazole | 129722-12-9 | >99.50% | |
An atypical antipsychotic | ||||
| GC10242 | Loxapine Succinate | 27833-64-3 | >99.50% | |
An atypical antipsychotic drug | ||||
| GC10310 | SB 206553 hydrochloride | 1197334-04-5 | - | |
A 5-HT 2C and 5-HT 2B receptor antagonist | ||||
| GC10357 | Metergoline | 17692-51-2 | >99.50% | |
A serotonin receptor antagonist | ||||
| GC10401 | SB 204070 | 148688-01-1 | - | |
Potent and selective 5-HT4 receptor antagonist | ||||
| GC10495 | EMD 281014 hydrochloride | 443144-27-2 | - | |
5-HT2A antagonist | ||||
| GC10535 | S 32212 hydrochloride | 847871-78-7 | - | |
An inverse agonist of 5-HT 2C receptors | ||||
| GC10674 | LY 266097 hydrochloride | 172895-39-5 | - | |
A 5-HT 2B receptor antagonist | ||||
| GC10679 | DR 4485 hydrochloride | 402942-53-4 | - | |
DR4485 (hydrochloride) 是一种具有口服活性的选择性 5-HT7 拮抗剂 (pKi=8.14)。 | ||||
| GC10698 | Cyproheptadine hydrochloride | 969-33-5 | >99.50% | |
An antihistamine with antiserotonergic and anticholinergic activities | ||||
| GC10743 | Cyclobenzaprine HCl | 6202-23-9 | >99.50% | |
An Analytical Reference Material | ||||
| GC10891 | Alverine Citrate | 5560-59-8 | >99.00% | |
An antispasmodic agent | ||||
| GC10919 | LY 272015 hydrochloride | 172895-15-7 | - | |
A 5-HT 2B receptor antagonist | ||||
| GC10991 | SGS 518 oxalate | 445441-27-0 | - | |
SGS 518 oxalate 是一种选择性 5-HT6R 拮抗剂。 | ||||
| GC11020 | Ziprasidone | 146939-27-7 | >98.00% | |
齐拉西酮 (CP-88059) 是一种口服活性抗精神病药，是一种 5-HT 和多巴胺受体拮抗剂的组合。 | ||||
| GC11033 | Rupatadine Fumarate | 182349-12-8 | >99.50% | |
A histamine H 1 and PAF receptor antagonist | ||||
| GC11100 | Flibanserin | 167933-07-5 | >99.00% | |
A 5-HT 1A receptor agonist and 5-HT 2A receptor antagonist | ||||
| GC11119 | MDL 11,939 | 107703-78-6 | - | |
A potent 5-HT 2A receptor antagonist | ||||
| GC11176 | 2-Methyl-5-hydroxytryptamine hydrochloride | 845861-49-6 | - | |
2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。 | ||||
| GC11186 | Brexpiprazole | 913611-97-9 | >97.00% | |
Brexpiprazole是一种口服非典型抗精神病药物，是5-HT1A（K i =0.12nM）和dopamine D2L（K i =0.3nM）受体的强效部分激动剂，以及5-HT2A受体（K i =0.47nM）的拮抗剂。 | ||||
| GC11191 | Buspirone HCl | 33386-08-2 | >99.50% / >99.00% | |
An Analytical Reference Standard | ||||
| GC11231 | BW 723C86 hydrochloride | 160521-72-2 | - | |
A selective HT2B receptor agonist | ||||