5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(481)
- GC12986RisperidoneCAS: 106266-06-2纯度: >98.00%
Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂,对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。
- GC14518Asenapine hydrochlorideCAS: 1412458-61-7纯度: >99.50%
Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。
- GC15013VilazodoneCAS: 163521-12-8纯度: >99.00%
Vilazodone (EMD 68843; SB 659746A) 是一种强效、选择性和口服活性的血清素再摄取抑制剂 (SSRI) 和部分 5-HT1A 受体激动剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC12541 | Bilobalide | 33570-04-6 | >98.00% | |
A neuroprotective natural product | ||||
| GC12782 | CP-809101 hydrochloride | 1215721-40-6 | >99.50% | |
A potent 5-HT 2C receptor agonist | ||||
| GC12986 | Risperidone | 106266-06-2 | >98.00% | |
Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂,对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。 | ||||
| GC13053 | Pizotifen | 15574-96-6 | >98.00% | |
A triptan | ||||
| GC13081 | Loxapine | 1977-10-2 | >99.50% | |
洛沙平是一种口服活性多巴胺抑制剂、5-HT 受体拮抗剂,也是一种二苯并沙西平抗精神病药物。 | ||||
| GC13092 | Fluvoxamine | 54739-18-3 | - | |
Fluvoxamine是一种选择性血清素(5-HT)再摄取抑制剂(SSRI),具有抗抑郁活性。 | ||||
| GC13428 | Mosapride | 112885-41-3 | - | |
A 5-HT 4 receptor agonist | ||||
| GC13478 | Pizotifen Malate | 5189-11-7 | - | |
A triptan | ||||
| GC13501 | VUF 10166 | 155584-74-0 | - | |
A 5-HT 3 receptor antagonist | ||||
| GC13533 | Cisapride | 81098-60-4 | >99.50% | |
A 5-HT 4 receptor agonist | ||||
| GC13723 | Amitriptyline HCl | 549-18-8 | >99.50% | |
A tricyclic antidepressant | ||||
| GC13871 | Duloxetine HCl | 136434-34-9 | >99.50% | |
A serotonin and norepinephrine reuptake inhibitor | ||||
| GC14160 | Blonanserin | 132810-10-7 | >98.50% | |
A dopamine and serotonin receptor antagonist | ||||
| GC14262 | Desvenlafaxine Succinate | 386750-22-7 | >99.50% | |
An active metabolite of venlafaxine | ||||
| GC14437 | Vortioxetine (Lu AA21004) HBr | 960203-27-4 | >99.50% | |
A multimodal serotonergic agent | ||||
| GC14512 | Fenspiride HCl | 5053-08-7 | >99.50% | |
A histamine H 1 receptor antagonist | ||||
| GC14518 | Asenapine hydrochloride | 1412458-61-7 | >99.50% | |
Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。 | ||||
| GC14550 | SB271046 | 209481-20-9 | - | |
An orally-available 5-HT 6 antagonist | ||||
| GC14563 | Ketanserin | 74050-98-9 | >99.00% / >97.00% | |
A potent 5-HT 2 receptor antagonist | ||||
| GC14788 | Tianeptine | 66981-73-5 | >98.00% | |
An atypical antidepressant | ||||
| GC14927 | Trazodone HCl | 25332-39-2 | >98.00% | |
An Analytical Reference Material | ||||
| GC15013 | Vilazodone | 163521-12-8 | >99.00% | |
Vilazodone (EMD 68843; SB 659746A) 是一种强效、选择性和口服活性的血清素再摄取抑制剂 (SSRI) 和部分 5-HT1A 受体激动剂。 | ||||
| GC15025 | Fluvoxamine maleate | 61718-82-9 | >99.50% | |
A selective serotonin reuptake inhibitor | ||||
| GC15107 | Clomipramine HCl | 17321-77-6 | >99.00% | |
A tricyclic antidepressant | ||||
