GlpBio

Cannabinoid Receptor

Cannabinoid Receptor(大麻素受体)

The cannabinoid receptor (CB1 and CB2) is a member of G-protein coupled receptor which plays a significant role in physiologic processes such as cognitive and immune functions.

Cannabinoid Receptor 相关产品(116)

  • GC10147 structure
    GC10147AM630
    CAS: 164178-33-0
    纯度: >99.50% / >98.00%

    AM630是一种强效且选择性的CB 2 受体反向激动剂。

  • GC10664 structure
    GC10664Org 27569
    CAS: 868273-06-7
    纯度: >99.50%

    Org 27569 是一种有效的 CB1 受体变构调节剂，可增加激动剂的结合，但阻断激动剂诱导的 CB1 信号传导。

  • GC10843 structure
    GC10843Otenabant
    CAS: 686344-29-6
    纯度: >99.00%

    Otenabant 是一种有效的选择性大麻素受体 CB1 拮抗剂，Ki 为 0.7 nM，对人 CB2 受体的选择性高 10,000 倍。

  • GC11376 structure
    GC11376BML-190
    CAS: 2854-32-2
    纯度: >99.00%

    A CB 2 receptor inverse agonist

  • GC11760 structure
    GC11760GW842166X
    CAS: 666260-75-9
    纯度: >99.50%

    A CB 2 receptor agonist

  • GC15414 structure
    GC15414AM1241
    CAS: 444912-48-5

    AM1241是一种氨基烷基吲哚类似物，是II型大麻素受体（CB2）的选择性配体，对CB2受体的亲和力（K i =3.4nM）高于对CB1受体（K i =280nM）。

  • GC15574 structure
    GC15574Taranabant
    CAS: 701977-09-5
    纯度: >99.00%

    A CB 1 receptor inverse agonist

  • GC15717 structure
    GC15717AM251
    CAS: 183232-66-8
    纯度: >98.50%

    AM251是一种 1 型大麻素受体 (CB1) 拮抗剂，IC 50 为8nM，同时也是G蛋白偶联受体55 (GPR55) 激动剂，其EC 50 为39nM。

  • GC16466 structure
    GC16466Rimonabant hydrochloride
    CAS: 158681-13-1
    纯度: >99.00%

    A potent and selective CB 1 receptor antagonist

  • GC17205 structure
    GC17205CP-945598 HCl
    CAS: 686347-12-6

    A selective CB 1 receptor antagonist

  • GC17259 structure
    GC17259Rimonabant
    CAS: 168273-06-1

    A potent and selective CB 1 receptor antagonist

  • GC10028 structure
    GC10028(R)-SLV 319
    CAS: 656827-86-0

    The inactive enantiomer of SLV 319

  • GC10032 structure
    GC10032SR 144528
    CAS: 192703-06-3
    纯度: >99.00% / >98.00%

    SR 144528是一种高效、选择性且具有口服活性的CB2受体拮抗剂，对 CB2 受体的K i 值为0.6nM。

  • GC10205 structure
    GC10205Arvanil
    CAS: 128007-31-8
    纯度: >98.00%

    A structural analog of capsaicin with analgesic activity

  • GC10646 structure
    GC10646TC-C 14G
    CAS: 656804-72-7

    CB1 receptor inverse agonist

  • GC10753 structure
    GC10753(S)-SLV 319
    CAS: 464213-10-3

    A selective antagonist of CB 1

  • GC10907 structure
    GC10907(±)-SLV 319
    CAS: 362519-49-1
    纯度: >99.50%

    A selective antagonist of CB 1

  • GC11453 structure
    GC11453ML-191
    CAS: 931695-79-3

    An antagonist of GPR55

  • GC11849 structure
    GC11849Arachidonyl serotonin
    CAS: 187947-37-1
    纯度: >98.00%

    An inhibitor of FAAH

  • GC12420 structure
    GC12420MAFP
    CAS: 188404-10-6
    纯度: >98.00%

    An inhibitor of MAGL, FAAH, cPLA 2 , and iPLA 2

  • GC12538 structure
    GC12538LH 21
    CAS: 611207-11-5

    Weak CB 1 antagonist

  • GC12868 structure
    GC12868S-2 Methanandamide
    CAS: 157182-48-4

    A potent CB 1 receptor agonist

  • GC12920 structure
    GC12920Pregnenolone
    CAS: 145-13-1
    纯度: >98.00%

    A natural steroid hormone

  • GC12978 structure
    GC12978Tocrifluor T1117
    CAS: 1186195-59-4

    Tocrifluor T1117 (T1117) 是大麻素 CB1 受体拮抗剂 AM251 的荧光形式，是一种选择性荧光 GPR55 配体。