Ras
Ras(Ras蛋白)
Ras belongs to a class of small GTPase and is involved in transmitting signals within cells.
Ras 相关产品(138)
- GC10015Rac1 Inhibitor W56CAS: 1095179-01-3
Rac1 Inhibitor W56 是一种含有 Rac1 残基 45-60 的肽。 Rac1 Inhibitor W56 抑制 Rac1 与鸟嘌呤核苷酸交换因子 TrioN、GEF-H1 和 Tiam 的相互作用。
- GC10069NSC 23766 trihydrochlorideCAS: 1177865-17-6纯度: >99.50% / >99.00%
NSC 23766 trihydrochloride是一种选择性Rac1 GTPase抑制剂,通过特异性阻断Rac1的鸟嘌呤核苷酸交换因子Trio和Tiam1来抑制Rac1的激活,对Rac1的IC₅₀约为50μM。
- GC12247K-Ras(G12C) inhibitor 12CAS: 1469337-95-8纯度: >98.00%
An allosteric inhibitor of oncogenic K-Ras(G12C)
- GC14266CCG 203971CAS: 1443437-74-8纯度: >99.00%
An inhibitor of the Rho/MKL1/SRF transcriptional pathway
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11204 | kobe2602 | 454453-49-7 | >99.50% | |
A selective Ras inhibitor | ||||
| GC16922 | Kobe0065 | 436133-68-5 | >99.50% | |
A selective Ras inhibitor | ||||
| GC19546 | AMG-510 racemate | 2252403-56-6 | >98.00% | |
A covalent inhibitor of K-Ras G12C | ||||
| GC10015 | Rac1 Inhibitor W56 | 1095179-01-3 | - | |
Rac1 Inhibitor W56 是一种含有 Rac1 残基 45-60 的肽。 Rac1 Inhibitor W56 抑制 Rac1 与鸟嘌呤核苷酸交换因子 TrioN、GEF-H1 和 Tiam 的相互作用。 | ||||
| GC10030 | EHop-016 | 1380432-32-5 | >99.00% | |
EHop-016是一种高效的Rac GTP酶Rac1抑制剂,IC 50 值为1.1μM。 | ||||
| GC10069 | NSC 23766 trihydrochloride | 1177865-17-6 | >99.50% / >99.00% | |
NSC 23766 trihydrochloride是一种选择性Rac1 GTPase抑制剂,通过特异性阻断Rac1的鸟嘌呤核苷酸交换因子Trio和Tiam1来抑制Rac1的激活,对Rac1的IC₅₀约为50μM。 | ||||
| GC10265 | Manumycin A | 52665-74-4 | >98.00% | |
A farnesyltransferase inhibitor with antitumor activity | ||||
| GC10528 | Salirasib | 162520-00-5 | >98.00% | |
A Ras inhibitor with anti-cancer and anti-atherogenic activity | ||||
| GC10612 | BQU57 | 1637739-82-2 | >99.50% | |
An inhibitor of RalA and RalB | ||||
| GC10660 | EHT 1864 | 754240-09-0 | >98.00% | |
An inhibitor of Rac GTPases | ||||
| GC10906 | RBC8 | 361185-42-4 | >98.00% | |
A Ral inhibitor | ||||
| GC12060 | Deltarasin hydrochloride | 1440898-82-7 | >99.50% | |
A KRAS inhibitor | ||||
| GC12247 | K-Ras(G12C) inhibitor 12 | 1469337-95-8 | >98.00% | |
An allosteric inhibitor of oncogenic K-Ras(G12C) | ||||
| GC12470 | ZCL278 | 587841-73-4 | >98.00% | |
A selective Cdc42 inhibitor | ||||
| GC12795 | CCG-1423 | 285986-88-1 | >99.50% | |
An inhibitor of Rho-mediated cell signalling | ||||
| GC12948 | CID-1067700 | 314042-01-8 | >98.00% | |
CID-1067700是Rab GTPases的抑制剂,特别是对Rab2和Rab7具有显著的抑制作用。 | ||||
| GC13076 | Deltarasin | 1440898-61-2 | - | |
A KRAS inhibitor | ||||
| GC13315 | ML-098 | 878978-76-8 | >99.50% | |
A selective Rab7 activator | ||||
| GC14266 | CCG 203971 | 1443437-74-8 | >99.00% | |
An inhibitor of the Rho/MKL1/SRF transcriptional pathway | ||||
| GC14800 | ML 141 | 71203-35-5 | >98.50% / >98.00% | |
An allosteric Cdc42 inhibitor | ||||
| GC14860 | Oncrasin 1 | 75629-57-1 | >99.50% | |
An anticancer agent | ||||
| GC15478 | 6H05 | 1469338-01-9 | - | |
An allosteric inhibitor of oncogenic K-Ras(G12C) | ||||
| GC16692 | Casin | 425399-05-9 | >98.00% | |
A Cdc42 GTPase inhibitor | ||||
| GC19037 | ARS-853 | 1629268-00-3 | >98.00% | |
An inhibitor of KRAS G12C | ||||
