GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC10756[Arg14,Lys15]NociceptinCAS: 236098-40-1
[Arg14,Lys15]Nociceptin 是一种高效的选择性 NOP 受体 (ORL1; OP4) 激动剂，EC50 为 1 nM。
- GC10818Oxprenolol hydrochlorideCAS: 6452-73-9纯度: >98.00%
A non-selective β-adrenergic receptor antagonist
- GC10862Galanin (1-30) (human)CAS: 119418-04-1纯度: >98.00%
Galanin (1-30) (human) 是一种 30 个氨基酸的神经肽，作为\u200b\u200b GalR1 和 GalR2 受体的激动剂，Kis 均为 1 nM。
- GC10863Otilonium BromideCAS: 26095-59-0纯度: >99.00%
An L- and T-type calcium channel inhibitor and mAChR antagonist
- GC10927CGRP 8-37 (rat)CAS: 129121-73-9纯度: >98.50%
CGRP 8-37 (rat) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) 是一种高度选择性的 CGRP 受体拮抗剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10738 | Brimonidine Tartrate | 70359-46-5 | >99.00% | |
An α 2 -adrenergic receptor agonist | ||||
| GC10743 | Cyclobenzaprine HCl | 6202-23-9 | >99.50% | |
An Analytical Reference Material | ||||
| GC10747 | HS 024 | 212370-59-7 | - | |
HS 024 是一种选择性 MC4 受体拮抗剂，对 MC4、MC5、MC3 和 MC1 的 Kis 分别为 0.29、3.29、5.45 和 18.6 nM。 | ||||
| GC10753 | (S)-SLV 319 | 464213-10-3 | - | |
A selective antagonist of CB 1 | ||||
| GC10756 | [Arg14,Lys15]Nociceptin | 236098-40-1 | - | |
[Arg14,Lys15]Nociceptin 是一种高效的选择性 NOP 受体 (ORL1; OP4) 激动剂，EC50 为 1 nM。 | ||||
| GC10771 | CJ-023423 | 415903-37-6 | >99.00% | |
An EP 4 receptor antagonist | ||||
| GC10777 | Cortistatin-8 | 485803-62-1 | - | |
ghrelin receptor antagonist | ||||
| GC10790 | FSLLRY-NH2 | 245329-02-6 | - | |
FSLLRY-NH2是蛋白酶激活受体2（PAR-2）的拮抗剂。 | ||||
| GC10818 | Oxprenolol hydrochloride | 6452-73-9 | >98.00% | |
A non-selective β-adrenergic receptor antagonist | ||||
| GC10821 | 11-keto-β-Boswellic Acid | 17019-92-0 | >99.50% | |
A 5-LO inhibitor | ||||
| GC10826 | PIT | 56583-49-4 | - | |
Purinergic P2Y receptor ligand | ||||
| GC10862 | Galanin (1-30) (human) | 119418-04-1 | >98.00% | |
Galanin (1-30) (human) 是一种 30 个氨基酸的神经肽，作为\u200b\u200b GalR1 和 GalR2 受体的激动剂，Kis 均为 1 nM。 | ||||
| GC10863 | Otilonium Bromide | 26095-59-0 | >99.00% | |
An L- and T-type calcium channel inhibitor and mAChR antagonist | ||||
| GC10865 | TC-MCH 7c | 864756-35-4 | >99.00% | |
TC-MCH 7c 是一种苯基吡啶酮衍生物，是一种口服的、选择性的、可穿透脑的 MCH1R 拮抗剂，对 hMCH1R 的 IC50 为 5.6 nM。 | ||||
| GC10887 | Labetalol HCl | 32780-64-6 | >99.50% | |
An antagonist of α- and β-adrenoreceptors | ||||
| GC10891 | Alverine Citrate | 5560-59-8 | >99.00% | |
An antispasmodic agent | ||||
| GC10903 | YIL 781 | 875258-85-8 | >98.00% / >97.00% | |
YIL 781是一种选择性的胃饥饿素受体（GHSR1a）拮抗剂，K i 值为17nM。 | ||||
| GC10906 | RBC8 | 361185-42-4 | >98.00% | |
A Ral inhibitor | ||||
| GC10907 | (±)-SLV 319 | 362519-49-1 | >99.50% | |
A selective antagonist of CB 1 | ||||
| GC10919 | LY 272015 hydrochloride | 172895-15-7 | - | |
A 5-HT 2B receptor antagonist | ||||
| GC10927 | CGRP 8-37 (rat) | 129121-73-9 | >98.50% | |
CGRP 8-37 (rat) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) 是一种高度选择性的 CGRP 受体拮抗剂。 | ||||
| GC10935 | EHNA hydrochloride | 58337-38-5 | >95.00% | |
A dual inhibitor of PDE2 and ADA | ||||
| GC10937 | FR 171113 | 173904-50-2 | - | |
FR171113 是一种特异性的非肽类凝血酶受体拮抗剂。 | ||||
| GC10942 | NNC 63-0532 | 250685-44-0 | - | |
NOP receptor agonist | ||||