GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC10960[Ala2,8,9,11,19,22,24,25,27,28]-VIPCAS: 866552-34-3
Highly selective agonist for the VPAC1 receptor
- GC10972Gallamine TriethiodideCAS: 65-29-2纯度: >98.00%
An allosteric modulator of muscarinic acetylcholine receptors
- GC10976Noradrenaline bitartrate monohydrateCAS: 108341-18-0纯度: >99.50%
Noradrenaline bitartrate monohydrate是一种β1选择性肾上腺素受体激动剂，EC 50 值为5.37μM。
- GC110025'-(N-Cyclopropyl)carboxamidoadenosineCAS: 50908-62-8
A specific adenosine A 2 receptor agonist
- GC11012Proglumide sodium saltCAS: 99247-33-3纯度: >99.50%
Proglumide sodium salt 是一种非肽类和具有口服活性的胆囊收缩素 (CCK)-A/B 受体拮抗剂。
- GC11026RS 102895 hydrochlorideCAS: 1173022-16-6纯度: >98.00%
RS 102895 hydrochloride是一种有效的CCR2抑制剂，IC 50 值为0.36μM。
- GC11067PF 04418948CAS: 1078166-57-0纯度: >98.50%
PF 04418948是一种具有口服活性、强效且选择性的前列腺素EP2受体拮抗剂，IC 50 值为16nM。
- GC11074BIBP 3226 trifluoroacetateCAS: 1068148-47-9纯度: >98.00%
BIBP 3226 trifluoroacetate是一种强效的非肽类neuropeptide Y (NPY) Y1 受体拮抗剂，对rNPY Y1、hNPFF2和rNPFF的K i 值分别为1.1、79和108nM。
- GC11100FlibanserinCAS: 167933-07-5纯度: >99.00%
A 5-HT 1A receptor agonist and 5-HT 2A receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10947 | [D-Trp8]-γ-MSH | 321351-81-9 | - | |
An MC3R agonist | ||||
| GC10960 | [Ala2,8,9,11,19,22,24,25,27,28]-VIP | 866552-34-3 | - | |
Highly selective agonist for the VPAC1 receptor | ||||
| GC10961 | Apelin-17 (human, bovine) | 217082-57-0 | >98.50% | |
Apelin-17（人，牛）是一种内源性孤儿 G 蛋白偶联受体 APJ 激动剂。 | ||||
| GC10965 | ARC 239 dihydrochloride | 55974-42-0 | - | |
An α2B-adrenergic receptor antagonist | ||||
| GC10972 | Gallamine Triethiodide | 65-29-2 | >98.00% | |
An allosteric modulator of muscarinic acetylcholine receptors | ||||
| GC10976 | Noradrenaline bitartrate monohydrate | 108341-18-0 | >99.50% | |
Noradrenaline bitartrate monohydrate是一种β1选择性肾上腺素受体激动剂，EC 50 值为5.37μM。 | ||||
| GC10991 | SGS 518 oxalate | 445441-27-0 | - | |
SGS 518 oxalate 是一种选择性 5-HT6R 拮抗剂。 | ||||
| GC10992 | LY 255283 | 117690-79-6 | >98.50% | |
A BLT 2 receptor antagonist | ||||
| GC10994 | ATC 0065 | 510732-84-0 | - | |
MCH1 antagonist,potent and selective | ||||
| GC11002 | 5'-(N-Cyclopropyl)carboxamidoadenosine | 50908-62-8 | - | |
A specific adenosine A 2 receptor agonist | ||||
| GC11004 | A 779 | 159432-28-7 | >98.00% | |
A 779是一种有效的选择性血管紧张素-(1-7)/ Mas受体拮抗剂，IC 50 值为0.3nM。 | ||||
| GC11012 | Proglumide sodium salt | 99247-33-3 | >99.50% | |
Proglumide sodium salt 是一种非肽类和具有口服活性的胆囊收缩素 (CCK)-A/B 受体拮抗剂。 | ||||
| GC11017 | ZM 241385 | 139180-30-6 | >99.00% | |
An A 2A adenosine receptor antagonist | ||||
| GC11020 | Ziprasidone | 146939-27-7 | >98.00% | |
齐拉西酮 (CP-88059) 是一种口服活性抗精神病药，是一种 5-HT 和多巴胺受体拮抗剂的组合。 | ||||
| GC11026 | RS 102895 hydrochloride | 1173022-16-6 | >98.00% | |
RS 102895 hydrochloride是一种有效的CCR2抑制剂，IC 50 值为0.36μM。 | ||||
| GC11033 | Rupatadine Fumarate | 182349-12-8 | >99.50% | |
A histamine H 1 and PAF receptor antagonist | ||||
| GC11035 | Hyoscyamine | 101-31-5 | >98.00% | |
A muscarinic receptor antagonist | ||||
| GC11042 | WAY 267464 dihydrochloride | 847375-16-0 | - | |
WAY 267464 dihydrochloride 是一种非肽催产素受体 (OTR) 激动剂。 | ||||
| GC11067 | PF 04418948 | 1078166-57-0 | >98.50% | |
PF 04418948是一种具有口服活性、强效且选择性的前列腺素EP2受体拮抗剂，IC 50 值为16nM。 | ||||
| GC11074 | BIBP 3226 trifluoroacetate | 1068148-47-9 | >98.00% | |
BIBP 3226 trifluoroacetate是一种强效的非肽类neuropeptide Y (NPY) Y1 受体拮抗剂，对rNPY Y1、hNPFF2和rNPFF的K i 值分别为1.1、79和108nM。 | ||||
| GC11077 | Imiloxan hydrochloride | 81167-22-8 | >98.00% | |
α2-adrenoceptor antagonist | ||||
| GC11100 | Flibanserin | 167933-07-5 | >99.00% | |
A 5-HT 1A receptor agonist and 5-HT 2A receptor antagonist | ||||
| GC11112 | 2'-MeCCPA | 205171-12-6 | - | |
An adenosine A 1 receptor agonist | ||||
| GC11119 | MDL 11,939 | 107703-78-6 | - | |
A potent 5-HT 2A receptor antagonist | ||||