GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC11161C 021 dihydrochlorideCAS: 864289-85-0纯度: >98.00%
C 021 dihydrochloride 是一种有效的 CC 趋化因子受体 4 (CCR4) 拮抗剂。
- GC111762-Methyl-5-hydroxytryptamine hydrochlorideCAS: 845861-49-6
2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。
- GC11186BrexpiprazoleCAS: 913611-97-9纯度: >97.00%
Brexpiprazole是一种口服非典型抗精神病药物，是5-HT1A（K i =0.12nM）和dopamine D2L（K i =0.3nM）受体的强效部分激动剂，以及5-HT2A受体（K i =0.47nM）的拮抗剂。
- GC11219(R)-(+)-TolterodineCAS: 124937-51-5纯度: >99.50%
(R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂，在体内对膀胱的选择性优于唾液腺。
- GC11227[D-Trp34]-Neuropeptide YCAS: 153549-84-9
[D-Trp34]-Neuropeptide Y 是一种有效的选择性神经肽 Y (NPY) Y5 受体激动剂。
- GC11311MRS 2179 tetrasodium saltCAS: 1454889-37-2
MRS 2179 tetrasodium salt 是一种竞争性 P2Y1 受体拮抗剂，对火鸡 P2Y1 受体的 Kb 值为 102 nM，pA2 值为 6.99。
- GC11314Atrial natriuretic factor (1-28) (rat)CAS: 88898-17-3
Atrial natriuretic factor (1-28) (rat) 是大鼠体内 ANP 的主要循环形式，以浓度依赖性方式有效抑制血管紧张素 II (Ang II) 刺激的 endothelin-1 分泌。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11122 | TCS 2510 | 346673-06-1 | >98.00% | |
Agonist of the PGE 2 receptor EP 4 | ||||
| GC11130 | Indacaterol Maleate | 753498-25-8 | >98.00% | |
A long-acting β 2 -adrenergic receptor agonist | ||||
| GC11131 | CART (55-102) (rat) | 209615-79-2 | - | |
CART (55-102) (rat) 是一种具有有效抑制食欲活性的大鼠饱腹感因子。 | ||||
| GC11133 | 16,16-Dimethyl Prostaglandin E2 | 39746-25-3 | - | |
derivative of prostaglandin E2 | ||||
| GC11161 | C 021 dihydrochloride | 864289-85-0 | >98.00% | |
C 021 dihydrochloride 是一种有效的 CC 趋化因子受体 4 (CCR4) 拮抗剂。 | ||||
| GC11174 | ZD 2079 | 178600-17-4 | - | |
ZD 2079 (ZD2079 hydrochloride) 是一种有效的 β3-adrenoceptor 激动剂，对去氧肾上腺素预收缩的大鼠肠系膜动脉的 pD2 为 3.72。 | ||||
| GC11176 | 2-Methyl-5-hydroxytryptamine hydrochloride | 845861-49-6 | - | |
2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。 | ||||
| GC11182 | LY404039 | 635318-11-5 | >98.00% | |
An agonist of mGluR2 and mGluR3 | ||||
| GC11186 | Brexpiprazole | 913611-97-9 | >97.00% | |
Brexpiprazole是一种口服非典型抗精神病药物，是5-HT1A（K i =0.12nM）和dopamine D2L（K i =0.3nM）受体的强效部分激动剂，以及5-HT2A受体（K i =0.47nM）的拮抗剂。 | ||||
| GC11188 | GR 135531 | 190277-13-5 | - | |
MT3 receptor agonist | ||||
| GC11191 | Buspirone HCl | 33386-08-2 | >99.50% / >99.00% | |
An Analytical Reference Standard | ||||
| GC11201 | ARM1 | 68729-05-5 | - | |
An inhibitor of LTA 4 hydrolase | ||||
| GC11219 | (R)-(+)-Tolterodine | 124937-51-5 | >99.50% | |
(R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂，在体内对膀胱的选择性优于唾液腺。 | ||||
| GC11227 | [D-Trp34]-Neuropeptide Y | 153549-84-9 | - | |
[D-Trp34]-Neuropeptide Y 是一种有效的选择性神经肽 Y (NPY) Y5 受体激动剂。 | ||||
| GC11231 | BW 723C86 hydrochloride | 160521-72-2 | - | |
A selective HT2B receptor agonist | ||||
| GC11239 | Midodrine (hydrochloride) | 43218-56-0 | >99.00% | |
A prodrug form of desglymidodrine | ||||
| GC11257 | Fluocinolone Acetonide | 67-73-2 | >99.50% | |
A synthetic corticosteroid | ||||
| GC11278 | Boc-MLF | 67247-12-5 | - | |
formyl peptide receptor 1 (FPR1) antagonist | ||||
| GC11283 | FPL 55712 | 40785-97-5 | - | |
A leukotriene receptor antagonist | ||||
| GC11288 | 2-Phenylmelatonin | 151889-03-1 | - | |
A MT receptor mixed partial agonist and antagonist | ||||
| GC11305 | LY 225910 | 133040-77-4 | - | |
LY 225910是一种有效的胆囊收缩素受体拮抗剂，可特异性阻断CCK2受体并影响神经递质释放 | ||||
| GC11308 | L-703,664 succinate | 144776-01-2 | - | |
5-HT1D receptor agonist | ||||
| GC11311 | MRS 2179 tetrasodium salt | 1454889-37-2 | - | |
MRS 2179 tetrasodium salt 是一种竞争性 P2Y1 受体拮抗剂，对火鸡 P2Y1 受体的 Kb 值为 102 nM，pA2 值为 6.99。 | ||||
| GC11314 | Atrial natriuretic factor (1-28) (rat) | 88898-17-3 | - | |
Atrial natriuretic factor (1-28) (rat) 是大鼠体内 ANP 的主要循环形式，以浓度依赖性方式有效抑制血管紧张素 II (Ang II) 刺激的 endothelin-1 分泌。 | ||||