GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC13549Setiptiline maleateCAS: 85650-57-3纯度: >98.00%
Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。
- GC13618TarafenacinCAS: 385367-47-5
Tarafenacin(SVT-40776) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM)，选择性比 M2 受体高约 200 倍。
- GC13638Betamethasone ValerateCAS: 2152-44-5纯度: >99.00%
A glucocorticoid with anti-inflammatory activity
- GC13652DyphyllineCAS: 479-18-5纯度: >99.00%
An adenosine receptor antagonist and phosphodiesterase inhibitor
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13549 | Setiptiline maleate | 85650-57-3 | >98.00% | |
Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。 | ||||
| GC13552 | UK 14,304 | 59803-98-4 | >99.50% | |
An α 2 -adrenergic receptor agonist | ||||
| GC13565 | SHU 9119 | 168482-23-3 | >98.00% | |
An MC1R agonist and MC4R antagonist | ||||
| GC13583 | CJ 033466 | 519148-48-2 | - | |
CJ 033466 是一种新型选择性 5-HT4 受体部分激动剂，EC50 为 9 nM，具有促胃动力作用。 | ||||
| GC13588 | 5-OMe-UDP trisodium salt | 1207530-98-0 | - | |
Potent P2Y6 agonist | ||||
| GC13597 | Pyrrolidino PAF C-16 | 91021-63-5 | - | |
A potent analog of PAF C-16 | ||||
| GC13605 | S-1 Methanandamide | 157182-50-8 | - | |
A CB 1 receptor ligand | ||||
| GC13607 | LY 215840 | 137328-52-0 | - | |
5-HT2/5-HT7 receptor antagonist | ||||
| GC13609 | L-670,596 | 121083-05-4 | - | |
thromboxane A2/prostaglandin endoperoxide receptor antagonist | ||||
| GC13610 | [Sar9,Met(O2)11]-Substance P | 110880-55-2 | - | |
A peptide NK 1 receptor agonist | ||||
| GC13618 | Tarafenacin | 385367-47-5 | - | |
Tarafenacin(SVT-40776) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM)，选择性比 M2 受体高约 200 倍。 | ||||
| GC13623 | SDZ 21009 | 39731-05-0 | - | |
β-adrenoceptor and 5-HT1A/1B receptor antagonist | ||||
| GC13627 | Ziprasidone hydrochloride monohydrate | 138982-67-9 | >99.50% | |
An atypical antipsychotic | ||||
| GC13638 | Betamethasone Valerate | 2152-44-5 | >99.00% | |
A glucocorticoid with anti-inflammatory activity | ||||
| GC13652 | Dyphylline | 479-18-5 | >99.00% | |
An adenosine receptor antagonist and phosphodiesterase inhibitor | ||||
| GC13654 | Alosetron | 122852-42-0 | - | |
A 5-HT 3 receptor antagonist | ||||
| GC13660 | JD5037 | 1392116-14-1 | >98.00% | |
JD5037 是一种有效的 CB1R 拮抗剂，IC50 为 1.5 nM。 | ||||
| GC13666 | Bay 55-9837 | 463930-25-8 | - | |
Bay 55-9837 是一种有效且高度选择性的 VPAC2 激动剂，Kd 为 0.65 nM。 | ||||
| GC13674 | Talopram hydrochloride | 7013-41-4 | - | |
noradrenalin transporter (NET) inhibitor | ||||
| GC13686 | CH 275 | 174688-78-9 | - | |
CH 275 是生长抑素的肽类似物，优选与生长抑素受体 1 (sst1) 结合，Ki 为 52 nM。 | ||||
| GC13695 | 2-PMDQ | 139047-55-5 | - | |
α1-adrenoceptor antagonist | ||||
| GC13712 | FTY720 Phosphate | 402615-91-2 | - | |
The active metabolite of FTY720 | ||||
| GC13720 | TY 52156 | 934369-14-9 | >99.50% | |
A S1P 3 receptor antagonist | ||||
| GC13732 | TG4-155 | 1164462-05-8 | >99.50% | |
A brain penetrant EP 2 antagonist | ||||