GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC50245(+/-)-ADX 71743CAS: 1431641-29-0
Negative allosteric modulator of mGlu7 receptors; brain penetrant
- GC50246TASP 0390325CAS: 1642187-96-9纯度: >98.00%
TASP 0390325 是一种高亲和力和口服活性精氨酸加压素受体 1B（V1B 受体）拮抗剂，具有抗抑郁和抗焦虑活性。
- GC50278[Pro3]-GIP (Mouse)
[Pro3]-GIP (Mouse)是一种高效的酶抵抗型gastric inhibitory polypeptide (GIP)受体拮抗剂，IC 50 值为2.6μM。
- GC50351KRH 3955 hydrochlorideCAS: 2253744-59-9
Highly potent CXCR4 antagonist; inhibits HIV-1 replication
- GC503548-Cyclopentyl-1,3-dimethylxanthineCAS: 35873-49-5纯度: >98.00%
An adenosine A 1 receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC50229 | VUF 11222 | 1414376-84-3 | - | |
High affinity non-peptide CXCR3 agonist | ||||
| GC50230 | SB 332235 | 276702-15-9 | - | |
A CXCR2 antagonist | ||||
| GC50240 | AMG 853 | 1169483-24-2 | >98.00% | |
AMG 853 (AMG 853) 是一种苯乙酸衍生物。 | ||||
| GC50245 | (+/-)-ADX 71743 | 1431641-29-0 | - | |
Negative allosteric modulator of mGlu7 receptors; brain penetrant | ||||
| GC50246 | TASP 0390325 | 1642187-96-9 | >98.00% | |
TASP 0390325 是一种高亲和力和口服活性精氨酸加压素受体 1B（V1B 受体）拮抗剂，具有抗抑郁和抗焦虑活性。 | ||||
| GC50247 | A 127722 | 195704-72-4 | - | |
Highly potent, selective ETA antagonist; orally bioavailable | ||||
| GC50253 | PF 543 hydrochloride | 1706522-79-3 | >98.00% | |
A potent inhibitor of SPHK1 | ||||
| GC50258 | (R)-Citalopram oxalate | 219861-53-7 | - | |
Enantiomer of escitalopram oxalate | ||||
| GC50271 | SCH 336 | 447459-51-0 | - | |
SCH 336 是一种有效的、选择性的、反向的和口服活性的 CB2 激动剂。 | ||||
| GC50273 | LEI 101 hydrochloride | - | - | |
Potent and selective CB2 partial agonist; orally biovailable | ||||
| GC50275 | Ex 26 | 1233332-37-0 | - | |
Ex 26 (S1P1-IN-Ex 26) 是一种有效的选择性 1-磷酸鞘氨醇受体 1 (S1P1) 拮抗剂 (IC50\u003d0.93 nM)。 | ||||
| GC50277 | [Pro3]-GIP (Rat) | - | - | |
High affinity rat GIP partial agonist | ||||
| GC50278 | [Pro3]-GIP (Mouse) | - | - | |
[Pro3]-GIP (Mouse)是一种高效的酶抵抗型gastric inhibitory polypeptide (GIP)受体拮抗剂，IC 50 值为2.6μM。 | ||||
| GC50286 | Neuropeptide S (Mouse) | 412938-74-0 | - | |
Neuropeptide S (Mouse) 是一种生物活性肽。 | ||||
| GC50293 | CATPB | 1322598-09-3 | >98.00% | |
CATPB 是一种有效的选择性游离脂肪酸受体 2 (FFA2R/GPR43) 拮抗剂。 | ||||
| GC50303 | MSG 606 | 1416983-77-1 | - | |
MSG-606 对人黑皮质素 1 受体 (hMC1R) 具有强效拮抗活性和受体选择性（IC50 = 17 nM）。 | ||||
| GC50310 | MM 54 | 1313027-43-8 | - | |
MM 54 (compound 5) 是 APJ 的竞争性拮抗剂，IC50 为 93 nM。 MM 54 作为 apelin 结合和 APLNR 激活的有效和选择性抑制剂。 | ||||
| GC50313 | ZQ 16 | 376616-73-8 | - | |
Selective GPR84 agonist | ||||
| GC50333 | AMG 837 hemicalcium salt | 1291087-14-3 | - | |
An FFAR1 (GPR40) partial | ||||
| GC50336 | SHIP 2a | 2165706-30-7 | >99.00% | |
SHIP 2a 是一种选择性胱硫醚 γ-裂解酶 (CSE) 酶抑制剂，IC50 为 6.3 μM。 | ||||
| GC50351 | KRH 3955 hydrochloride | 2253744-59-9 | - | |
Highly potent CXCR4 antagonist; inhibits HIV-1 replication | ||||
| GC50354 | 8-Cyclopentyl-1,3-dimethylxanthine | 35873-49-5 | >98.00% | |
An adenosine A 1 receptor antagonist | ||||
| GC50365 | AC 265347 | 1253901-26-6 | >99.00% | |
A calcimimetic and positive allosteric modulator of CaSR | ||||
| GC50373 | Retrobradykinin | 5991-13-9 | - | |
逆缓激肽具有与缓激肽相反的序列。 | ||||