GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC15829Urapidil HClCAS: 64887-14-5纯度: >99.00%
An α 1 -AR antagonist and 5-HT 1A receptor partial agonist
- GC16004NE 100 hydrochlorideCAS: 149409-57-4纯度: >98.00%
NE 100 hydrochloride是一种选择性sigma-1受体（IC 50 =4.16nM）拮抗剂。
- GC16029Granisetron HClCAS: 107007-99-8纯度: >99.50%
A 5-HT 3 receptor antagonist with antiemetic activity
- GC16100SCH 527123CAS: 473727-83-2纯度: >99.00%
SCH 527123是一种强效、选择性的CXCR1和CXCR2受体拮抗剂，对小鼠（K d =0.20nM）、大鼠（K d =0.20nM）和食蟹猴（K d =0.08nM）的CXCR2受体具有高亲和力。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15690 | Desonide | 638-94-8 | >99.00% | |
A nonfluorinated synthetic corticosteroid | ||||
| GC15694 | VPC 23019 | 449173-19-7 | >99.50% | |
A sphingosine-1-phosphate receptor antagonist | ||||
| GC15698 | Epinephrine HCl | 55-31-2 | - | |
An adrenergic receptor agonist | ||||
| GC15717 | AM251 | 183232-66-8 | >98.50% | |
AM251是一种 1 型大麻素受体 (CB1) 拮抗剂，IC 50 为8nM，同时也是G蛋白偶联受体55 (GPR55) 激动剂，其EC 50 为39nM。 | ||||
| GC15719 | Silodosin | 160970-54-7 | >99.50% | |
A potent α 1A -adrenoceptor antagonist | ||||
| GC15754 | WAY-100635 Maleate | 1092679-51-0 | >99.00% | |
A serotonin 5-HT 1A antagonist | ||||
| GC15808 | TC LPA5 4 | 1393814-38-4 | - | |
TC LPA5 4是一种强效的LPA5选择性受体拮抗剂和heparanase（乙酰肝素酶）抑制剂，IC 50 值分别为0.8μM和10μM。 | ||||
| GC15829 | Urapidil HCl | 64887-14-5 | >99.00% | |
An α 1 -AR antagonist and 5-HT 1A receptor partial agonist | ||||
| GC15838 | BD 1063 dihydrochloride | 206996-13-6 | >98.00% | |
An antagonist of σ 1 receptors | ||||
| GC15839 | Zafirlukast | 107753-78-6 | >99.50% | |
A selective CysLT 1 receptor antagonist | ||||
| GC15903 | CYM 50308 | 1345858-76-5 | >98.00% | |
A selective S1P 4 receptor agonist | ||||
| GC15908 | AM-095 free base | 1228690-36-5 | >99.00% | |
A selective LPA 1 receptor antagonist | ||||
| GC15918 | Formoterol Hemifumarate | 43229-80-7 | >98.50% | |
强效、选择性和长效 β2-肾上腺素能受体激动剂 | ||||
| GC15926 | BAN ORL 24 | 475150-69-7 | >98.00% | |
A nociceptin receptor antagonist | ||||
| GC15973 | Tozadenant | 870070-55-6 | >99.50% | |
An adenosine A 2A receptor antagonist | ||||
| GC15989 | WZ811 | 55778-02-4 | >98.00% | |
CXCR4 antagonist | ||||
| GC16004 | NE 100 hydrochloride | 149409-57-4 | >98.00% | |
NE 100 hydrochloride是一种选择性sigma-1受体（IC 50 =4.16nM）拮抗剂。 | ||||
| GC16017 | Rotigotine hydrochloride | 125572-93-2 | >99.00% | |
A non-selective dopamine receptor agonist | ||||
| GC16026 | Talnetant | 174636-32-9 | >99.00% | |
A nonpeptide NK 3 antagonist | ||||
| GC16029 | Granisetron HCl | 107007-99-8 | >99.50% | |
A 5-HT 3 receptor antagonist with antiemetic activity | ||||
| GC16100 | SCH 527123 | 473727-83-2 | >99.00% | |
SCH 527123是一种强效、选择性的CXCR1和CXCR2受体拮抗剂，对小鼠（K d =0.20nM）、大鼠（K d =0.20nM）和食蟹猴（K d =0.08nM）的CXCR2受体具有高亲和力。 | ||||
| GC16142 | Ondansetron | 99614-02-5 | >99.00% | |
A Certified Reference Material | ||||
| GC16176 | GSK 137647 | 349085-82-1 | >99.50% | |
A selective GPR120 agonist | ||||
| GC16226 | BRL-15572 dihydrochloride | 193611-72-2 | >99.00% | |
A 5-HT 1D receptor antagonist | ||||