GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(481)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(404)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(116)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(78)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(78)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(95)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(5)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
-
GC14818
Bisoprolol fumarate
比索洛尔富马酸盐
A β1-AR antagonist
-
GC14563
Ketanserin
酮色林; R41468
A potent 5-HT2 receptor antagonist
-
GC11191
Buspirone HCl
盐酸丁螺环酮
An Analytical Reference Standard
-
GC10434
Triamcinolone
曲安西龙
A synthetic glucocorticoid
-
GC17974
Latrepirdine dihydrochloride
2,3,4,5-四氢-2,8-二甲基-5-[2-(6-甲基-3-吡啶基)乙基]-1H-吡啶并[4,3-B]吲哚二盐酸盐,Dimebolin dihydrochloride
A neuroprotective agent
-
GC17061
Dapoxetine HCl
盐酸达泊西汀; LY-210448 hydrochloride
An Analytical Reference Standard
-
GC15829
Urapidil HCl
盐酸乌拉地尔
An α1-AR antagonist and 5-HT1A receptor partial agonist
-
GC12376
Maprotiline HCl
盐酸马普替林
A tricyclic antidepressant
-
GC13993
Terazosin HCl
盐酸特拉唑嗪(二水合物)
A potent and selective α1-AR antagonist
-
GC15107
Clomipramine HCl
盐酸氯米帕明; Chlorimipramine hydrochloride; G-34586 hydrochloride; NSC-169865 hydrochloride
A tricyclic antidepressant
-
GC13134
Tiotropium Bromide hydrate
噻托溴铵一水合物,BA-679 BR (hydrate)
A muscarinic receptor antagonist
-
GC14927
Trazodone HCl
盐酸曲唑酮; AF-1161
An Analytical Reference Material
-
GC17367
Rebamipide
瑞巴派特; OPC12759; Proamipide
A gastroprotective agent and mucin secretagogue
-
GC14021
Betaxolol
倍他洛尔
An Analytical Reference Standard
-
GC17825
Methscopolamine
甲溴东莨菪碱
A muscarinic acetylcholine receptor antagonist
-
GC12724
Phenoxybenzamine HCl
盐酸酚苄明
An α-AR antagonist
-
GC16142
Ondansetron
昂丹司琼; GR 38032; SN 307
A Certified Reference Material
-
GC15153
Almotriptan Malate
马来酸阿莫曲坦; PNU180638
An agonist of 5-HT1B and 5-HT1D receptors
-
GC15063
Ritodrine HCl
盐酸利托君; DU21220 hydrochloride
A β2-AR agonist
-
GC15150
Tropicamide
托吡卡胺; Ro 1-7683
A selective muscarinic M4 antagonist
-
GC15687
Azasetron HCl
盐酸阿扎司琼; Y-25130 hydrochloride
A 5-HT3 receptor antagonist
-
GC16291
Phentolamine Mesylate
甲磺酸酚妥拉明; Phentolamine methanesulfonate
A reversible α-adrenergic receptor antagonist
-
GC11447
Mirtazapine
米氮平
Mirtazapine是一种去甲肾上腺素能和特异性血清素抗抑郁药(NaSSA),可抑制5-HT2A、5-HT2B、5-HT2C和5-HT3受体,pKi值分别为8.2、6.7、7.9和8.1。
-
GC14216
Chlorpromazine HCl
盐酸氯丙嗪
Chlorpromazine HCl是一种口服有效的、可透过血脑屏障的吩噻嗪类抗精神病药,能够有效抑制D2多巴胺受体和5-HT2A,具有很强的镇静作用。
-
GC11343
Propranolol HCl
盐酸普萘洛尔
A β-adrenergic receptor antagonist
-
GC10738
Brimonidine Tartrate
酒石酸溴莫尼定; UK 14304 tartrate; AGN190342 tartrate
An α2-adrenergic receptor agonist
-
GC14988
Naphazoline HCl
盐酸萘甲唑啉; Naphthazoline hydrochloride
A vasoconstrictor
-
GC13974
Salbutamol Sulfate
沙丁胺醇半硫酸盐; Albuterol hemisulfate; AH-3365 hemisulfate
A β2-AR agonist
-
GC10750
Dexmedetomidine HCl
盐酸右美托咪定; (+)-Medetomidine hydrochloride; (S)-Medetomidine hydrochloride
An α2-adrenoceptor agonist
-
GC12403
Ozagrel HCl
盐酸奥扎格雷,OKY-046 hydrochloride
A selective inhibitor of TXA synthase
-
GC13173
Sotalol
索他洛尔,(R)-Sotalol
An Analytical Reference Standard
-
GC17296
Xylazine HCl
盐酸甲苯噻嗪,BAY 1470 hydrochloride
An α2-adrenergic receptor agonist
-
GC11029
Isoprenaline HCl
盐酸异丙肾上腺素; Isoproterenol hydrochloride
A β1- and β2-AR agonist
-
GC12231
Sulfisoxazole
磺胺异恶唑; Sulfafurazole
An antibiotic and endothelin receptor antagonist
-
GC15243
Carbazochrome sodium sulfonate (AC-17)
卡络磺钠; AC-17
Carbazochrome sodium sulfonate (AC-17) (AC-17) 是一种毛细血管稳定剂,用于研究出血。
-
GC14536
Metoprolol Tartrate
酒石酸美托洛尔
An Analytical Reference Standard
-
GC11479
Xylometazoline HCl
盐酸赛洛唑啉
An α-adrenergic receptor agonist
-
GC15754
WAY-100635 Maleate
A serotonin 5-HT1A antagonist
-
GC13501
VUF 10166
A 5-HT3 receptor antagonist
-
GC13281
VU 0364770
An mGluR4 and mGluR6 positive allosteric modulator and mGluR5 antagonist
-
GC13962
VU 0361737
ML-128
A selective positive allosteric modulator of mGluR4
-
GC13031
Trifluoperazine 2HCl
盐酸三氟拉嗪;甲哌氟丙嗪;三氟吡拉嗪
An anti-adrenergic and anti-dopaminergic agent
-
GC18092
Tolazoline HCl
盐酸妥拉唑林; Imidaline hydrochloride; NSC35110 hydrochloride
An α1- and α2-adrenergic receptor antagonist
-
GC14962
Tetrahydrozoline HCl
盐酸四氢唑林; Tetryzoline hydrochloride
An α1-adrenergic receptor agonist
-
GC11211
Terbutaline Sulfate
硫酸特布他林
An Analytical Reference Standard
-
GC12715
Synephrine HCl
辛弗林盐酸盐; Oxedrine hydrochloride
An alkaloid
-
GC14843
Serotonin HCl
5-羟基色胺盐酸盐; 5-Hydroxytryptamine hydrochloride; 5-HT hydrochloride
Serotonin HCl是一种神经递质,是介导人体多种中枢和外周功能的关键信使。
-
GC14550
SB271046
An orally-available 5-HT6 antagonist
-
GC11033
Rupatadine Fumarate
富马酸卢帕他定; UR-12592 Fumarate
A histamine H1 and PAF receptor antagonist
-
GC13291
Prucalopride Succinat
琥珀酸普芦卡必利; R-108512
A selective 5-HT4 receptor agonist