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GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC14818 Bisoprolol fumarate

    比索洛尔富马酸盐

    A β1-AR antagonist
  3. GC14563 Ketanserin

    酮色林; R41468

    A potent 5-HT2 receptor antagonist
  4. GC11191 Buspirone HCl

    盐酸丁螺环酮

    An Analytical Reference Standard
  5. GC10434 Triamcinolone

    曲安西龙

    A synthetic glucocorticoid
  6. GC17974 Latrepirdine dihydrochloride

    2,3,4,5-四氢-2,8-二甲基-5-[2-(6-甲基-3-吡啶基)乙基]-1H-吡啶并[4,3-B]吲哚二盐酸盐,Dimebolin dihydrochloride

    A neuroprotective agent
  7. GC17061 Dapoxetine HCl

    盐酸达泊西汀; LY-210448 hydrochloride

    An Analytical Reference Standard
  8. GC15829 Urapidil HCl

    盐酸乌拉地尔

    An α1-AR antagonist and 5-HT1A receptor partial agonist
  9. GC12376 Maprotiline HCl

    盐酸马普替林

    A tricyclic antidepressant
  10. GC13993 Terazosin HCl

    盐酸特拉唑嗪(二水合物)

    A potent and selective α1-AR antagonist
  11. GC15107 Clomipramine HCl

    盐酸氯米帕明; Chlorimipramine hydrochloride; G-34586 hydrochloride; NSC-169865 hydrochloride

    A tricyclic antidepressant
  12. GC13134 Tiotropium Bromide hydrate

    噻托溴铵一水合物,BA-679 BR (hydrate)

    A muscarinic receptor antagonist
  13. GC14927 Trazodone HCl

    盐酸曲唑酮; AF-1161

    An Analytical Reference Material
  14. GC17367 Rebamipide

    瑞巴派特; OPC12759; Proamipide

    A gastroprotective agent and mucin secretagogue
  15. GC14021 Betaxolol

    倍他洛尔

    An Analytical Reference Standard
  16. GC17825 Methscopolamine

    甲溴东莨菪碱

    A muscarinic acetylcholine receptor antagonist
  17. GC12724 Phenoxybenzamine HCl

    盐酸酚苄明

    An α-AR antagonist
  18. GC16142 Ondansetron

    昂丹司琼; GR 38032; SN 307

    A Certified Reference Material
  19. GC15153 Almotriptan Malate

    马来酸阿莫曲坦; PNU180638

    An agonist of 5-HT1B and 5-HT1D receptors
  20. GC15063 Ritodrine HCl

    盐酸利托君; DU21220 hydrochloride

    A β2-AR agonist
  21. GC15150 Tropicamide

    托吡卡胺; Ro 1-7683

    A selective muscarinic M4 antagonist
  22. GC15687 Azasetron HCl

    盐酸阿扎司琼; Y-25130 hydrochloride

    A 5-HT3 receptor antagonist
  23. GC16291 Phentolamine Mesylate

    甲磺酸酚妥拉明; Phentolamine methanesulfonate

    A reversible α-adrenergic receptor antagonist
  24. GC11447 Mirtazapine

    米氮平

    Mirtazapine是一种去甲肾上腺素能和特异性血清素抗抑郁药(NaSSA),可抑制5-HT2A、5-HT2B、5-HT2C和5-HT3受体,pKi值分别为8.2、6.7、7.9和8.1。
  25. GC14216 Chlorpromazine HCl

    盐酸氯丙嗪

    Chlorpromazine HCl是一种口服有效的、可透过血脑屏障的吩噻嗪类抗精神病药,能够有效抑制D2多巴胺受体和5-HT2A,具有很强的镇静作用。
  26. GC11343 Propranolol HCl

    盐酸普萘洛尔

    A β-adrenergic receptor antagonist
  27. GC10738 Brimonidine Tartrate

    酒石酸溴莫尼定; UK 14304 tartrate; AGN190342 tartrate

    An α2-adrenergic receptor agonist
  28. GC14988 Naphazoline HCl

    盐酸萘甲唑啉; Naphthazoline hydrochloride

    A vasoconstrictor
  29. GC13974 Salbutamol Sulfate

    沙丁胺醇半硫酸盐; Albuterol hemisulfate; AH-3365 hemisulfate

    A β2-AR agonist
  30. GC10750 Dexmedetomidine HCl

    盐酸右美托咪定; (+)-Medetomidine hydrochloride; (S)-Medetomidine hydrochloride

    An α2-adrenoceptor agonist
  31. GC12403 Ozagrel HCl

    盐酸奥扎格雷,OKY-046 hydrochloride

    A selective inhibitor of TXA synthase
  32. GC13173 Sotalol

    索他洛尔,(R)-Sotalol

    An Analytical Reference Standard
  33. GC17296 Xylazine HCl

    盐酸甲苯噻嗪,BAY 1470 hydrochloride

    An α2-adrenergic receptor agonist

  34. GC11029 Isoprenaline HCl

    盐酸异丙肾上腺素; Isoproterenol hydrochloride

    A β1- and β2-AR agonist

  35. GC12231 Sulfisoxazole

    磺胺异恶唑; Sulfafurazole

    An antibiotic and endothelin receptor antagonist
  36. GC15243 Carbazochrome sodium sulfonate (AC-17)

    卡络磺钠; AC-17

    Carbazochrome sodium sulfonate (AC-17) (AC-17) 是一种毛细血管稳定剂,用于研究出血。
  37. GC14536 Metoprolol Tartrate

    酒石酸美托洛尔

    An Analytical Reference Standard
  38. GC11479 Xylometazoline HCl

    盐酸赛洛唑啉

    An α-adrenergic receptor agonist
  39. GC15754 WAY-100635 Maleate A serotonin 5-HT1A antagonist
  40. GC13501 VUF 10166 A 5-HT3 receptor antagonist
  41. GC13281 VU 0364770 An mGluR4 and mGluR6 positive allosteric modulator and mGluR5 antagonist
  42. GC13962 VU 0361737

    ML-128

    A selective positive allosteric modulator of mGluR4
  43. GC13031 Trifluoperazine 2HCl

    盐酸三氟拉嗪;甲哌氟丙嗪;三氟吡拉嗪

    An anti-adrenergic and anti-dopaminergic agent
  44. GC18092 Tolazoline HCl

    盐酸妥拉唑林; Imidaline hydrochloride; NSC35110 hydrochloride

    An α1- and α2-adrenergic receptor antagonist
  45. GC14962 Tetrahydrozoline HCl

    盐酸四氢唑林; Tetryzoline hydrochloride

    An α1-adrenergic receptor agonist
  46. GC11211 Terbutaline Sulfate

    硫酸特布他林

    An Analytical Reference Standard
  47. GC12715 Synephrine HCl

    辛弗林盐酸盐; Oxedrine hydrochloride

    An alkaloid
  48. GC14843 Serotonin HCl

    5-羟基色胺盐酸盐; 5-Hydroxytryptamine hydrochloride; 5-HT hydrochloride

    Serotonin HCl是一种神经递质,是介导人体多种中枢和外周功能的关键信使。

  49. GC14550 SB271046 An orally-available 5-HT6 antagonist
  50. GC11033 Rupatadine Fumarate

    富马酸卢帕他定; UR-12592 Fumarate

    A histamine H1 and PAF receptor antagonist
  51. GC13291 Prucalopride Succinat

    琥珀酸普芦卡必利; R-108512

    A selective 5-HT4 receptor agonist

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