GlpBio

GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

研究方向

GPCR/G protein 相关产品(3377)

  • GC18867 structure
    GC18867SER-601
    CAS: 1048038-90-9

    A selective CB 2 receptor agonist

  • GC18951 structure
    GC18951Obscurolide A1
    CAS: 144397-99-9

    A phosphodiesterase inhibitor

  • GC19023 structure
    GC19023AF38469
    CAS: 1531634-31-7
    纯度: >98.00%

    AF38469是一种具有口服活性的Sortilin（SORT1；IC 50 =330nM）受体抑制剂。

  • GC19030 structure
    GC19030AMG 837
    CAS: 865231-46-5

    An FFAR1 (GPR40) partial

  • GC19031 structure
    GC19031Amiselimod hydrochloride
    CAS: 942398-84-7
    纯度: >99.00%

    A prodrug form of amiselimod phosphate

  • GC19032 structure
    GC19032AVex-73 hydrochloride
    CAS: 195615-84-0
    纯度: >98.00%

    AVex-73 hydrochloride 是一种 Sigma-1 Receptor 激动剂，IC50 为 860 nM。

  • GC19033 structure
    GC19033APD597
    CAS: 897732-93-3
    纯度: >99.50%

    An agonist of GPR119

  • GC19037 structure
    GC19037ARS-853
    CAS: 1629268-00-3
    纯度: >98.00%

    An inhibitor of KRAS G12C

  • GC19049 structure
    GC19049AZD4635
    CAS: 1321514-06-0
    纯度: >99.50%

    AZD4635是一种强效、选择性的口服腺苷2A受体（A2AR）抑制剂，K i 值为1.7nM。

  • GC19051 structure
    GC19051AZD7594
    CAS: 1196509-60-0
    纯度: >99.00%

    AZD7594 是一种有效的选择性非甾体糖皮质激素受体调节剂，IC50 为 0.9 nM。

  • GC19060 structure
    GC19060Bay 59-3074
    CAS: 406205-74-1
    纯度: >98.50%

    A partial agonist of CB 1 and CB 2 receptors

  • GC19071 structure
    GC19071BIBS 39
    CAS: 133085-33-3
    纯度: >98.00%

    A nonpeptide AT 1 receptor antagonist

  • GC19077 structure
    GC19077BMS-813160
    CAS: 1286279-29-5
    纯度: >99.50%

    A dual antagonist of CCR2 and CCR5

  • GC19078 structure
    GC19078BMS-986020
    CAS: 1257213-50-5
    纯度: >99.50%

    An LPA 1 receptor antagonist

  • GC19081 structure
    GC19081BPTU
    CAS: 870544-59-5
    纯度: >99.00%

    A P2Y 1 receptor antagonist

  • GC19087 structure
    GC19087Capromorelin Tartrate
    CAS: 193273-69-7
    纯度: >98.50%

    A growth hormone secretagogue and GHS-R1a agonist

  • GC19100 structure
    GC19100Cenerimod
    CAS: 1262414-04-9
    纯度: >98.00%

    A S1P 1 receptor modulator

  • GC19101 structure
    GC19101Cenicriviroc
    CAS: 497223-25-3
    纯度: >98.00%

    Cenicriviroc (CVC) 是一种口服的 CCR2/CCR5 双重拮抗剂，对这两种受体具有纳摩尔效力。

  • GC19116 structure
    GC19116Danirixin
    CAS: 954126-98-8
    纯度: >98.00%

    A CXCR2 antagonist

  • GC19137 structure
    GC19137EMA401
    CAS: 1316755-16-4
    纯度: >99.00%

    A selective AT 2 receptor antagonist

  • GC19146 structure
    GC19146Etrasimod
    CAS: 1206123-37-6
    纯度: >99.50%

    A potent S1P 1 receptor antagonist

  • GC19147 structure
    GC19147Evatanepag
    CAS: 223488-57-1
    纯度: >99.00%

    Evatanepag (CP-533536) 是一种非前列腺素、强效和选择性 EP2 受体激动剂。

  • GC19153 structure
    GC19153Fevipiprant
    CAS: 872365-14-5
    纯度: >99.50%

    A DP 2 /CRTH 2 antagonist

  • GC19164 structure
    GC19164GGTI298 Trifluoroacetate
    CAS: 1217457-86-7
    纯度: >95.00% / >98.00% / >99.50%

    GGTI298 Trifluoroacetate是一种选择性、不可逆的香叶基香叶酰转移酶I（GGTase-I）抑制剂（IC 50 = 3μM)。