GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC18139DevazepideCAS: 103420-77-5纯度: >98.50%
Devazepide (L-364,718) 是一种有效、竞争性、选择性和口服活性的胆囊收缩素 (CCK) 受体非肽拮抗剂，对大鼠胰腺、牛胆囊和豚鼠脑 CCK 受体的 IC50 分别为 81 pM、45 pM 和 245 nM .
- GC18244Eltoprazine (hydrochloride)CAS: 98206-09-8纯度: >99.50%
A partial agonist of 5-HT 1A , 5-HT 1B , and 5-HT 2B receptors
- GC18412VU0409551 (JNJ-46778212)CAS: 1363281-27-9纯度: >99.00% / >99.50%
VU0409551 (JNJ-46778212)是一种强效且选择性的偏向性代谢型谷氨酸受体5亚型正变构调节剂（mGlu 5 PAM；EC 50 =260nM）。
- GC18435Arachidonoyl 2'-ChloroethylamideCAS: 220556-69-4纯度: >95.00%
A potent and selective CB 1 receptor agonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC18125 | DC260126 | 346692-04-4 | >98.00% | |
An FFAR1 (GPR40) antagonist | ||||
| GC18128 | L-732,138 | 148451-96-1 | >99.00% | |
An NK 1 receptor antagonist | ||||
| GC18132 | U-44069 | 56985-32-1 | - | |
A TP receptor agonist | ||||
| GC18138 | CYM 50769 | 1421365-63-0 | - | |
An NPBWR1 antagonist | ||||
| GC18139 | Devazepide | 103420-77-5 | >98.50% | |
Devazepide (L-364,718) 是一种有效、竞争性、选择性和口服活性的胆囊收缩素 (CCK) 受体非肽拮抗剂，对大鼠胰腺、牛胆囊和豚鼠脑 CCK 受体的 IC50 分别为 81 pM、45 pM 和 245 nM . | ||||
| GC18145 | Urotensin II (human) | 251293-28-4 | - | |
A neuropeptide agonist of the urotensin II receptor | ||||
| GC18202 | Temocaprilat | 110221-53-9 | - | |
An ACE inhibitor | ||||
| GC18216 | ML314 | 1448895-09-7 | >99.50% | |
An NTS 1 agonist | ||||
| GC18244 | Eltoprazine (hydrochloride) | 98206-09-8 | >99.50% | |
A partial agonist of 5-HT 1A , 5-HT 1B , and 5-HT 2B receptors | ||||
| GC18255 | Xanomeline (oxalate) | 141064-23-5 | >99.50% | |
Potent agonist of muscarinic receptors | ||||
| GC18318 | CAY10441 | 221529-58-4 | >98.00% | |
An IP receptor antagonist | ||||
| GC18327 | Todralazine (hydrochloride) | 3778-76-5 | >98.00% | |
A β 2 -adrenergic receptor antagonist | ||||
| GC18348 | Ceralifimod | 891859-12-4 | >95.00% | |
An agonist of S1P 1 and S1P 5 receptors | ||||
| GC18412 | VU0409551 (JNJ-46778212) | 1363281-27-9 | >99.00% / >99.50% | |
VU0409551 (JNJ-46778212)是一种强效且选择性的偏向性代谢型谷氨酸受体5亚型正变构调节剂（mGlu 5 PAM；EC 50 =260nM）。 | ||||
| GC18435 | Arachidonoyl 2'-Chloroethylamide | 220556-69-4 | >95.00% | |
A potent and selective CB 1 receptor agonist | ||||
| GC18458 | Terrein | 582-46-7 | >98.00% | |
A fungal metabolite with diverse biological activities | ||||
| GC18472 | Elinogrel | 936500-94-6 | - | |
A reversible P2Y 12 antagonist | ||||
| GC18496 | Leelamine (hydrochloride) | 16496-99-4 | - | |
An inhibitor of pyruvate dehydrogenase kinase | ||||
| GC18501 | Kendomycin | 183202-73-5 | - | |
A cytotoxic macrolide | ||||
| GC18648 | Echothiophate (iodide) | 513-10-0 | - | |
An AChE inhibitor | ||||
| GC18661 | Vercirnon | 698394-73-9 | >98.00% | |
Vercirnon是一种新型的、具有口服活性的CCR9趋化因子受体选择性拮抗剂，抑制CCR9介导的Molt-4细胞钙离子动员和趋化作用的IC₅₀值分别为5.4nM和3.4nM | ||||
| GC18678 | CAY10595 | 916047-16-0 | - | |
A potent CRTH2/DP 2 receptor antagonist | ||||
| GC18719 | Docosatetraenoyl Ethanolamide | 150314-35-5 | >98.00% | |
An endocannabinoid | ||||
| GC18866 | MCHB-1 | 1046140-32-2 | - | |
A CB 2 receptor agonist | ||||