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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

Cat.No. 产品名称 Information
GC14527 A 61603 hydrobromide
A61603氢溴酸
An α_1A-adrenoceptor agonist
GC16111 Zinterol hydrochloride
净特罗,MJ 9184 hydrochloride
Zinterol hydrochloride (MJ 9184) 是一种有效的选择性 β2-adrenoceptor 激动剂。
GC12532 CHPG
Chlorohydroxyphenylglycine, CHPG
A potent and selective mGluR5 agonist
GC11017 ZM 241385 An A_2A adenosine receptor antagonist
GC16020 8-M-PDOT
AH-002
An MT₂ receptor agonist
GC16186 4-P-PDOT
AH 024
4-P-PDOT是一种具有口服活性的、高选择性的褪黑激素MT2受体拮抗剂，它对MT2受体的选择性是MT1的300倍以上（Ki值分别为0.46nM和56nM）。
GC10068 CP 93129 dihydrochloride A 5-HT_1B receptor agonist
GC17383 PHCCC
N-苯基-7-(羟基亚胺基)环丙烯并[B]苯并吡喃-1A-甲酰胺
PHCCC 是 I 组 mGluR 拮抗剂，IC50 为 3 μM。 PHCCC 是 mGlu4 受体的选择性正调节剂。抗帕金森效应。
GC15482 Nisoxetine hydrochloride
盐酸尼索西汀
A NET inhibitor
GC15354 CGP 20712 dihydrochloride β1 antagonist,highly potent and selective
GC11305 LY 225910
2-[2-(5-溴-1H-吲哚-3-基)乙基]-3-[3-(1-甲基乙氧基)苯基]-4-(3H-)-喹唑啉酮
LY 225910是一种有效的胆囊收缩素受体拮抗剂，可特异性阻断CCK2受体并影响神经递质释放
GC15979 RS 16566 dihydrochloride (R)-zacopride 结合位点的配体
GC13192 E4CPG
(RS)-ECPG
An antagonist of mGluR1 and mGluR2
GC16553 N-Desmethylclozapine
N-去甲基氯氮平; Norclozapine; Desmethylclozapine; Normethylclozapine
An active metabolite of clozapine
GC10197 AH 11110 hydrochloride α1B-AR ligand,subtype-selective
GC14696 RS 67506 hydrochloride potent and selective 5-HT4 partial agonist
GC15137 RS 56812 hydrochloride
5-HT3 partial agonist
GC10723 RS 79948 hydrochloride α2-adrenoreceptor antagonist
GC11077 Imiloxan hydrochloride α2-adrenoceptor antagonist
GC17070 RS 17053 hydrochloride
RS-17053
An α_1A-adrenergic receptor antagonist
GC15374 BD 1047 dihydrobromide
BD-1047盐酸盐
A selective antagonist of σ₁ receptors
GC17666 Xamoterol hemifumarate
富马酸扎莫特罗,Corwin hemifumarate; ICI 118587 hemifumarate
A β₁-adrenergic receptor partial agonist
GC13785 BRL 37344, sodium salt
BRL37344钠盐,BRL 37344A
A selective β₃-adrenergic receptor agonist
GC17745 MK 212 hydrochloride
2-氯-6-哌嗪吡嗪盐酸盐,CPP monohydrochloride
A 5-HT_2C receptor agonist
GC17543 ZD 7114 hydrochloride β3-adrenoceptor agonist
GC10965 ARC 239 dihydrochloride
ARC?239二盐酸盐
An α2B-adrenergic receptor antagonist
GC11188 GR 135531
N-甲氧基羰基琥珀酰亚胺,5-METHOXYCARBONYLAMINO-N-ACETYLTRYPTAMINE
MT3 receptor agonist
GC15838 BD 1063 dihydrochloride
BD1063(盐酸盐)
An antagonist of σ₁ receptors
GC17777 Palmitoylethanolamide
十六酰胺乙醇,Palmidrol; Loramine P 256
An endogenous cannabinoid
GC14042 Oleamide
油酸酰胺
An amide of oleic acid and agonist of CB₁ receptors
GC17898 Luzindole
N-乙酰-2-苄基色胺,N-0774
Luzindole是一种选择性褪黑激素受体（MT）拮抗剂，对MT1的Ki值为158nM，对MT2的Ki值为10.2nM。
GC11119 MDL 11,939
MDL11939
A potent 5-HT_2A receptor antagonist
GC18128 L-732,138 An NK₁ receptor antagonist
GC12761 ICI 89406
N-[2-[[3-(2-氰基苯氧基)-2-羟基丙基]氨基]乙基]-N'-苯基脲
ICI 89406 是一种选择性 β1 肾上腺素能受体拮抗剂，适合用正电子发射器标记，用于 PET。
GC17185 MSOP MSOP 是一种选择性 III 族代谢型谷氨酸受体拮抗剂，对 L-AP4 敏感的突触前 mGluR 的表观 KD 为 51 μM。
GC15813 Idazoxan hydrochloride
盐酸咪唑克生
盐酸咪唑克生（Idazoxan hydrochloride ，RX 781094 hydrochloride ，IDA）是一种分子量为241的α2-肾上腺和咪唑啉受体配体。
GC15672 Efaroxan hydrochloride
盐酸盐依法克生
An α₂-AR and I₁ receptor antagonist
GC15465 N-[2-(Piperidinylamino)ethyl]-4-iodobenzamide σ-1 selective ligand
GC11575 SM-21 maleate Increases release of acetylcholine，σ2 antagonist
GC17929 PG-9 maleate Increases release of acetylcholine
GC17723 4-IBP
NSC 667672
A σ1 receptor ligand
GC14690 2-Iodomelatonin
2-碘褪黑激素
A potent MT₁ receptor agonist
GC14959 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 5-HT4 receptor
GC16861 RS 23597-190 hydrochloride
3-(哌啶-1-基)丙基4-氨基-5-氯-2-甲氧基苯甲酸酯盐酸盐
RS 23597-190 hydrochloride是一种高效且有选择性的5-羟色胺4型（5-HT₄）受体（5-HT₄R）拮抗剂。
GC11288 2-Phenylmelatonin
2-Phenylmelatonin
A MT receptor mixed partial agonist and antagonist
GC15569 3-AQC 5-HT3 antagonist
GC16412 2-MPMDQ α1-adrenoceptor antagonist,potent and selective
GC13338 Spiroxatrine
三氮螺癸苯恶烷
5-HT1A拮抗剂和α2C肾上腺素能受体拮抗剂
GC13695 2-PMDQ α1-adrenoceptor antagonist
GC13357 4-PPBP maleate 4-PPBP maleate 是一种有效的 σ 1 受体配体和激动剂。