GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC16111Zinterol hydrochlorideCAS: 37000-20-7
Zinterol hydrochloride (MJ 9184) 是一种有效的选择性 β2-adrenoceptor 激动剂。
- GC16172MPEP HydrochlorideCAS: 219911-35-0纯度: >98.00%
MPEP Hydrochloride是一种非竞争性、选择性的、强效、有口服活性和系统活性的mGlu5受体拮抗剂，其完全抑制quisqualate 刺激的磷酸肌醇水解的IC 50 为36nM。
- GC16250Rauwolscine hydrochlorideCAS: 6211-32-1纯度: ≥98%
A reversible α 2 -adrenergic receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16106 | Atipamezole hydrochloride | 104075-48-1 | >99.00% | |
An α 2A -adrenergic receptor antagonist | ||||
| GC16110 | R 715 | 185052-09-9 | - | |
缓激肽 B1 受体拮抗剂 | ||||
| GC16111 | Zinterol hydrochloride | 37000-20-7 | - | |
Zinterol hydrochloride (MJ 9184) 是一种有效的选择性 β2-adrenoceptor 激动剂。 | ||||
| GC16135 | Cinanserin hydrochloride | 54-84-2 | >99.50% | |
A 5-HT receptor antagonist | ||||
| GC16137 | CCG 2046 | 13017-69-1 | - | |
CCG 2046 是一种 RGS4 抑制剂，IC50 为 4.3 μM 针对 RGS4-Gαo 相互作用信号。 | ||||
| GC16141 | Nicergoline | 27848-84-6 | >99.50% | |
An α 1 -AR antagonist | ||||
| GC16147 | CGRP 8-37 (human) | 119911-68-1 | >98.00% | |
CGRP 8-37 (human)是一种高选择性的CGRP受体拮抗剂。 | ||||
| GC16150 | VU 0364439 | 1246086-78-1 | >98.50% | |
A positive allosteric modulator of mGluR4 | ||||
| GC16159 | ANR 94 | 634924-89-3 | - | |
ANR 94 是一种有效的选择性腺苷 A2A 受体 (AA2AR) 拮抗剂，对 hAA2AR 的 Ki 值为 46 nM。 | ||||
| GC16168 | PACAP 1-38 | 137061-48-4 | >99.50% | |
A PACAP receptor agonist | ||||
| GC16170 | Ethamsylate | 2624-44-4 | >98.00% | |
Ethamsylate 是一种止血药，也抑制这些前列腺素的生物合成和作用。 | ||||
| GC16171 | PF 514273 | 851728-60-4 | - | |
CB1 receptor antagonist | ||||
| GC16172 | MPEP Hydrochloride | 219911-35-0 | >98.00% | |
MPEP Hydrochloride是一种非竞争性、选择性的、强效、有口服活性和系统活性的mGlu5受体拮抗剂，其完全抑制quisqualate 刺激的磷酸肌醇水解的IC 50 为36nM。 | ||||
| GC16186 | 4-P-PDOT | 134865-74-0 | >98.00% | |
4-P-PDOT是一种具有口服活性的、高选择性的褪黑激素MT2受体拮抗剂，它对MT2受体的选择性是MT1的300倍以上（Ki值分别为0.46nM和56nM）。 | ||||
| GC16196 | 2-Palmitoylglycerol | 23470-00-0 | >95.00% | |
An endogenous fatty acid ester | ||||
| GC16216 | Asterric Acid | 577-64-0 | - | |
An antiangiogenic agent | ||||
| GC16217 | TC-G 1000 | 245744-18-7 | - | |
α2D-adrenoceptor agonist | ||||
| GC16218 | Astressin | 170809-51-5 | >98.00% / >98.50% | |
Astressin是一种有效的非选择性的促肾上腺皮质激素释放因子（CRF）拮抗剂，对CRF结合蛋白具有低亲和力，而对克隆的垂体受体具有高亲和力（K i =2nM）。 | ||||
| GC16222 | Oxytocin | 50-56-6 | >98.00% / >97.00% | |
Oxytocin是一种多效的下丘脑肽，有助于分娩、哺乳和亲社会行为。 | ||||
| GC16232 | BETP | 1371569-69-5 | >99.00% | |
A positive allosteric modulator of GLP-1R | ||||
| GC16246 | Fosaprepitant | 172673-20-0 | - | |
A prodrug form of aprepitant | ||||
| GC16250 | Rauwolscine hydrochloride | 6211-32-1 | ≥98% | |
A reversible α 2 -adrenergic receptor antagonist | ||||
| GC16276 | Melanotan II | 121062-08-6 | >99.50% | |
A melanocortin receptor agonist | ||||
| GC16281 | IRL-1038 | 144602-02-8 | - | |
ETB endothelin receptor antagonist | ||||