JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

Cat.No. 产品名称 Information
GC13497 BML-111
BML-111
A potent bioactive analog of lipoxin A₄
GC11002 5'-(N-Cyclopropyl)carboxamidoadenosine
CPCA
A specific adenosine A₂ receptor agonist
GC14661 AM6545 A peripherally restricted CB₁ receptor antagonist
GC12948 CID-1067700
2-[[(苯甲酰基氨基)硫代甲酰]氨基]-4,7-二氢-5,5-二甲基-5H-噻吩并[2,3-C]吡喃-3-羧酸,ML-282
CID-1067700是Rab GTPases的抑制剂，特别是对Rab2和Rab7具有显著的抑制作用。
GC14026 ML-193
CID-1261822
A selective GPR55 antagonist
GC12023 Celiprolol (hydrochloride)
盐酸塞利洛尔
A β₁ adrenergic receptor antagonist
GC16216 Asterric Acid
曲地酸,Dimethylosoic Acid,RES-1214-1,TAN 1415A
An antiangiogenic agent
GC11952 (R)-(+)-Atenolol
(R)-(+)-阿替洛尔
An enantiomer of (±)-atenolol
GC15087 (±)-Talinolol
他林洛尔,Cordanum
A β₁-adrenergic receptor blocker
GC13720 TY 52156 A S1P₃ receptor antagonist
GC11239 Midodrine (hydrochloride)
盐酸米多君; (±)-Midodrine hydrochloride
A prodrug form of desglymidodrine
GC10673 E7046
E7046
An EP₄ receptor antagonist
GC11201 ARM1
4BSA
An inhibitor of LTA₄ hydrolase
GC14859 BW 246C
8-epi BW 245C
The less active C-8 diastereomer of BW 245C
GC17719 5-trans U-46619
5,6-trans U-46619
An isomer of U-46619
GC10433 ML-178
CID 44620892,CYM 50179,SID 87544119
A selective S1P₄ agonist
GC17720 W123 Antagonist of spingosine 1-phosphate type 1 receptor
GC14433 7α,25-dihydroxy Cholesterol
7Α,25-二羟基胆固醇,7α,25-DHC
A potent and selective agonist of GPR183
GC11603 AG-041R A potent gastrin/CCK_B receptor antagonist
GC13712 FTY720 Phosphate
2-氨基-2-(羟基甲基)-4-(4-辛基苯基)丁基磷酸二氢酯,FTY720P
The active metabolite of FTY720
GC16826 Arachidonoyl amide
Arachidonamide,Arachidonic Acid amide
An AEA analog with similar biological activity
GC16663 (±)-4-hydroxy Propranolol (hydrochloride)
4-羟基普萘洛尔盐酸盐,(±)-4-hydroxy Propranolol hydrochloride
An active metabolite of propranolol
GC13284 CJ-42794
4-[(1S)-1-[[5-氯-2-(4-氟苯氧基)苄基]氨基]乙基]苯甲酸,RQ-00015986
A selective EP₄ receptor antagonist
GC12290 Norgestimate
诺孕酯
A progestin
GC15640 BAY u3405
雷马曲班; BAY u3405
A dual TP and DP₂/CRTH₂ receptor antagonist
GC18111 Seratrodast
塞曲司特; AA 2414
A thromboxane A₂ receptor antagonist
GC14758 BM 567 A dual thromboxane synthase inhibitor/TP receptor antagonist
GC12538 LH 21 Weak CB₁ antagonist
GC10771 CJ-023423
RQ-00000007
An EP₄ receptor antagonist
GC10284 Apelin-13
人牛APELIN-13
Apelin-13 是一种肽，被称为 G 蛋白偶联受体 APJ 的配体。
GC17699 O-1821
Cannabidiorcin, Cannabidiorcol, Cannabidiorocol, CBD-C1, CBDO
An analog of O-1918, a selective antagonist of a non-CB₁/CB₂ receptor
GC13333 Zilpaterol
齐帕特罗,RU-42173,Zilmax?
β-adrenergic receptor agonist
GC16800 MF498 A selective EP₄ antagonist
GC13020 BayCysLT2
CAY10633
A potent CysLT₂ receptor antagonist
GC10116 2-chloro-3-Deazaadenosine
6-Amino-2-chloropurine riboside,2-CADO,NSC 158900
Agonist of adenosine receptors
GC15758 BQCA
1-(4-甲氧基苄基)-4-氧代-1,4-二氢喹啉-3-羧酸
A positive allosteric modulator of the M₁ mAChR
GC13302 Guanabenz (hydrochloride)
Wytensin
An α₂-adrenergic receptor agonist
GC16027 ONO-8711
(5Z)-6-[(2R,3S)-3-[[[(4-氯-2-甲基苯基)磺酰基]氨基]甲基]双环[2.2.2]辛-2-基]-5-己烯酸
A potent EP₁ receptor antagonist
GC17064 Lofexidine (hydrochloride)
盐酸洛非西定; Baq-168; MDL-14042
An α₂-adrenergic receptor agonist
GC15657 Rilmenidine (hemifumarate)
Oxaminozoline,S 3341

An antihypertensive agent
GC10643 Pimozide
匹莫齐特; R6238
Pimozide是一种化学结构新颖、高效且口服长效的神经阻滞剂类多巴胺受体抑制剂，对多巴胺D2、D3和D4 受体的Ki值分别为2.4nM、0.2nM和1.8nM。
GC17218 2-fluoro Palmitic Acid
2-氟十六酸
Inhibitor of sphingosine biosynthesis and long-chain acyl-CoA synthetase
GC13190 R-Palmitoyl-(1-methyl) Ethanolamide
R-1 PMA
A synthetic analog of palmitoyl ethanolamide
GC17348 BW A868C
3-[(2-环己基-2-羟乙基)氨基]-2,5-二氧代-1-(苯甲基)-4-咪唑啶庚酸
A DP receptor antagonist
GC12587 1-(1-Naphthyl) piperazine (hydrochloride)
1-(1-萘基)哌嗪盐酸盐,1-NP
A serotonin receptor antagonist
GC17100 4-Quinolone-3-Carboxamide CB2 Ligand
4Q3C CB2 Ligand
An Analytical Reference Standard
GC15850 4-Quinolone-3-Carboxamide Furan CB2 Agonist
4Q3C CB2 Agonist
Selective CB₂ agonist
GC13660 JD5037 JD5037 是一种有效的 CB1R 拮抗剂，IC50 为 1.5 nM。
GC10753 (S)-SLV 319
伊必那班,Ibipinabant|BMS 646256|JD 5001
A selective antagonist of CB₁
GC11800 SB 290157 (trifluoroacetate salt) SB 290157（三氟乙酸盐）用作选择性非肽类 C3aR 拮抗剂。