GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(481)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(404)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(116)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(78)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(78)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(95)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(5)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
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GC18202
Temocaprilat
替莫普利
An ACE inhibitor
-
GC18152
AZ-3451
(S)-2-(6-溴苯并[D][1,3]二氧杂环戊烯-5-基)-N-(4-氰基苯基)-1-(1-环己基乙基)-1H-苯并[D]咪唑-5-甲酰胺
A PAR2 antagonist
-
GC10311
Liraglutide
利拉鲁肽
利拉鲁肽是一种高效、长效的 GLP-1 受体激动剂 (EC50 = 61 pM)，其氨基酸序列与人 GLP-1 有 97% 的同一性 .用 PA/LPS 处理的肝细胞中的活细胞数量显着减少，利拉鲁肽以浓度依赖性方式逆转细胞活力的下降。
-
GC16403
2-Arachidonoyl Glycerol
2-花生酰基甘油乙腈溶液,2-AG
Endogenous CB1 and CB2 receptor agonist
-
GC16539
Butaprost
布他前列素
A selective agonist for the EP2 receptors
-
GC17888
Metipranolol
美替洛尔
A β-AR antagonist
-
GC12238
Oxomemazine
双氧异丁嗪
Oxomemazine 是一种基于吩噻嗪的组胺 H1 受体阻滞剂，具有明显的抗毒蕈碱特性。
-
GC13844
p-iodo-Clonidine (hydrochloride)
An α2-adrenergic receptor partial agonist
-
GC14211
ONO-8130
A selective, orally bioavailable EP1 antagonist
-
GC14300
GPR120 Compound A
GPR120 cpdA
A selective GPR120/FFAR4 agonist
-
GC13180
Carazolol
卡拉洛尔; (±)-Carazolol; DL-Carazolol; Suacron
A β-AR ligand
-
GC10283
γ-Linolenic Acid
γ-亚麻酸 ;Gamma-Linolenic acid
γ-Linolenic Acid是一种来源于琉璃苣油的口服ω-6多不饱和脂肪酸，可作为β-分泌酶（BACE1）的特异性抑制剂，IC50值为7.6×10−5mol/L，Ki值为3.5×10−5mol/L。
-
GC14939
REV 5901
An antagonist of cysteinyl-leukotriene receptors
-
GC12868
S-2 Methanandamide
(S)-(+)-Arachidonyl-2'-Hydroxy-1'-Propylamide
A potent CB1 receptor agonist
-
GC13605
S-1 Methanandamide
(S)-(−)-Arachidonyl-1'-Hydroxy-2'-Propylamide
A CB1 receptor ligand
-
GC17736
Anisodamine
山莨菪碱; 6-Hydroxyhyoscyamine
Anisodamine (6-Hydroxyhyoscyamine) 是一种颠茄生物碱，是一种非亚型选择性毒蕈碱，也是一种烟碱型胆碱受体拮抗剂。
-
GC17488
Trimipramine (maleate)
三甲丙咪嗪马来酸盐
A tricyclic antidepressant
-
GC11667
VU0483605
A selective mGlu1 PAM
-
GC11668
ML-031
CID-2113511
A S1P2 agonist
-
GC18132
U-44069
9,11-dideoxy-9α,11α-epoxymethano PGF2α,9,11-dideoxy-9α,11α-epoxymethano Prostaglandin F2α,9,11-epoxymethano Prostaglandin H2
A TP receptor agonist
-
GC15365
N-Acetylserotonin
N-乙酰-5-羟色胺,N-Acetyl-5-hydroxytryptamine,NAS
N-Acetylserotonin是褪黑素生物合成中的一个化学中间体，以昼夜节律的方式激活酪氨酸激酶受体B（TrkB）。
-
GC11350
6-OAU
GTPL5846
6-OAU是G蛋白偶联受体84（GPR84）的特异性激动剂，可以诱导PMNs（polymorphonuclear leukocytes）和巨噬细胞的趋化以及巨噬细胞的促炎反应。
-
GC11966
O-Phospho-D-Serine
D-O-Phosphoserine,D-Serine-O-Phosphate,D-SOP
weak agonist of the metabotropic glutamate receptor mGluR4
-
GC12620
Calindol (hydrochloride)
A calcimimetic and CaSR agonist
-
GC12823
(R,S)-Atenolol
阿替洛尔; (RS)-Atenolol
A β1-AR antagonist
-
GC16930
Adenosine Kinase Inhibitor (hydrate)
ABT-702
Blocks the action of adenosine kinase
-
GC18041
NESS 0327
A potent CB1 receptor antagonist
-
GC15327
Tetrahydromagnolol
二丙基联苯二醇,Magnolignan
An agonist of CB1 and CB2 and antagonist of GPR55
-
GC15528
(±)trans-2,5-bis-(3,4,5-Trimethoxyphenyl)-1,3-dioxolane
trans-BTP Dioxolane
A PAF receptor antagonist
-
GC11584
Butenoyl PAF
A PAF analog
-
GC13732
TG4-155
A brain penetrant EP2 antagonist
-
GC14445
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine
咪唑并二甲基吡啶
An angiotensin II receptor antagonist
-
GC10020
γ-Linolenic Acid methyl ester
r-亚麻酸甲酯,Methyl GLA,Methyl γ-Linolenate
A dietary ω-6 PUFA
-
GC12671
Angiotensin Fragment 1-7 (acetate)
A type 1 angiotensin II receptor agonist
-
GC14940
5-Methoxytryptamine
5-甲氧基色胺
-
GC13597
Pyrrolidino PAF C-16
A potent analog of PAF C-16
-
GC13752
Hexanolamino PAF C-16
A PAF analog
-
GC18125
DC260126
An FFAR1 (GPR40) antagonist
-
GC17224
AH 23848 (calcium salt)
Dual antagonist of TP and EP4 receptors
-
GC10028
(R)-SLV 319
The inactive enantiomer of SLV 319
-
GC15347
Bufuralol (hydrochloride)
丁呋洛尔盐酸盐,Ro 3-4787
An antagonist of β-adrenergic receptors
-
GC17757
1H-1-ethyl Candesartan Cilexetil
坎地沙坦EP杂质E
A potential impurity found in bulk preparations of candesartan cilexetil
-
GC14115
AVE-1625
屈那班,Drinabant
A potent CB1 receptor antagonist
-
GC18097
Arachidonoyl Serinol
A CB1 receptor agonist
-
GC10360
Lorglumide (sodium salt)
CR-1409 sodium salt
A selective antagonist of CCK1
-
GC15765
CYM 5520
A selective S1P2 receptor agonist
-
GC13315
ML-098
CID-7345532
A selective Rab7 activator
-
GC16414
ML-233
CID-46905036
A selective apelin receptor agonist
-
GC11453
ML-191
CCG-152883,CID-23612552
An antagonist of GPR55
-
GC10189
LY223982
CGS 23131,SKF 107324
A LTB4 receptor antagonist