GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC14317BMS CCR2 22CAS: 445479-97-0纯度: >99.00%
BMS CCR2 22 是一种有效、特异性和高亲和力的 CC 型趋化因子受体 2 (CCR2) 拮抗剂，具有出色的结合亲和力（结合 IC50 为 5.1 nM）和有效的功能拮抗作用（钙通量 IC50 为 18 nM，趋化性 IC50 为 1 nM） 。
- GC144337α,25-dihydroxy CholesterolCAS: 64907-22-8纯度: ≥95.00% / >99.50%
A potent and selective agonist of GPR183
- GC144452-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridineCAS: 133240-06-9
An angiotensin II receptor antagonist
- GC14463RX 821002 hydrochlorideCAS: 109544-45-8纯度: >98.50%
RX 821002 hydrochloride (RX821002 hydrochloride) 是一种高度选择性的 α 2-肾上腺素受体拮抗剂，几乎没有或没有咪唑啉拮抗剂作用。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC14279 | BIM 189 | 142062-55-3 | - | |
Bombesin antagonist | ||||
| GC14286 | [Ala17]-MCH | 359784-84-2 | >98.00% | |
An MCH-derived peptide and MCH receptor agonist | ||||
| GC14290 | SLV 320 | 251945-92-3 | >98.00% | |
An adenosine A1 receptor antagonist | ||||
| GC14293 | [Ala11,22,28]VIP | 291524-04-4 | >95.50% | |
agonist for the human VPAC1 receptor | ||||
| GC14300 | GPR120 Compound A | 1599477-75-4 | >99.00% | |
A selective GPR120/FFAR4 agonist | ||||
| GC14317 | BMS CCR2 22 | 445479-97-0 | >99.00% | |
BMS CCR2 22 是一种有效、特异性和高亲和力的 CC 型趋化因子受体 2 (CCR2) 拮抗剂，具有出色的结合亲和力（结合 IC50 为 5.1 nM）和有效的功能拮抗作用（钙通量 IC50 为 18 nM，趋化性 IC50 为 1 nM） 。 | ||||
| GC14347 | SB 228357 | 181629-93-6 | - | |
SB 228357 是一种选择性、有效的口服活性 5-HT2C/2B 受体拮抗剂，5-HT2A、5-HT2B 和 5-HT2C 的 pKi 值分别为 6.9、8.0 和 9.0。 | ||||
| GC14360 | Ozanimod (RPC1063) | 1306760-87-1 | >99.50% | |
An S1P 1 and S1P 5 agonist | ||||
| GC14369 | N6-Cyclopentyladenosine | 41552-82-3 | >98.50% | |
A selective A 1 R agonist | ||||
| GC14373 | GR 46611 | 185259-85-2 | - | |
GR 46611是一种5-HT1B和5-HT1D受体激动剂，可调节动物的摄食行为。 | ||||
| GC14374 | α-MSH | 581-05-5 | >98.00% | |
α -黑色素细胞刺激激素(α-MSH)是一种具有免疫调节特性的神经肽,由原黑素皮质素(POMC)翻译后加工产生。 | ||||
| GC14392 | SB 242084 | 181632-25-7 | >98.00% | |
Specific antagonist of 5-HT 2C | ||||
| GC14393 | BVD 10 | 262418-00-8 | - | |
NPY Y1 receptor antagonist,highly selective | ||||
| GC14408 | ML 154 | 1345964-89-7 | - | |
An NPSR antagonist | ||||
| GC14416 | BQ-3020 | 143113-45-5 | - | |
A peptide ET B receptor antagonist | ||||
| GC14419 | Bethanechol chloride | 590-63-6 | - | |
A muscarinic acetylcholine receptor agonist | ||||
| GC14423 | Motilin (human, porcine) | 52906-92-0 | >98.50% | |
内源性胃动素受体配体 | ||||
| GC14430 | JNJ 5207787 | 683746-68-1 | - | |
An antagonist of NPY receptor Y 2 | ||||
| GC14433 | 7α,25-dihydroxy Cholesterol | 64907-22-8 | ≥95.00% / >99.50% | |
A potent and selective agonist of GPR183 | ||||
| GC14445 | 2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine | 133240-06-9 | - | |
An angiotensin II receptor antagonist | ||||
| GC14455 | M617 | 860790-38-1 | - | |
M617 是一种选择性甘丙肽受体 1 (GAL1) 激动剂，对 GAL1 和 GAL2 的 Kis 分别为 0.23 和 5.71 nM。 | ||||
| GC14463 | RX 821002 hydrochloride | 109544-45-8 | >98.50% | |
RX 821002 hydrochloride (RX821002 hydrochloride) 是一种高度选择性的 α 2-肾上腺素受体拮抗剂，几乎没有或没有咪唑啉拮抗剂作用。 | ||||
| GC14467 | MA 2029 | 287206-61-5 | >99.00% | |
MA 2029 是一种选择性、口服活性和竞争性胃动素受体拮抗剂 (IC50\u003d4.9 nM)。 | ||||
| GC14468 | PSB 0739 | 1052087-90-7 | >98.50% / >98.00% | |
PSB 0739 是一种高亲和力、竞争性、非选择性血小板 P2Y12 受体拮抗剂，Ki 值为 24.9 nM。 | ||||