GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

研究方向

GPCR/G protein 相关产品(3377)

  • GC14478 structure
    GC14478LUF 6283
    CAS: 92933-48-7

    A partial agonist of GPR109A/HCA 2 receptors

  • GC14491 structure
    GC14491B-HT 920
    CAS: 36085-73-1
    纯度: >99.50%

    A potent agonist of D 2 receptors

  • GC14514 structure
    GC14514B-HT 933 dihydrochloride
    CAS: 36067-72-8

    An α 2 -AR agonist

  • GC14516 structure
    GC14516Mesulergine hydrochloride
    CAS: 72786-12-0

    5-HT2A and 2C receptor antagonist

  • GC14519 structure
    GC14519BX 471
    CAS: 217645-70-0
    纯度: >99.50%

    A selective CCR1 antagonist

  • GC14527 structure
    GC14527A 61603 hydrobromide
    CAS: 107756-30-9
    纯度: >98.00%

    An α 1A -adrenoceptor agonist

  • GC14533 structure
    GC14533Kynurenic acid
    CAS: 492-27-3
    纯度: >99.00% / >98.00%

    Kynurenic acid 是一种内源性色氨酸代谢物,是一种针对 NMDA、谷氨酸、α7 烟碱乙酰胆碱受体的广谱拮抗剂。

  • GC14535 structure
    GC14535PAF (C16)
    CAS: 74389-68-7
    纯度: >98.00%

    PAF(C16)是一种膜源磷脂,也是血小板活化因子和PAF G蛋白偶联受体(PAFR)的配体。

  • GC14554 structure
    GC14554J 113863
    CAS: 353791-85-2

    J 113863 是一种有效的选择性 CCR1 (CD18) 拮抗剂,对人和小鼠 CCR1 受体的 IC50 值分别为 0.9 nM 和 5.8 nM。

  • GC14555 structure
    GC14555LY341495
    CAS: 201943-63-7
    纯度: >99.00% / >98.50%

    Selective antagonist of mGluR2 and mGluR3

  • GC14565 structure
    GC14565SCH 58261
    CAS: 160098-96-4
    纯度: >99.50% / >98.00%

    SCH 58261是一种强效选择性非黄嘌呤类A2A腺苷受体拮抗剂,IC 50 值为15nM。

  • GC14583 structure
    GC14583R 59-022
    CAS: 93076-89-2
    纯度: 不显示

    R 59-022是一种二酰甘油激酶抑制剂(IC 50 = 2.8µM)。

  • GC14605 structure
    GC14605Nocistatin (human)
    CAS: 212609-11-5
    纯度: >97.00%

    Nocistatin (human) 阻断 nociceptin 诱导的异常性疼痛和痛觉过敏,并减轻由前列腺素 E2 引起的疼痛。

  • GC14607 structure
    GC146071-Methylpsilocin
    CAS: 1465-16-3

    5-HT2C agonist,potent and selective

  • GC14612 structure
    GC14612JNJ-31020028
    CAS: 1094873-14-9
    纯度: >98.00%

    An antagonist of NPY receptor Y 2

  • GC14625 structure
    GC14625RS 39604 hydrochloride
    CAS: 167710-87-4

    RS 39604 hydrochloride 是一种有效的、选择性的、具有口服活性的 5-HT4 受体拮抗剂,在豚鼠纹状体膜中的 pKi 为 9.1。

  • GC14626 structure
    GC14626MM-22
    CAS: 956605-71-3

    biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide

  • GC14629 structure
    GC14629Bombinakinin-GAP
    CAS: 573671-91-7

    Bioactive bradykinin-related peptide

  • GC14657 structure
    GC14657Rotundine
    CAS: 483-14-7
    纯度: >99.50%

    An antinociceptive alkaloid

  • GC14661 structure
    GC14661AM6545
    CAS: 1245626-05-4

    A peripherally restricted CB 1 receptor antagonist

  • GC14662 structure
    GC14662Litorin
    CAS: 55749-97-8

    A peptide with diverse biological activities

  • GC14674 structure
    GC14674CGH 2466 dihydrochloride
    CAS: 1177618-54-0

    adenosine receptor antagonist

  • GC14678 structure
    GC14678Sarafotoxin S6b
    CAS: 116303-65-2

    Sarafotoxin S6b 是一种血管收缩肽和非选择性内皮素受体激动剂。

  • GC14690 structure
    GC146902-Iodomelatonin
    CAS: 93515-00-5
    纯度: >99.00%

    A potent MT 1 receptor agonist