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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

Cat.No. 产品名称 Information
GC44247 Mozavaptan (hydrochloride)
莫扎伐普坦盐酸盐,OPC-31260 hydrochloride
A vasopressin V₂ receptor antagonist
GC44217 ML-184
CID2440433
A synthetic agonist of GPR55
GC44185 Metipranolol (hydrochloride)
Trimepranol
A β-AR antagonist
GC44169 Metaproterenol (hemisulfate)
硫酸奥西那林,Orciprenaline hemisulfate
A long-acting β₂-adrenergic receptor agonist
GC44096 LY293111
Etalocib; VML 295
A LTB₄ receptor antagonist
GC44021 L-826,266
A selective EP₃ antagonist
GC43999 Ketanserin (tartrate)
酒石酸酮色林,R41468 tartrate
A potent 5-HT₂ receptor antagonist
GC43932 JP-1302 (hydrochloride) An α_2C-adrenergic receptor antagonist
GC43926 Jatrorrhizine (chloride)
盐酸药根碱
An alkaloid with diverse biological activities
GC43888 Icatibant (acetate)
艾替班特乙酸盐,HOE 140 acetate
A synthetic peptide antagonist of the bradykinin B₂ receptor
GC43877 Hydroxy Bupropion
羟基1-(3-氯苯基)-2-[(1,1-二甲基乙基)氨基]-1-丙酮盐酸盐,Hydroxy Bupropion
Hydroxy Bupropion是bupropion的主要代谢产物，可抑制去甲肾上腺(NE)摄取，IC₅₀值为1.7μM。
GC43761 GLP-1 (1-37) (human, rat, mouse, bovine) (trifluoroacetate salt)
胰高血糖素样肽-1（GLP-1）,Glucagon-like Peptide-1
GLP-1 (1-37) (human, rat, mouse, bovine) (trifluoroacetate salt)是由肠道分泌的胰高血糖素样肽-1的全长前体。
GC43739 GAT228 An allosteric agonist of the CB₁ receptor
GC43666 Fingolimod
芬戈莫德; FTY720 free base
A fungal metabolite with immune modulating activities
GC43644 Exendin-4 (acetate)
醋酸艾塞那肽; Exenatide acetate
A GLP-1R agonist
GC43580 DX600 A peptide inhibitor of ACE2
GC43353 Cyproheptadine (hydrochloride hydrate)
盐酸赛庚啶半水合物
An antihistamine with antiserotonergic and anticholinergic activities
GC43347 Cyclopentolate (hydrochloride)
盐酸环喷托酯,DL-Cyclopentolate hydrochloride
A muscarinic receptor antagonist
GC43341 Cyclic GMP
鸟苷-3ˊ,5ˊ-环磷酸一钠盐

A second messenger
GC43276 CL 316,243 (disodium salt) CL 316,243 (disodium salt) 是一种高效的 β3 肾上腺素受体选择性激动剂，EC₅₀ 为 3 nM。它是一种有效的脂肪细胞脂解刺激剂，可增加棕色脂肪组织的产热和代谢率，具有治疗肥胖症、糖尿病和急迫性尿失禁的潜力。
GC43232 Cevimeline (hydrochloride)
盐酸西维美林; AF102B hydrochloride
Cevimeline (hydrochloride)是一种强效的直接作用muscarinic受体激动剂，具有口服生物利用度。
GC43210 CB-25 A stable analog of Δ⁹-THC
GC43163 CAY10508 A CB₁ inverse agonist
GC43137 Cangrelor (sodium salt)
坎格雷洛四钠盐,AR-C69931MX tetrasodium
An ATP analog with antithrombic properties
GC42927 BGC 20-1531 (hydrochloride)
PGN 1531
A potent and selective EP₄ receptor antagonist
GC42851 Arformoterol (tartrate)
酒石酸福莫特罗; (R,R)-Formoterol tartrate
A β₂-AR agonist
GC42831 AR420626 AR420626是一种口服活性、选择性的游离脂肪酸受体3(FFAR3)激动剂，EC₅₀值为2.2µM。
GC42817 Antileukinate Antileukinate是一种强效的α-chemokine受体结合抑制剂，可抑制Growth-related oncogene-α (GROα)与相关受体的结合。
GC42810 Angiotensin II (5-8) (human, rat, mouse) An endogenous angiotensin II fragment
GC42782 Amcinonide
安西奈德; CL-34699
A synthetic corticosteroid
GC42664 A-971432 A sphingosine-1-phosphate receptor 5 (S1P₅) agonist
GC42625 8-DY547-cGMP 通过结合环核苷酸激活，环核苷酸门控 (CNG) 离子通道介导光感受器和嗅觉细胞中的感觉信号转导。
GC42587 6α-Methylprednisolone 21-hemisuccinate
甲基泼尼松龙琥珀酸酯; Methylprednisolone hydrogen succinate
A prodrug form of methylprednisolone
GC42460 4-Nitrophenyl Phenylphosphonate
苯膦酸单-4-硝基苯酯
A 5′-nucleotide phosphodiesterase substrate
GC42011 1-Oleoyl Lysophosphatidic Acid
1-Oleoyl LPA, Oleoyl-sn-3-Glycerophosphate

A potent LPA receptor agonist
GC41883 12(S)-HHTrE
12(S)-HHTrE
An agonist of BLT₂
GC41668 (±)-Clopidogrel (hydrochloride) A prodrug of the platelet purinergic P2Y12 receptor antagonist
GC41442 Misoprostol (free acid)
米索前列醇酸
An EP₂, EP₃, and EP₄ receptor agonist
GC41327 Aaptamine Aaptamine 是一种从海绵 Aaptos aaptos 中分离出来的海绵类生物碱，是 α-肾上腺素受体的竞争性拮抗剂，以不依赖 p53 的方式激活 p21 启动子。
GC41311 CB-52 A stable analog of Δ⁹-THC and AEA
GC41229 Latanoprost (free acid)
拉坦前列腺素(游离酸)
Potent FP receptor agonist
GC41087 PSB-SB1202 A CB₁ and CB₂ receptor agonist
GC40854 Latanoprost Lactone Diol
拉坦前列腺素内酯二醇
An intermediate in the synthesis of latanoprost
GC40787 γ-Linolenic Acid ethyl ester
γ-亚麻酸乙酯
Esterified form of γ-linolenic acid
GC40775 Dexamethasone
地塞米松; Hexadecadrol; Prednisolone F
地塞米松是糖皮质激素家族的一员，可以保护软骨结构和功能免受关节炎相关变化的影响，包括基质丢失、炎症和软骨活力。
GC40771 Fluorometholone
氟米龙
A synthetic glucocorticoid
GC40750 Agnuside
穗花牡荆苷; Agnoside
An iridoid glycoside with diverse biological activities
GC40637 BAR501 A selective GP-BAR1 agonist
GC40591 Prostaglandin F2β
同分异构体(物),同质异能素
The 9β-hydroxy stereoisomer of PGF_2α
GC40406 2-Oleoyl Glycerol
2-十八烯酸单甘油酯；2-甘油单油酸酯
A natural monoacylglycerol