GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

研究方向

GPCR/G protein 相关产品(3377)

GC10308 Apelin-36 (rat, mouse)
CAS: 230299-95-3
Mature peptide and APJ agonist
GC10310 SB 206553 hydrochloride
CAS: 1197334-04-5
A 5-HT 2C and 5-HT 2B receptor antagonist
GC10311 Liraglutide
CAS: 204656-20-2
纯度: >99.50% / >99.00% / >98.00%
利拉鲁肽是一种高效、长效的 GLP-1 受体激动剂 (EC50 = 61 pM)，其氨基酸序列与人 GLP-1 有 97% 的同一性 .用 PA/LPS 处理的肝细胞中的活细胞数量显着减少，利拉鲁肽以浓度依赖性方式逆转细胞活力的下降。
GC10320 MRS 1706
CAS: 264622-53-9
纯度: >98.00%
A selective adenosine A 2B receptor inverse agonist
GC10328 TT 232
CAS: 147159-51-1
A synthetic peptide derivative of somatostatin
GC10357 Metergoline
CAS: 17692-51-2
纯度: >99.50%
A serotonin receptor antagonist
GC10360 Lorglumide (sodium salt)
CAS: 1021868-76-7
纯度: >99.50%
A selective antagonist of CCK 1
GC10401 SB 204070
CAS: 148688-01-1
Potent and selective 5-HT4 receptor antagonist
GC10432 IT1t dihydrochloride
CAS: 1092776-63-0
纯度: >99.50%
A CXCR4 antagonist
GC10433 ML-178
CAS: 1355026-47-9
A selective S1P 4 agonist
GC10434 Triamcinolone
CAS: 124-94-7
A synthetic glucocorticoid
GC10437 [(pF)Phe4]Nociceptin(1-13)NH2
CAS: 380620-88-2
[(pF)Phe4]Nociceptin(1-13)NH2 是一种高效的选择性 NOP 受体 (OP4) 激动剂，pKi 为 10.68，pEC50 为 9.31。
GC10475 Proxyphylline
CAS: 603-00-9
纯度: >98.50%
A methylxanthine derivative and an adenosine receptor antagonist
GC10483 CID 2745687
CAS: 264233-05-8
纯度: >95.00%
An antagonist of GPR35
GC10494 ADX-47273
CAS: 851881-60-2
纯度: >99.00%
A positive allosteric modulator of mGluR5
GC10495 EMD 281014 hydrochloride
CAS: 443144-27-2
5-HT2A antagonist
GC10508 Solifenacin hydrochloride
CAS: 180468-39-7
纯度: >99.00%
Solifenacin hydrochloride (YM905 hydrochloride) 是一种毒蕈碱受体拮抗剂，对 M1、M2 和 M3 受体的 pKis 分别为 7.6、6.9 和 8.0。
GC10509 Cladribine
CAS: 4291-63-8
纯度: >99.50%
A nucleoside analog and prodrug form of 2-CdATP
GC10514 RWJ 52353
CAS: 245744-10-9
An α 2D -adrenergic receptor agonist
GC10527 PCA 4248
CAS: 123875-01-4
PAF antagonist
GC10528 Salirasib
CAS: 162520-00-5
纯度: >98.00%
A Ras inhibitor with anti-cancer and anti-atherogenic activity
GC10535 S 32212 hydrochloride
CAS: 847871-78-7
An inverse agonist of 5-HT 2C receptors
GC10536 Pronethalol hydrochloride
CAS: 51-02-5
Pronethalol ((±)-Pronethalo) 是一种非选择性 β-肾上腺素能拮抗剂。
GC10548 CP 376395 hydrochloride
CAS: 1013933-37-3
A CRF 1 antagonist

分类产品列表
货号	产品名称	CAS号	纯度
GC10308	Apelin-36 (rat, mouse)	230299-95-3	-
GC10308	Mature peptide and APJ agonist
GC10310	SB 206553 hydrochloride	1197334-04-5	-
GC10310	A 5-HT 2C and 5-HT 2B receptor antagonist
GC10311	Liraglutide	204656-20-2	>99.50% / >99.00% / >98.00%
GC10311	利拉鲁肽是一种高效、长效的 GLP-1 受体激动剂 (EC50 = 61 pM)，其氨基酸序列与人 GLP-1 有 97% 的同一性 .用 PA/LPS 处理的肝细胞中的活细胞数量显着减少，利拉鲁肽以浓度依赖性方式逆转细胞活力的下降。
GC10320	MRS 1706	264622-53-9	>98.00%
GC10320	A selective adenosine A 2B receptor inverse agonist
GC10328	TT 232	147159-51-1	-
GC10328	A synthetic peptide derivative of somatostatin
GC10357	Metergoline	17692-51-2	>99.50%
GC10357	A serotonin receptor antagonist
GC10360	Lorglumide (sodium salt)	1021868-76-7	>99.50%
GC10360	A selective antagonist of CCK 1
GC10401	SB 204070	148688-01-1	-
GC10401	Potent and selective 5-HT4 receptor antagonist
GC10432	IT1t dihydrochloride	1092776-63-0	>99.50%
GC10432	A CXCR4 antagonist
GC10433	ML-178	1355026-47-9	-
GC10433	A selective S1P 4 agonist
GC10434	Triamcinolone	124-94-7	-
GC10434	A synthetic glucocorticoid
GC10437	[(pF)Phe4]Nociceptin(1-13)NH2	380620-88-2	-
GC10437	[(pF)Phe4]Nociceptin(1-13)NH2 是一种高效的选择性 NOP 受体 (OP4) 激动剂，pKi 为 10.68，pEC50 为 9.31。
GC10475	Proxyphylline	603-00-9	>98.50%
GC10475	A methylxanthine derivative and an adenosine receptor antagonist
GC10483	CID 2745687	264233-05-8	>95.00%
GC10483	An antagonist of GPR35
GC10494	ADX-47273	851881-60-2	>99.00%
GC10494	A positive allosteric modulator of mGluR5
GC10495	EMD 281014 hydrochloride	443144-27-2	-
GC10495	5-HT2A antagonist
GC10508	Solifenacin hydrochloride	180468-39-7	>99.00%
GC10508	Solifenacin hydrochloride (YM905 hydrochloride) 是一种毒蕈碱受体拮抗剂，对 M1、M2 和 M3 受体的 pKis 分别为 7.6、6.9 和 8.0。
GC10509	Cladribine	4291-63-8	>99.50%
GC10509	A nucleoside analog and prodrug form of 2-CdATP
GC10514	RWJ 52353	245744-10-9	-
GC10514	An α 2D -adrenergic receptor agonist
GC10527	PCA 4248	123875-01-4	-
GC10527	PAF antagonist
GC10528	Salirasib	162520-00-5	>98.00%
GC10528	A Ras inhibitor with anti-cancer and anti-atherogenic activity
GC10535	S 32212 hydrochloride	847871-78-7	-
GC10535	An inverse agonist of 5-HT 2C receptors
GC10536	Pronethalol hydrochloride	51-02-5	-
GC10536	Pronethalol ((±)-Pronethalo) 是一种非选择性 β-肾上腺素能拮抗剂。
GC10548	CP 376395 hydrochloride	1013933-37-3	-
GC10548	A CRF 1 antagonist