GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC10181L-803,087 trifluoroacetateCAS: 217480-26-7纯度: >96.00%
L-803,087 trifluoroacetate 是一种有效的选择性生长抑素 sst4 受体激动剂，Ki 为 0.7 nM。
- GC10257Losartan Potassium (DuP 753)CAS: 124750-99-8纯度: >99.50%
Losartan Potassium (DuP 753)是一种血管紧张素II受体拮抗剂（IC 50 =20nM）。
- GC10283γ-Linolenic AcidCAS: 506-26-3纯度: >98.00% / >98.50%
γ-Linolenic Acid是一种来源于琉璃苣油的口服ω-6多不饱和脂肪酸，可作为β-分泌酶（BACE1）的特异性抑制剂，IC 50 值为7.6×10 −5 mol/L，K i 值为3.5×10 −5 mol/L。
- GC10287Ibutamoren MesylateCAS: 159752-10-0纯度: >98.00%
A growth hormone secretagogue and ghrelin receptor agonist
- GC10291SCH 79797 dihydrochlorideCAS: 1216720-69-2纯度: >98.50% / >98.00%
SCH 79797 dihydrochloride是一种高效的、具有选择性的非肽类蛋白酶激活受体 1（PAR1）拮抗剂，其IC 50 值为70nM，Ki值为35nM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10161 | [D-Lys3]-GHRP-6 | 136054-22-3 | - | |
[D-Lys3]-GHRP-6是一种高选择性的生长激素促分泌素受体（GHSR）拮抗剂，IC 50 值为0.9μM。 | ||||
| GC10167 | CGP 71683 hydrochloride | 192322-50-2 | >99.00% | |
An antagonist of NPY receptor Y 5 | ||||
| GC10175 | GW 803430 | 515141-51-2 | >98.00% | |
An antagonist of MCH 1 | ||||
| GC10181 | L-803,087 trifluoroacetate | 217480-26-7 | >96.00% | |
L-803,087 trifluoroacetate 是一种有效的选择性生长抑素 sst4 受体激动剂，Ki 为 0.7 nM。 | ||||
| GC10189 | LY223982 | 117423-74-2 | >99.00% | |
A LTB 4 receptor antagonist | ||||
| GC10197 | AH 11110 hydrochloride | 179388-65-9 | - | |
α1B-AR ligand,subtype-selective | ||||
| GC10202 | MRS 1334 | 192053-05-7 | - | |
MRS 1334 是一种有效的选择性人腺苷 A3 受体拮抗剂，对 hA3、rA1、rA2A 的 Kis 分别为 2.69 nM、\u003e100 nM、\u003e100 nM。 | ||||
| GC10205 | Arvanil | 128007-31-8 | >98.00% | |
A structural analog of capsaicin with analgesic activity | ||||
| GC10207 | INCB3344 | 1262238-11-8 | >99.50% | |
An antagonist of CCR2 | ||||
| GC10219 | AF-DX 116 | 102394-31-0 | >99.50% | |
A muscarinic M 2 receptor antagonist | ||||
| GC10242 | Loxapine Succinate | 27833-64-3 | >99.50% | |
An atypical antipsychotic drug | ||||
| GC10246 | TC-G 1004 | 1061747-72-5 | - | |
TC-G 1004（化合物 16j）是一种具有口服活性的 A2A 腺苷受体拮抗剂，对 hA2A 和 hA1 的 Ki 值分别为 0.44 nM 和 80 nM。 | ||||
| GC10255 | Lys-[Des-Arg9]Bradykinin | 71800-36-7 | - | |
bradykinin B1 receptor agonist | ||||
| GC10257 | Losartan Potassium (DuP 753) | 124750-99-8 | >99.50% | |
Losartan Potassium (DuP 753)是一种血管紧张素II受体拮抗剂（IC 50 =20nM）。 | ||||
| GC10264 | Arecoline hydrobromide | 300-08-3 | >99.50% | |
Muscarinic acetylcholine receptor agonist | ||||
| GC10265 | Manumycin A | 52665-74-4 | >98.00% | |
A farnesyltransferase inhibitor with antitumor activity | ||||
| GC10266 | BAY-u 9773 | 154978-38-8 | - | |
Antagonist of CysLT1/CysLT2 receptors | ||||
| GC10271 | [Ac-Tyr1,D-Phe2]GRF 1-29, amide (human) | 93965-89-0 | - | |
VIP receptor antagonist | ||||
| GC10283 | γ-Linolenic Acid | 506-26-3 | >98.00% / >98.50% | |
γ-Linolenic Acid是一种来源于琉璃苣油的口服ω-6多不饱和脂肪酸，可作为β-分泌酶（BACE1）的特异性抑制剂，IC 50 值为7.6×10 −5 mol/L，K i 值为3.5×10 −5 mol/L。 | ||||
| GC10284 | Apelin-13 | 217082-58-1 | >98.00% | |
Apelin-13 是一种肽，被称为 G 蛋白偶联受体 APJ 的配体。 | ||||
| GC10287 | Ibutamoren Mesylate | 159752-10-0 | >98.00% | |
A growth hormone secretagogue and ghrelin receptor agonist | ||||
| GC10291 | SCH 79797 dihydrochloride | 1216720-69-2 | >98.50% / >98.00% | |
SCH 79797 dihydrochloride是一种高效的、具有选择性的非肽类蛋白酶激活受体 1（PAR1）拮抗剂，其IC 50 值为70nM，Ki值为35nM。 | ||||
| GC10300 | Diphenidol HCl | 3254-89-5 | >99.00% | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC10304 | L-798,106 | 244101-02-8 | >99.50% | |
A selective EP 3 receptor antagonist | ||||