GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC16836NaftopidilCAS: 57149-07-2纯度: >98.50%
Naftopidil (KT-611) 是一种选择性 alpha1-adrenoceptor 拮抗剂，对克隆的人 α1a-、α1b- 和 α1d-adrenoceptor 亚型的 Kis 分别为 3.7 nM、20 nM 和 1.2 nM。
- GC16839Guanabenz AcetateCAS: 23256-50-0纯度: 99.45%
Guanabenz (Acetate) (BR-750) 是一种 alpha-2 选择性肾上腺素能激动剂，用作抗高血压药。
- GC16936OlmesartanCAS: 144689-24-7纯度: >98.00%
An AT 1 receptor antagonist and active metabolite of olmesartan medoxomil
- GC17088SA 4503 dihydrochlorideCAS: 165377-44-6纯度: >98.00%
SA 4503 dihydrochloride是一种具有高效选择性的σ1受体激动剂，IC 50 值为17nM。
- GC172182-fluoro Palmitic AcidCAS: 16518-94-8纯度: >98.00%
Inhibitor of sphingosine biosynthesis and long-chain acyl-CoA synthetase
- GC17244Calcium-Sensing Receptor Antagonists ICAS: 478963-79-0纯度: >99.50%
钙敏感受体拮抗剂 I 是钙敏感甲状旁腺激素受体的拮抗剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16836 | Naftopidil | 57149-07-2 | >98.50% | |
Naftopidil (KT-611) 是一种选择性 alpha1-adrenoceptor 拮抗剂，对克隆的人 α1a-、α1b- 和 α1d-adrenoceptor 亚型的 Kis 分别为 3.7 nM、20 nM 和 1.2 nM。 | ||||
| GC16839 | Guanabenz Acetate | 23256-50-0 | 99.45% | |
Guanabenz (Acetate) (BR-750) 是一种 alpha-2 选择性肾上腺素能激动剂，用作抗高血压药。 | ||||
| GC16862 | Zibotentan (ZD4054) | 186497-07-4 | >98.00% | |
A selective ET A receptor antagonist | ||||
| GC16871 | Perindopril | 82834-16-0 | - | |
An orally active ACE inhibitor | ||||
| GC16873 | N,N-Dimethylsphingosine | 119567-63-4 | >98.00% | |
A SPHK inhibitor | ||||
| GC16922 | Kobe0065 | 436133-68-5 | >99.50% | |
A selective Ras inhibitor | ||||
| GC16936 | Olmesartan | 144689-24-7 | >98.00% | |
An AT 1 receptor antagonist and active metabolite of olmesartan medoxomil | ||||
| GC16943 | NPS-2143 | 284035-33-2 | >99.00% | |
NPS-2143 是一种钙化药物，可作为钙敏感受体 (CaSR) 的拮抗剂，从而刺激甲状旁腺激素的释放。 | ||||
| GC16946 | CYM 5541 | 945128-26-7 | >98.00% | |
A selective agonist of S1P 3 | ||||
| GC17004 | Sphingosine-1-phosphate | 26993-30-6 | >98.00% | |
1-磷酸鞘氨醇是细胞膜鞘脂的代谢产物。 | ||||
| GC17018 | AMD-070 hydrochloride | 880549-30-4 | - | |
CXCR4 antagonist,potent and selective | ||||
| GC17019 | TC-SP 14 | 1257093-40-5 | - | |
TC-SP 14 (compound 14) 是一种口服有效的 S1P1 激动剂 (EC50 = 0.042 μM)，在 S1P3 (EC50 = 3.47 μM) 的活性最低。 | ||||
| GC17053 | Eletriptan HBr | 177834-92-3 | >98.00% | |
An agonist of 5-HT 1B and 5-HT 1D receptors | ||||
| GC17061 | Dapoxetine HCl | 129938-20-1 | >99.50% | |
An Analytical Reference Standard | ||||
| GC17081 | Detomidine HCl | 90038-01-0 | >99.50% | |
An α 2 -adrenoceptor agonist | ||||
| GC17088 | SA 4503 dihydrochloride | 165377-44-6 | >98.00% | |
SA 4503 dihydrochloride是一种具有高效选择性的σ1受体激动剂，IC 50 值为17nM。 | ||||
| GC17130 | BRL-54443 | 57477-39-1 | >99.00% | |
A potent agonist of 5-HT 1E and 5-HT 1F | ||||
| GC17138 | LY310762 | 192927-92-7 | >98.00% | |
A 5-HT 1D antagonist | ||||
| GC17149 | 4-CMTB | 300851-67-6 | >99.00% | |
4-CMTB是一种选择性的游离脂肪酸受体2（FFA2/GPR43）激动剂和正变构调节剂。 | ||||
| GC17197 | Detomidine | 76631-46-4 | - | |
Detomidine 是一种咪唑衍生物，是一种有效的 α2-肾上腺素能激动剂。 | ||||
| GC17205 | CP-945598 HCl | 686347-12-6 | - | |
A selective CB 1 receptor antagonist | ||||
| GC17218 | 2-fluoro Palmitic Acid | 16518-94-8 | >98.00% | |
Inhibitor of sphingosine biosynthesis and long-chain acyl-CoA synthetase | ||||
| GC17244 | Calcium-Sensing Receptor Antagonists I | 478963-79-0 | >99.50% | |
钙敏感受体拮抗剂 I 是钙敏感甲状旁腺激素受体的拮抗剂。 | ||||
| GC17259 | Rimonabant | 168273-06-1 | - | |
A potent and selective CB 1 receptor antagonist | ||||