GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

研究方向

GPCR/G protein 相关产品(3377)

GC32439 Ferulic acid sodium (Sodium ferulate)
CAS: 24276-84-4
纯度: >99.00%
A phenol with diverse biological activities
GC32453 Lixivaptan (VPA-985)
CAS: 168079-32-1
纯度: >99.50%
A nonpeptide vasopressin V 2 receptor antagonist
GC32463 Terlipressin
CAS: 14636-12-5
A prodrug form of lysipressin
GC32464 MK-0354
CAS: 851776-28-8
纯度: >99.00%
MK-0354是特异性的GPR109a受体激动剂,作用于hGPR109a/mGPR109a,EC50分别为1.65μM和1.08μM,对GPR109b没有作用效果。
GC32476 Ralinepag (APD811)
CAS: 1187856-49-0
纯度: >99.50%
An IP receptor agonist
GC32478 Pirmenol hydrochloride (Cl-845)
CAS: 61477-94-9
纯度: >98.00%
A class I antiarrhythmic agent
GC32479 Sparsentan (RE-021)
CAS: 254740-64-2
纯度: >98.50%
A dual antagonist of AT 1 and ET A
GC32481 Vincamine
CAS: 1617-90-9
纯度: >99.50%
A plant alkaloid with vasodilator effects
GC32485 Moxisylyte hydrochloride (Thymoxamine hydrochloride)
CAS: 964-52-3
纯度: >99.50%
Moxisylyte hydrochloride (thymoxamine) is an alpha-adrenergic blocking agent used for the treatment of Raynaud's disease.
GC32494 Penbutolol sulfate ((-)-Terbuclomine)
CAS: 38363-32-5
纯度: >99.00%
A β-adrenergic and 5-HT 1A receptor antagonist
GC32507 Tasosartan (WAY-ANA 756)
CAS: 145733-36-4
纯度: >99.00%
An AT 2 receptor antagonist
GC32511 Naftidrofuryl oxalate (Nafronyl oxalate salt)
CAS: 3200-06-4
纯度: >98.00%
Nafronyl oxalate salt is the oxalate salt form of nafronyl, which is a selective antagonist of 5-HT2 receptors and a vasodilator used in the management of peripheral and cerebral vascular disorders.
GC32512 Indanidine
CAS: 85392-79-6
Indanidine是一种α-肾上腺素能激动剂。
GC32516 Amezinium methylsulfate (Amezinium metilsulfate)
CAS: 30578-37-1
纯度: >98.50%
Amezinium is a sympathomimetic used for its vasopressor effects in the treatment of hypotensive states. It is a MAO inhibitor, antagonizes the response to tyramine and blocks neuronal uptake of noradrenaline.
GC32523 (±)-Befunolol
CAS: 39552-01-7
(±)-Befunolol是一种β-肾上腺素能受体阻断剂。
GC32528 Ro 46-2005
CAS: 150725-87-4
纯度: >98.00%
Ro46-2005是一种新型非肽类内皮素拮抗剂,抑制人血管平滑肌细胞(ETA受体),IC50分别为220nM。
GC32530 Pratosartan (FW 7203)
CAS: 153804-05-8
Pratosartan (FW 7203) 是一种选择性血管紧张素 II 受体拮抗剂。
GC32532 Pamatolol
CAS: 59110-35-9
Pamatolol是一种心选择性的beta-adrenoceptor拮抗剂，没有拟交感活性。
GC32536 Elisartan (HN 65021)
CAS: 149968-26-3
Elisartan (HN 65021) 是一种具有口服活性的血管紧张素 II AT1 受体拮抗剂 HN-12206 的非肽前体药物，具有抗高血压活性。
GC32538 Pronethalol ((±)-Pronethalo)
CAS: 54-80-8
纯度: >99.00%
Pronethalol ((±)-Pronethalo) ((±)-Pronethalo) 是一种非选择性的 β-肾上腺素能拮抗剂。
GC32540 Etersalate (Eterylate)
CAS: 62992-61-4
Etersalate (Eterylate) 抑制血小板功能并降低血栓素 A2 (TXA2) 水平。
GC32542 Cicloprolol hydrochloride
CAS: 63686-79-3
Cicloprolol是部分β1-肾上腺素能受体(β1-adrenoceptor)激动剂。
GC32543 OPC-28326
CAS: 167626-17-7
OPC-28326是一种外周血管扩张药，同时为α2-adrenergicreceptor的拮抗剂，对α2A-，α2B-和α2C肾上腺素受体的Ki值分别为2040，285和55 nM。
GC32547 Ecastolol
CAS: 77695-52-4
Ecastolol是一种betaadrenergicreceptor拮抗剂，具有防心绞痛的作用。

分类产品列表
货号	产品名称	CAS号	纯度
GC32439	Ferulic acid sodium (Sodium ferulate)	24276-84-4	>99.00%
GC32439	A phenol with diverse biological activities
GC32453	Lixivaptan (VPA-985)	168079-32-1	>99.50%
GC32453	A nonpeptide vasopressin V 2 receptor antagonist
GC32463	Terlipressin	14636-12-5	-
GC32463	A prodrug form of lysipressin
GC32464	MK-0354	851776-28-8	>99.00%
GC32464	MK-0354是特异性的GPR109a受体激动剂,作用于hGPR109a/mGPR109a,EC50分别为1.65μM和1.08μM,对GPR109b没有作用效果。
GC32476	Ralinepag (APD811)	1187856-49-0	>99.50%
GC32476	An IP receptor agonist
GC32478	Pirmenol hydrochloride (Cl-845)	61477-94-9	>98.00%
GC32478	A class I antiarrhythmic agent
GC32479	Sparsentan (RE-021)	254740-64-2	>98.50%
GC32479	A dual antagonist of AT 1 and ET A
GC32481	Vincamine	1617-90-9	>99.50%
GC32481	A plant alkaloid with vasodilator effects
GC32485	Moxisylyte hydrochloride (Thymoxamine hydrochloride)	964-52-3	>99.50%
GC32485	Moxisylyte hydrochloride (thymoxamine) is an alpha-adrenergic blocking agent used for the treatment of Raynaud's disease.
GC32494	Penbutolol sulfate ((-)-Terbuclomine)	38363-32-5	>99.00%
GC32494	A β-adrenergic and 5-HT 1A receptor antagonist
GC32507	Tasosartan (WAY-ANA 756)	145733-36-4	>99.00%
GC32507	An AT 2 receptor antagonist
GC32511	Naftidrofuryl oxalate (Nafronyl oxalate salt)	3200-06-4	>98.00%
GC32511	Nafronyl oxalate salt is the oxalate salt form of nafronyl, which is a selective antagonist of 5-HT2 receptors and a vasodilator used in the management of peripheral and cerebral vascular disorders.
GC32512	Indanidine	85392-79-6	-
GC32512	Indanidine是一种α-肾上腺素能激动剂。
GC32516	Amezinium methylsulfate (Amezinium metilsulfate)	30578-37-1	>98.50%
GC32516	Amezinium is a sympathomimetic used for its vasopressor effects in the treatment of hypotensive states. It is a MAO inhibitor, antagonizes the response to tyramine and blocks neuronal uptake of noradrenaline.
GC32523	(±)-Befunolol	39552-01-7	-
GC32523	(±)-Befunolol是一种β-肾上腺素能受体阻断剂。
GC32528	Ro 46-2005	150725-87-4	>98.00%
GC32528	Ro46-2005是一种新型非肽类内皮素拮抗剂,抑制人血管平滑肌细胞(ETA受体),IC50分别为220nM。
GC32530	Pratosartan (FW 7203)	153804-05-8	-
GC32530	Pratosartan (FW 7203) 是一种选择性血管紧张素 II 受体拮抗剂。
GC32532	Pamatolol	59110-35-9	-
GC32532	Pamatolol是一种心选择性的beta-adrenoceptor拮抗剂，没有拟交感活性。
GC32536	Elisartan (HN 65021)	149968-26-3	-
GC32536	Elisartan (HN 65021) 是一种具有口服活性的血管紧张素 II AT1 受体拮抗剂 HN-12206 的非肽前体药物，具有抗高血压活性。
GC32538	Pronethalol ((±)-Pronethalo)	54-80-8	>99.00%
GC32538	Pronethalol ((±)-Pronethalo) ((±)-Pronethalo) 是一种非选择性的 β-肾上腺素能拮抗剂。
GC32540	Etersalate (Eterylate)	62992-61-4	-
GC32540	Etersalate (Eterylate) 抑制血小板功能并降低血栓素 A2 (TXA2) 水平。
GC32542	Cicloprolol hydrochloride	63686-79-3	-
GC32542	Cicloprolol是部分β1-肾上腺素能受体(β1-adrenoceptor)激动剂。
GC32543	OPC-28326	167626-17-7	-
GC32543	OPC-28326是一种外周血管扩张药，同时为α2-adrenergicreceptor的拮抗剂，对α2A-，α2B-和α2C肾上腺素受体的Ki值分别为2040，285和55 nM。
GC32547	Ecastolol	77695-52-4	-
GC32547	Ecastolol是一种betaadrenergicreceptor拮抗剂，具有防心绞痛的作用。