GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC17549[Nphe1]Nociceptin(1-13)NH2CAS: 267234-08-2
[Nphe1]Nociceptin(1-13)NH2 是一种新型的 nociceptin/orphanin FQ (NC) 内源性配体，是一种选择性和竞争性的 ociceptin 受体拮抗剂，没有任何残留的激动剂活性。
- GC17570Galanin (1-15) (porcine, rat)CAS: 112747-70-3
N-terminal galanin fragment used to mediate central cardiovascular effects
- GC17736AnisodamineCAS: 55869-99-3纯度: >98.00%
Anisodamine (6-Hydroxyhyoscyamine) 是一种颠茄生物碱，是一种非亚型选择性毒蕈碱，也是一种烟碱型胆碱受体拮抗剂。
- GC17744[Ala1,3,11,15]-EndothelinCAS: 121204-87-3
[Ala1,3,11,15]-Endothelin是一种经过修饰的Endothelin-1线性类似物，特点在于将原始序列中第1，3，11，15位的氨基酸替换为Alanine。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC17547 | MEN 10376 | 135306-85-3 | - | |
An NK 2 receptor antagonist | ||||
| GC17549 | [Nphe1]Nociceptin(1-13)NH2 | 267234-08-2 | - | |
[Nphe1]Nociceptin(1-13)NH2 是一种新型的 nociceptin/orphanin FQ (NC) 内源性配体，是一种选择性和竞争性的 ociceptin 受体拮抗剂，没有任何残留的激动剂活性。 | ||||
| GC17570 | Galanin (1-15) (porcine, rat) | 112747-70-3 | - | |
N-terminal galanin fragment used to mediate central cardiovascular effects | ||||
| GC17596 | Netupitant | 290297-26-6 | >99.50% | |
An NK 1 receptor antagonist | ||||
| GC17617 | Tetradecyl Phosphonate | 4671-75-4 | - | |
A stable pan-antagonist at LPA receptors | ||||
| GC17626 | PG 931 | 667430-81-1 | - | |
PG 931 是 SHU 9119 的类似物，是一种有效的黑皮质素 4 (MC4) 受体 (IC50\u003d0.58 nM) 激动剂，比对 hMC3R (IC50\u003d55 nM) 或 hMC5R (IC50\u003d2.4 nM) 更具选择性。 | ||||
| GC17653 | Levobetaxolol HCl | 116209-55-3 | >98.00% | |
A β1-adrenergic receptor antagonist | ||||
| GC17664 | FR 139317 | 142375-60-8 | - | |
highly potent and selective ETA endothelin receptor antagonist | ||||
| GC17666 | Xamoterol hemifumarate | 73210-73-8 | >98.00% | |
A β 1 -adrenergic receptor partial agonist | ||||
| GC17668 | L-817,818 | 217480-27-8 | - | |
L-817,818 是一种有效的、亚型选择性的生长抑素受体激动剂。 | ||||
| GC17699 | O-1821 | 35482-50-9 | >97.00% | |
An analog of O-1918, a selective antagonist of a non-CB 1 /CB 2 receptor | ||||
| GC17706 | R-96544 hydrochloride | 167144-79-8 | - | |
5-HT2 receptor antagonist | ||||
| GC17714 | PNU 22394 hydrochloride | 15923-42-9 | - | |
5-HT2C agonist and partial 5-HT2A/5-HT2B agonist | ||||
| GC17717 | CGP 12177 hydrochloride | 64208-32-8 | >98.00% | |
β1/β2-AR拮抗剂，β3 AR部分激动剂 | ||||
| GC17719 | 5-trans U-46619 | 330796-58-2 | - | |
An isomer of U-46619 | ||||
| GC17720 | W123 | 1345982-24-2 | >98.00% | |
Antagonist of spingosine 1-phosphate type 1 receptor | ||||
| GC17721 | IPAG | 193527-91-2 | - | |
IPAG 是一种有效的 sigma-1 受体拮抗剂，pKi 为 4.3。 IPAG 诱导细胞凋亡。 | ||||
| GC17734 | Pindolol | 13523-86-9 | >99.50% / >99.00% | |
A β 1 - and β 2 -AR antagonist | ||||
| GC17736 | Anisodamine | 55869-99-3 | >98.00% | |
Anisodamine (6-Hydroxyhyoscyamine) 是一种颠茄生物碱，是一种非亚型选择性毒蕈碱，也是一种烟碱型胆碱受体拮抗剂。 | ||||
| GC17740 | WB 4101 hydrochloride | 2170-58-3 | - | |
An α-AR antagonist | ||||
| GC17742 | NF 340 | 202982-98-7 | - | |
NF 340 是一种有效的选择性 P2Y11 受体拮抗剂。 | ||||
| GC17744 | [Ala1,3,11,15]-Endothelin | 121204-87-3 | - | |
[Ala1,3,11,15]-Endothelin是一种经过修饰的Endothelin-1线性类似物，特点在于将原始序列中第1，3，11，15位的氨基酸替换为Alanine。 | ||||
| GC17745 | MK 212 hydrochloride | 61655-58-1 | - | |
A 5-HT 2C receptor agonist | ||||
| GC17756 | PSB 1115 | 152529-79-8 | - | |
PSB 1115是一种选择性A2B腺苷受体拮抗剂。 | ||||