GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC16655VU 0357017 hydrochlorideCAS: 1135242-13-5纯度: >99.00%
An M 1 muscarinic acetylcholine receptor agonist
- GC16668[Des-octanoyl]-Ghrelin (rat)CAS: 307950-60-3
Non-acylated, major circulating isoform of ghrelin
- GC16673N-Formyl-Met-Leu-PheCAS: 59880-97-6纯度: >99.50%
N-Formyl-Met-Leu-Phe是一种内源性趋化肽，也是甲酰肽受体1（FPR1）的激动剂，Ki值为38 nM。
- GC16745Orexin B (mouse)CAS: 202801-92-1纯度: >98.50%
Orexin B (mouse) (Rat orexin B) 是 Orexin 受体的内源性激动剂，对 OX1 和 OX2 的 Kis 分别为 420 和 36 nM。
- GC16791Benztropine mesylateCAS: 132-17-2纯度: >99.50%
An M 1 muscarinic acetylcholine receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16644 | JTE 907 | 282089-49-0 | - | |
A selective CB 2 receptor inverse agonist | ||||
| GC16646 | GLP-2(1-33) (human) | 223460-79-5 | >99.00% | |
GLP-2(1-33) (human)是一种内分泌激素，由肠道L细胞在营养摄入后释放。 | ||||
| GC16650 | NBI 35965 hydrochloride | 603151-83-3 | >95.00% | |
A selective CRF 1 antagonist | ||||
| GC16653 | CP 94253 hydrochloride | 845861-39-4 | - | |
A 5-HT 1B receptor agonist | ||||
| GC16655 | VU 0357017 hydrochloride | 1135242-13-5 | >99.00% | |
An M 1 muscarinic acetylcholine receptor agonist | ||||
| GC16660 | Ponesimod | 854107-55-4 | >98.00% | |
A potent S1P 1 receptor agonist | ||||
| GC16663 | (±)-4-hydroxy Propranolol (hydrochloride) | 14133-90-5 | - | |
An active metabolite of propranolol | ||||
| GC16668 | [Des-octanoyl]-Ghrelin (rat) | 307950-60-3 | - | |
Non-acylated, major circulating isoform of ghrelin | ||||
| GC16673 | N-Formyl-Met-Leu-Phe | 59880-97-6 | >99.50% | |
N-Formyl-Met-Leu-Phe是一种内源性趋化肽，也是甲酰肽受体1（FPR1）的激动剂，Ki值为38 nM。 | ||||
| GC16683 | SR 142948 | 184162-64-9 | >98.00% | |
A neurotensin receptor antagonist | ||||
| GC16688 | APC 366 | 158921-85-8 | - | |
A mast cell tryptase inhibitor | ||||
| GC16689 | 3-chloro-5-hydroxy BA | 53984-36-4 | >98.00% | |
An agonist of GPR81 | ||||
| GC16692 | Casin | 425399-05-9 | >98.00% | |
A Cdc42 GTPase inhibitor | ||||
| GC16693 | 13Z,16Z-Docosadienoic Acid | 17735-98-7 | >98.00% | |
A natural ω-6 PUFA | ||||
| GC16715 | Apelin-36 (human) | 252642-12-9 | - | |
Mature peptide and APJ agonist | ||||
| GC16728 | SB 706375 | 733734-61-7 | - | |
urotensin-II (UT) receptor antagonist | ||||
| GC16745 | Orexin B (mouse) | 202801-92-1 | >98.50% | |
Orexin B (mouse) (Rat orexin B) 是 Orexin 受体的内源性激动剂，对 OX1 和 OX2 的 Kis 分别为 420 和 36 nM。 | ||||
| GC16752 | Olmesartan medoxomil | 144689-63-4 | >99.50% | |
A prodrug form of olmesartan | ||||
| GC16761 | Bombinakinin M | 509151-65-9 | - | |
Potent bradykinin receptor agonist | ||||
| GC16791 | Benztropine mesylate | 132-17-2 | >99.50% | |
An M 1 muscarinic acetylcholine receptor antagonist | ||||
| GC16800 | MF498 | 915191-42-3 | >98.50% | |
A selective EP 4 antagonist | ||||
| GC16807 | AT 1015 | 190508-50-0 | - | |
Long-acting 5-HT2A antagonist | ||||
| GC16819 | VU0152100 | 409351-28-6 | >98.00% | |
A muscarinic M 4 receptor positive allosteric modulator | ||||
| GC16820 | ELN441958 | 913064-47-8 | >98.00% | |
ELN441958是一种强效、竞争性且选择性的bradykinin B1受体拮抗剂，K i 值为0.26nM。 | ||||