GPCR/G protein
GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(504)
- Acetylcholine(29)
- Adenosine Deaminase(9)
- Adenosine Receptor(132)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(421)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(114)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(160)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(81)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(80)
- CysLT1 receptor(1)
- Endothelin Receptor(52)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(18)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(21)
- GIP Receptor(5)
- Glucagon Receptor(61)
- Glucocorticoid Receptor(97)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(58)
- LPA Receptor(12)
- LPL Receptor(60)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(58)
- Melatonin Receptors(24)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(24)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(20)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(48)
- Oxytocin Receptors(22)
- P2Y Receptor(62)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(172)
- Protease-Activated Receptors(10)
- Prostanoid Receptors
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(59)
- Vasopressin Receptor(35)
- 17,20-lyase(5)
- Ras(142)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(185)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(27)
- GRK(1)
- GPR88
- Amylin Receptor
- Arrestin
- GCGR(2)
- GLP Receptor(2)
- Mas-related G-protein-coupled Receptor (MRGPR)
- Succinate Receptor 1
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
GPCR/G protein 相关产品(3377)
- GC13175Sarafotoxin S6aCAS: 126738-34-9
Sarafotoxin S6a 是一种 sarafotoxin 类似物，是一种内皮素受体激动剂，具有与 Endothelin-3 相似的 ETA/ETB 选择性特征。
- GC13190R-Palmitoyl-(1-methyl) EthanolamideCAS: 142128-47-0纯度: >98.00%
A synthetic analog of palmitoyl ethanolamide
- GC13236ACT-132577CAS: 1103522-45-7纯度: >98.00%
A dual ET A and ET B receptor antagonist and an active metabolite of macitentan
- GC13239Hemokinin 1 (mouse)CAS: 208041-90-1纯度: >98.00%
Hemokinin 1 (mouse) 是一种选择性的神经激肽-1 受体激动剂，对人 NK1 受体和人 NK2 受体的 Ki 分别为 0.175 nM 和 560 nM。
- GC13256Dihydroergocristine mesylateCAS: 24730-10-7纯度: >99.50%
An alkaloid with diverse biological activities
- GC13281VU 0364770CAS: 61350-00-3纯度: >99.50%
An mGluR4 and mGluR6 positive allosteric modulator and mGluR5 antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13167 | Pancreatic Polypeptide (human) | 75976-10-2 | >99.50% | |
An NPY receptor agonist | ||||
| GC13175 | Sarafotoxin S6a | 126738-34-9 | - | |
Sarafotoxin S6a 是一种 sarafotoxin 类似物，是一种内皮素受体激动剂，具有与 Endothelin-3 相似的 ETA/ETB 选择性特征。 | ||||
| GC13177 | CI 988 | 130332-27-3 | - | |
CI 988 (PD134308) 是一种有效的、选择性的、具有口服活性的 CCK2R（胆囊收缩素 2 受体）拮抗剂，对小鼠皮质 CCK2 的 IC50 为 1.7 nM。 | ||||
| GC13179 | R 892 | 229030-05-1 | - | |
bradykinin B1 receptor antagonist | ||||
| GC13180 | Carazolol | 57775-29-8 | - | |
A β-AR ligand | ||||
| GC13190 | R-Palmitoyl-(1-methyl) Ethanolamide | 142128-47-0 | >98.00% | |
A synthetic analog of palmitoyl ethanolamide | ||||
| GC13191 | Irsogladine | 57381-26-7 | >99.50% | |
A gastroprotective agent | ||||
| GC13192 | E4CPG | 170846-89-6 | >98.00% | |
An antagonist of mGluR1 and mGluR2 | ||||
| GC13193 | Galanin (porcine) | 88813-36-9 | - | |
Endogenous porcine galanin receptor agonist | ||||
| GC13205 | U 46619 | 56985-40-1 | >98.00% | |
A TP receptor agonist | ||||
| GC13221 | NF 546 | 1006028-37-0 | - | |
NF 546 是一种选择性非核苷酸 P2Y11 激动剂，pEC50 为 6.27。 | ||||
| GC13236 | ACT-132577 | 1103522-45-7 | >98.00% | |
A dual ET A and ET B receptor antagonist and an active metabolite of macitentan | ||||
| GC13239 | Hemokinin 1 (mouse) | 208041-90-1 | >98.00% | |
Hemokinin 1 (mouse) 是一种选择性的神经激肽-1 受体激动剂，对人 NK1 受体和人 NK2 受体的 Ki 分别为 0.175 nM 和 560 nM。 | ||||
| GC13242 | SR 48692 | 146362-70-1 | >98.00% | |
SR 48692（Meclinertant）是一种口服可生物利用的神经降压素受体NTS1的变构拮抗剂（K d =3.4nM）。 | ||||
| GC13254 | M 1145 | 1172089-00-7 | - | |
M 1145 是一种嵌合肽，是一种选择性甘丙肽受体 2 型 (GAL2) 激动剂，Ki 为 6.55 nM。 | ||||
| GC13256 | Dihydroergocristine mesylate | 24730-10-7 | >99.50% | |
An alkaloid with diverse biological activities | ||||
| GC13265 | Donitriptan hydrochloride | 170911-68-9 | - | |
5-HT1B/1D receptors agonist, potent and selective | ||||
| GC13267 | NIDA 41020 | 502486-89-7 | - | |
A CB 1 receptor antagonist | ||||
| GC13274 | 8-Aminoadenine | 28128-33-8 | - | |
Adenine receptor agonist | ||||
| GC13281 | VU 0364770 | 61350-00-3 | >99.50% | |
An mGluR4 and mGluR6 positive allosteric modulator and mGluR5 antagonist | ||||
| GC13284 | CJ-42794 | 847728-01-2 | >98.00% | |
A selective EP 4 receptor antagonist | ||||
| GC13291 | Prucalopride Succinat | 179474-85-2 | >99.50% | |
A selective 5-HT 4 receptor agonist | ||||
| GC13294 | PSN 375963 hydrochloride | 388575-52-8 | >98.00% | |
A selective agonist of GPR119 | ||||
| GC13298 | NAS-181 | 1217474-40-2 | - | |
NAS181 是一种有效的、选择性的大鼠 5-HT1B 受体拮抗剂，Ki 为 47 nM。 | ||||