Metabolism
Metabolism(代谢)
- PPAR(219)
- 5-alpha Reductase(11)
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Metabolism 相关产品(3072)
- GC12764AminophyllineCAS: 317-34-0纯度: >99.50%
A phosphodiesterase inhibitor and adenosine receptor antagonist
- GC12771Etazolate hydrochlorideCAS: 35838-58-5
PDE-4 inhibitor and selective GABA-A receptor modulator
- GC1304417-DMAG (Alvespimycin) HClCAS: 467214-21-7纯度: >98.00%
17-DMAG (Alvespimycin) HCl是一种有效的Hsp90的抑制剂,其IC 50 值为62nM。
- GC13204InolitazoneCAS: 223132-37-4
Inolitazone 是一种新型的高亲和力 PPARγ 激动剂,其生物活性依赖于 PPARγ,抑制生长的 IC50 为 0.8 nM。
- GC13535FluvastatinCAS: 93957-54-1纯度: >98.00%
Fluvastatin是一种亲脂性的3-羟基-3-甲基戊二酰辅酶A(HMG-CoA)还原酶抑制剂,可在多种癌细胞中抑制增殖并诱导凋亡。
- GC13652DyphyllineCAS: 479-18-5纯度: >99.00%
An adenosine receptor antagonist and phosphodiesterase inhibitor
- GC13771CanagliflozinCAS: 842133-18-0纯度: >99.50% / >98.00%
Canagliflozin是一种用于治疗2型糖尿病的钠葡萄糖共转运体(SGLT2)抑制剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC12596 | Nepicastat (SYN-117) HCl | 170151-24-3 | >98.50% | |
An inhibitor of dopamine β-hydroxylase | ||||
| GC12693 | JZL 195 | 1210004-12-8 | >98.00% | |
JZL 195是一种具有高效选择性、不可逆的脂肪酸酰胺水解酶(FAAH)和单酰甘油脂肪酶(MAGL)双重抑制剂,IC 50 值分别为2nM和4nM。 | ||||
| GC12764 | Aminophylline | 317-34-0 | >99.50% | |
A phosphodiesterase inhibitor and adenosine receptor antagonist | ||||
| GC12771 | Etazolate hydrochloride | 35838-58-5 | - | |
PDE-4 inhibitor and selective GABA-A receptor modulator | ||||
| GC12801 | Rasagiline Mesylate | 161735-79-1 | >99.50% | |
An inhibitor of MAO-B | ||||
| GC12808 | Pimobendan | 74150-27-9 | >99.00% | |
An inhibitor of PDE3 | ||||
| GC12820 | T0070907 | 313516-66-4 | >99.50% | |
T0070907是一种有效的选择性过氧化物酶体增殖物激活受体γ(PPARγ)拮抗剂,IC 50 值为1nM。 | ||||
| GC12878 | MMPX | 78033-08-6 | - | |
calmodulin-sensitive cyclic GMP phosphodiesterase inhibitor | ||||
| GC12880 | GSK 2830371 | 1404456-53-6 | >98.50% | |
An inhibitor of Wip1 phosphatase | ||||
| GC12894 | Balaglitazone | 199113-98-9 | >99.50% | |
A partial agonist of PPARγ | ||||
| GC12919 | Pralatrexate | 146464-95-1 | >98.00% | |
A dihydrofolate reductase inhibitor | ||||
| GC13044 | 17-DMAG (Alvespimycin) HCl | 467214-21-7 | >98.00% | |
17-DMAG (Alvespimycin) HCl是一种有效的Hsp90的抑制剂,其IC 50 值为62nM。 | ||||
| GC13076 | Deltarasin | 1440898-61-2 | - | |
A KRAS inhibitor | ||||
| GC13121 | Piclamilast | 144035-83-6 | - | |
A PDE4 inhibitor | ||||
| GC13204 | Inolitazone | 223132-37-4 | - | |
Inolitazone 是一种新型的高亲和力 PPARγ 激动剂,其生物活性依赖于 PPARγ,抑制生长的 IC50 为 0.8 nM。 | ||||
| GC13414 | AT13387 | 912999-49-6 | >99.50% | |
AT13387是一种小分子非安沙霉素类HSP90(热休克蛋白90)抑制剂,其作用机制是通过靶向AKT和ERK信号通路。 | ||||
| GC13495 | Trequinsin hydrochloride | 78416-81-6 | >99.50% | |
An inhibitor of PDE3 | ||||
| GC13535 | Fluvastatin | 93957-54-1 | >98.00% | |
Fluvastatin是一种亲脂性的3-羟基-3-甲基戊二酰辅酶A(HMG-CoA)还原酶抑制剂,可在多种癌细胞中抑制增殖并诱导凋亡。 | ||||
| GC13614 | Mycophenolate Mofetil | 128794-94-5 | >99.50% | |
A prodrug form of mycophenolic acid | ||||
| GC13633 | Ciprofibrate | 52214-84-3 | >99.50% | |
A selective PPARα agonist | ||||
| GC13652 | Dyphylline | 479-18-5 | >99.00% | |
An adenosine receptor antagonist and phosphodiesterase inhibitor | ||||
| GC13657 | Mesopram | 189940-24-7 | - | |
PDE4 inhibitor, orally active | ||||
| GC13683 | Rivaroxaban | 366789-02-8 | >99.50% | |
A selective inhibitor of Factor Xa | ||||
| GC13771 | Canagliflozin | 842133-18-0 | >99.50% / >98.00% | |
Canagliflozin是一种用于治疗2型糖尿病的钠葡萄糖共转运体(SGLT2)抑制剂。 | ||||
