Metabolism
Metabolism(代谢)
- PPAR(219)
- 5-alpha Reductase(11)
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- HSP(100)
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- P450(456)
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Metabolism 相关产品(3072)
- GC33023D,L-Buthionine-(S,R)-sulfoximine (Butionine sulfoximine)CAS: 5072-26-4纯度: >98.00%
A γ-glutamylcysteine synthetase inhibitor
- GC330593α-AminocholestaneCAS: 2206-20-4纯度: >98.00%
3α-Aminocholestane是肌醇-5'-磷酸酶1(SHIP1)的抑制剂,属于胆固醇衍生物,其IC 50 约为10μM。
- GC33067SophoflavescenolCAS: 216450-65-6纯度: >98.00%
Sophoflavescenol是一种异戊烯基黄酮类化合物,能够抑制PDE5的活性,IC50值为0.013μM;同时抑制RLAR,HRAR,BACE1,AChE和BChE,IC50值分别为0.30µM,0.17µM,10.98µM,8.37µM和8.21µM。
- GC330714'-MethylchrysoeriolCAS: 4712-12-3纯度: >99.00%
4'-Methylchrysoeriol是有效的细胞色素P450酶(P450)的抑制剂,其对人P4501B1依赖的乙氧基烯丙醇-O-脱乙基酶(EROD)的IC50值为19nM.
- GC33098L-Buthionine-(S,R)-sulfoximine (L-Butionine sulfoximine)CAS: 83730-53-4纯度: >98.00%
L-Buthionine-(S,R)-sulfoximine (L-Butionine sulfoximine)是一种谷胱甘肽合成抑制剂。
- GC33426Rocaglamide (Rocaglamide A)CAS: 84573-16-0纯度: >98.50%
Rocaglamide (Rocaglamide A) 是从 Aglaia 属(楝科)中分离出来的。
- GC334571-Naphthaleneacetic acid (1-Naphthylacetic acid)CAS: 86-87-3纯度: >99.50%
1-Naphthaleneacetic acid (α-Naphthaleneacetic acid) is a synthetic plant hormone in the auxin family.
- GC33671GNF-PF-3777 (8-Nitrotryptanthrin)CAS: 77603-42-0
A tryptanthrin derivative with diverse biological activities
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC32991 | Cecropin B | 80451-05-4 | - | |
Cecropin B是一种多肽抗菌素,对大肠杆菌及其他多种革兰氏阴性菌具有强效抗菌活性,具有广谱的抗菌活性。 | ||||
| GC33012 | IDO-IN-2 | 1668565-74-9 | >99.50% | |
An IDO1 inhibitor | ||||
| GC33023 | D,L-Buthionine-(S,R)-sulfoximine (Butionine sulfoximine) | 5072-26-4 | >98.00% | |
A γ-glutamylcysteine synthetase inhibitor | ||||
| GC33044 | RMC-4550 | 2172651-73-7 | >99.00% | |
RMC-4550口服活性的SHP2变构抑制剂(IC 50 =0.583nM)。 | ||||
| GC33047 | SNX-5422 Mesylate (PF-04929113 (Mesylate)) | 1173111-67-5 | - | |
A prodrug for an Hsp90 inhibitor | ||||
| GC33058 | IDO-IN-3 | 2070018-30-1 | >99.50% | |
An inhibitor of IDO1 | ||||
| GC33059 | 3α-Aminocholestane | 2206-20-4 | >98.00% | |
3α-Aminocholestane是肌醇-5'-磷酸酶1(SHIP1)的抑制剂,属于胆固醇衍生物,其IC 50 约为10μM。 | ||||
| GC33067 | Sophoflavescenol | 216450-65-6 | >98.00% | |
Sophoflavescenol是一种异戊烯基黄酮类化合物,能够抑制PDE5的活性,IC50值为0.013μM;同时抑制RLAR,HRAR,BACE1,AChE和BChE,IC50值分别为0.30µM,0.17µM,10.98µM,8.37µM和8.21µM。 | ||||
| GC33071 | 4'-Methylchrysoeriol | 4712-12-3 | >99.00% | |
4'-Methylchrysoeriol是有效的细胞色素P450酶(P450)的抑制剂,其对人P4501B1依赖的乙氧基烯丙醇-O-脱乙基酶(EROD)的IC50值为19nM. | ||||
| GC33073 | 1-Ethynylnaphthalene | 15727-65-8 | >99.00% | |
1-Ethynylnaphthalene 是细胞色素 P450 1B1 的选择性抑制剂。 | ||||
| GC33098 | L-Buthionine-(S,R)-sulfoximine (L-Butionine sulfoximine) | 83730-53-4 | >98.00% | |
L-Buthionine-(S,R)-sulfoximine (L-Butionine sulfoximine)是一种谷胱甘肽合成抑制剂。 | ||||
| GC33191 | IDO-IN-9 | 1888378-12-8 | - | |
IDO-IN-9是一个吲哚胺-2,3-双加氧酶(IDO)抑制剂,在激酶实验和Hela细胞实验中的IC50值分别为0.011和0.0018μM,来自专利WO2016041489A1,化合物6。 | ||||
| GC33227 | F1063-0967 | 613225-56-2 | - | |
A DUSP26 inhibitor | ||||
| GC33286 | TAS-116 | 1260533-36-5 | >99.00% | |
An Hsp90 inhibitor | ||||
| GC33287 | LY-3381916 | 2166616-75-5 | >98.00% | |
An IDO1 inhibitor | ||||
| GC33337 | CDC801 | 192819-27-5 | - | |
CDC801是一种强效的磷酸二酯酶4(PDE4)和肿瘤坏死因子-α(TNF-α)抑制剂。IC50分别为1.1μM和2.5μM。 | ||||
| GC33345 | BN82002 | 396073-89-5 | - | |
BN82002是CDC25磷酸酶的合成抑制剂,其对重组CDC25磷酸酶的IC50值为2.4-6.3μM。 | ||||
| GC33426 | Rocaglamide (Rocaglamide A) | 84573-16-0 | >98.50% | |
Rocaglamide (Rocaglamide A) 是从 Aglaia 属(楝科)中分离出来的。 | ||||
| GC33457 | 1-Naphthaleneacetic acid (1-Naphthylacetic acid) | 86-87-3 | >99.50% | |
1-Naphthaleneacetic acid (α-Naphthaleneacetic acid) is a synthetic plant hormone in the auxin family. | ||||
| GC33469 | NADPH tetracyclohexanamine | 100929-71-3 | - | |
A reduced form of NADP + | ||||
| GC33491 | Acetazolamide D3 | 1189904-01-5 | - | |
AcetazolamideD3是Acetazolamide氘代化合物标准品。 | ||||
| GC33663 | Teprenone (Geranylgeranylacetone) | 6809-52-5 | >99.50% | |
An inducer of Hsp expression | ||||
| GC33671 | GNF-PF-3777 (8-Nitrotryptanthrin) | 77603-42-0 | - | |
A tryptanthrin derivative with diverse biological activities | ||||
| GC33734 | Fonadelpar (NPS-005) | 515138-06-4 | - | |
Fonadelpar (NPS-005) 是 PPARδ;激动剂,用于神经麻痹性角膜病的研究。 | ||||
