Metabolism
Metabolism(代谢)
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Metabolism 相关产品(3072)
- GC16687(R)-EdelfosineCAS: 77286-66-9纯度: >98.00% / >99.00%
(R)-Edelfosine是一种属于具有抗肿瘤和抗寄生虫活性的合成脂质药物。(R)-Edelfosine可通过靶向线粒体和脂筏上的FOF1-ATP合酶,诱导肿瘤细胞发生凋亡样细胞死亡。
- GC16738Tunicamycin MixtureCAS: 11089-65-9纯度: >95.00%
Tunicamycin Mixture是一种同源核苷抗生素的混合物, 可抑制N-糖基化并阻断GlcNAc 磷酸转移酶(GPT)。
- GC16754ClarithromycinCAS: 81103-11-9纯度: >98.00%
Clarithromycin是一种大环内酯类抗生素,通过抑制细菌蛋白质合成发挥作用,与细菌核糖体的50S亚基结合,阻止肽链延长,从而抑制细菌生长。
- GC16966VER 155008CAS: 1134156-31-2纯度: >99.50%
VER 155008是一种强效的,源自腺苷的热休克蛋白70(Hsp70)家族抑制剂,对Hsp70、热休克同源蛋白70(Hsc70)和葡萄糖调节蛋白78(Grp78)的IC 50 值分别为0.5μM、2.6μM和2.6μM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16687 | (R)-Edelfosine | 77286-66-9 | >98.00% / >99.00% | |
(R)-Edelfosine是一种属于具有抗肿瘤和抗寄生虫活性的合成脂质药物。(R)-Edelfosine可通过靶向线粒体和脂筏上的FOF1-ATP合酶,诱导肿瘤细胞发生凋亡样细胞死亡。 | ||||
| GC16697 | fluoro-Dapagliflozin | 1181681-43-5 | - | |
A potent inhibitor of hSGLT2 | ||||
| GC16707 | Isavuconazole | 241479-67-4 | >98.00% | |
A broad-spectrum triazole antifungal agent | ||||
| GC16714 | PACOCF3 | 141022-99-3 | >98.00% | |
Antagonizes DP receptor agonist effects | ||||
| GC16733 | Vildagliptin (LAF-237) | 274901-16-5 | >98.00% | |
A DPP-4 inhibitor | ||||
| GC16738 | Tunicamycin Mixture | 11089-65-9 | >95.00% | |
Tunicamycin Mixture是一种同源核苷抗生素的混合物, 可抑制N-糖基化并阻断GlcNAc 磷酸转移酶(GPT)。 | ||||
| GC16751 | Chlorzoxazone | 95-25-0 | >99.50% | |
A centrally acting muscle relaxant | ||||
| GC16754 | Clarithromycin | 81103-11-9 | >98.00% | |
Clarithromycin是一种大环内酯类抗生素,通过抑制细菌蛋白质合成发挥作用,与细菌核糖体的50S亚基结合,阻止肽链延长,从而抑制细菌生长。 | ||||
| GC16756 | KT182 | 1402612-62-7 | >98.00% | |
A potent inhibitor of ABHD6 | ||||
| GC16770 | Arachidonic Acid Leelamide | - | - | |
A novel fatty acid amide | ||||
| GC16775 | Rotenone | 83-79-4 | >99.50% | |
Rotenone是一种线粒体电子传递链复合物 I 抑制剂,可通过增强线粒体活性氧的产生来诱导细胞凋亡。 | ||||
| GC16777 | YM 511 | 148869-05-0 | - | |
YM 511 是一种高度特异性的非甾体芳香酶抑制剂。 | ||||
| GC16816 | Galloflavin | 568-80-9 | - | |
An inhibitor of lactate dehydrogenase | ||||
| GC16824 | Pargyline (hydrochloride) | 306-07-0 | >99.50% / >99.00% | |
An irreversible MAO inhibitor | ||||
| GC16849 | MBCQ | 150450-53-6 | >99.00% | |
An inhibitor of PDE5 | ||||
| GC16856 | Avanafil | 330784-47-9 | >98.00% / >99.00% | |
A potent and selective PDE5 inhibitor | ||||
| GC16860 | NCT-502 | 1542213-00-2 | >99.00% | |
A PHGDH inhibitor | ||||
| GC16868 | Sulfasalazine | 599-79-1 | >99.00% / >98.00% | |
Sulfasalazine是一种磺胺类药物。 | ||||
| GC16892 | XL-888 | 1149705-71-4 | >99.50% | |
An orally bioavailable Hsp90 inhibitor | ||||
| GC16944 | SR 1664 | 1338259-05-4 | - | |
An inhibitor of Cdk5-mediated PPARγ phosphorylation | ||||
| GC16951 | Stiripentol | 49763-96-4 | >99.50% | |
An antiepileptic compound | ||||
| GC16966 | VER 155008 | 1134156-31-2 | >99.50% | |
VER 155008是一种强效的,源自腺苷的热休克蛋白70(Hsp70)家族抑制剂,对Hsp70、热休克同源蛋白70(Hsc70)和葡萄糖调节蛋白78(Grp78)的IC 50 值分别为0.5μM、2.6μM和2.6μM。 | ||||
| GC17003 | Benzenesulfonamide | 98-10-2 | - | |
carbonic anhydrase inhibitor | ||||
| GC17013 | Amidepsine D | 79786-34-8 | - | |
A diacylglycerol acyltransferase inhibitor | ||||
