Metabolism

Metabolism(代谢)

研究方向

Metabolism 相关产品(3072)

GC12962 Isatin
CAS: 91-56-5
纯度: >98.00%
Isatin (Indoline-2,3-dione) 是一种有效的单胺氧化酶 (MAO) 抑制剂，IC50 为 3 μM。
GC12981 OU749
CAS: 519170-13-9
Inhibitor of γ-glutamyl transferase
GC12992 Fluorometholone Acetate
CAS: 3801-06-7
纯度: >98.00%
A synthetic glucocorticoid
GC13063 N-Benzylpalmitamide
CAS: 74058-71-2
纯度: >98.00%
A long-chain fatty acid amide
GC13079 Voriconazole
CAS: 137234-62-9
纯度: >99.50%
Voriconazole是一种强效竞争性抑制剂，可抑制CYP2B6（IC 50 =1.71μM）、CYP2C9（IC 50 =3.62μM）、CYP2C19（IC 50 =5.25μM）和CYP3A（IC 50 =2.90μM）。
GC13083 Siramesine
CAS: 147817-50-3
A selective σ 2 receptor agonist
GC13124 LY2608204
CAS: 1234703-40-2
纯度: >98.00%
An activator of glucokinase
GC13130 Apixaban
CAS: 503612-47-3
纯度: >99.50%
An inhibitor of Factor Xa
GC13139 FG-4592 (ASP1517)
CAS: 808118-40-3
纯度: >99.50%
FG-4592 作为一种口服生物可利用的缺氧诱导因子 (HIF) 脯氨酰羟化酶抑制剂，可通过 HIF 介导的转录促进协调性红细胞生成。
GC13147 AG-221 (Enasidenib)
CAS: 1446502-11-9
纯度: >99.50%
An inhibitor of mutant IDH2
GC13262 A-771726
CAS: 163451-81-8
纯度: >98.00%
An active metabolite of leflunomide
GC13275 Ibudilast
CAS: 50847-11-5
纯度: >99.50%
An inhibitor of PDE4
GC13276 Oleyloxyethyl Phosphorylcholine
CAS: 84601-19-4
A PLA 2 inhibitor
GC13293 LP533401 hcl
CAS: 1040526-12-2
纯度: >98.50%
An inhibitor of gut-derived serotonin biosynthesis
GC13307 PU-WS13
CAS: 1454619-14-7
纯度: >98.00%
PU-WS13是一种嘌呤支架类Grp94特异性热休克蛋白90（Hsp90）抑制剂。
GC13319 5,8,11-Eicosatriynoic Acid
CAS: 13488-22-7
A nonselective inhibitor of lipoxygenases
GC13336 CBR-5884
CAS: 681159-27-3
纯度: >99.00%
A selective PHGDH inhibitor
GC13351 VU0359595
CAS: 1246303-14-9
纯度: >95.00%
A selective PLD 1 inhibitor
GC13362 TOK-001
CAS: 851983-85-2
纯度: >99.50%
A CYP17 inhibitor
GC13379 1-Naphthyl 3,5-dinitrobenzoate
CAS: 93261-39-3
A dual inhibitor of 5-LO and mPGES-1
GC13444 Doxofylline
CAS: 69975-86-6
纯度: >99.00%
A bronchodilator
GC13464 GSK 2837808A
CAS: 1445879-21-9
纯度: >99.00%
GSK2837808A 是一种选择性的 LDHA (lactate dehydrogenase A) 的抑制剂,对hLDHA和hLDHB的IC50分别为2.6 nM和43 nM.GSK2837808A(10 µM;24-72h)通过促进有氧糖酵解、增殖、细胞周期和细胞凋亡抵抗,阻断了着丝粒蛋白N (CENP-N)过表达对鼻咽癌细胞的影响。
GC13470 Rhapontigenin
CAS: 500-65-2
纯度: >98.00% / >99.50%
Rhapontigenin（丹叶大黄素）是一种有效的细胞色素P4501A1选择性灭活剂，IC 50 为0.4μM，对P4501A1的选择性分别是P4501A2和P4501B1的400倍和23倍。
GC13516 AS 1949490
CAS: 1203680-76-5
纯度: >98.00%
A selective SHIP2 inhibitor

分类产品列表
货号	产品名称	CAS号	纯度
GC12962	Isatin	91-56-5	>98.00%
GC12962	Isatin (Indoline-2,3-dione) 是一种有效的单胺氧化酶 (MAO) 抑制剂，IC50 为 3 μM。
GC12981	OU749	519170-13-9	-
GC12981	Inhibitor of γ-glutamyl transferase
GC12992	Fluorometholone Acetate	3801-06-7	>98.00%
GC12992	A synthetic glucocorticoid
GC13063	N-Benzylpalmitamide	74058-71-2	>98.00%
GC13063	A long-chain fatty acid amide
GC13079	Voriconazole	137234-62-9	>99.50%
GC13079	Voriconazole是一种强效竞争性抑制剂，可抑制CYP2B6（IC 50 =1.71μM）、CYP2C9（IC 50 =3.62μM）、CYP2C19（IC 50 =5.25μM）和CYP3A（IC 50 =2.90μM）。
GC13083	Siramesine	147817-50-3	-
GC13083	A selective σ 2 receptor agonist
GC13124	LY2608204	1234703-40-2	>98.00%
GC13124	An activator of glucokinase
GC13130	Apixaban	503612-47-3	>99.50%
GC13130	An inhibitor of Factor Xa
GC13139	FG-4592 (ASP1517)	808118-40-3	>99.50%
GC13139	FG-4592 作为一种口服生物可利用的缺氧诱导因子 (HIF) 脯氨酰羟化酶抑制剂，可通过 HIF 介导的转录促进协调性红细胞生成。
GC13147	AG-221 (Enasidenib)	1446502-11-9	>99.50%
GC13147	An inhibitor of mutant IDH2
GC13262	A-771726	163451-81-8	>98.00%
GC13262	An active metabolite of leflunomide
GC13275	Ibudilast	50847-11-5	>99.50%
GC13275	An inhibitor of PDE4
GC13276	Oleyloxyethyl Phosphorylcholine	84601-19-4	-
GC13276	A PLA 2 inhibitor
GC13293	LP533401 hcl	1040526-12-2	>98.50%
GC13293	An inhibitor of gut-derived serotonin biosynthesis
GC13307	PU-WS13	1454619-14-7	>98.00%
GC13307	PU-WS13是一种嘌呤支架类Grp94特异性热休克蛋白90（Hsp90）抑制剂。
GC13319	5,8,11-Eicosatriynoic Acid	13488-22-7	-
GC13319	A nonselective inhibitor of lipoxygenases
GC13336	CBR-5884	681159-27-3	>99.00%
GC13336	A selective PHGDH inhibitor
GC13351	VU0359595	1246303-14-9	>95.00%
GC13351	A selective PLD 1 inhibitor
GC13362	TOK-001	851983-85-2	>99.50%
GC13362	A CYP17 inhibitor
GC13379	1-Naphthyl 3,5-dinitrobenzoate	93261-39-3	-
GC13379	A dual inhibitor of 5-LO and mPGES-1
GC13444	Doxofylline	69975-86-6	>99.00%
GC13444	A bronchodilator
GC13464	GSK 2837808A	1445879-21-9	>99.00%
GC13464	GSK2837808A 是一种选择性的 LDHA (lactate dehydrogenase A) 的抑制剂,对hLDHA和hLDHB的IC50分别为2.6 nM和43 nM.GSK2837808A(10 µM;24-72h)通过促进有氧糖酵解、增殖、细胞周期和细胞凋亡抵抗,阻断了着丝粒蛋白N (CENP-N)过表达对鼻咽癌细胞的影响。
GC13470	Rhapontigenin	500-65-2	>98.00% / >99.50%
GC13470	Rhapontigenin（丹叶大黄素）是一种有效的细胞色素P4501A1选择性灭活剂，IC 50 为0.4μM，对P4501A1的选择性分别是P4501A2和P4501B1的400倍和23倍。
GC13516	AS 1949490	1203680-76-5	>98.00%
GC13516	A selective SHIP2 inhibitor