Tyrosine Kinase
Tyrosine Kinase(酪氨酸激酶)
- Bcr-Abl(73)
- Ack1(3)
- Axl(6)
- ALK(64)
- BMX Kinase(3)
- Broad Spectrum Protein Kinase Inhibitor(10)
- c-FMS(42)
- c-Kit(58)
- c-MET(99)
- c-RET(7)
- CSF-1R(3)
- DDR1/DDR2 Receptor(1)
- EGFR(278)
- EphB4(1)
- FAK(39)
- FGFR(104)
- FLT3(97)
- HER2(15)
- IGF1R(34)
- Insulin Receptor(46)
- IRAK(32)
- ITK(10)
- Lck(1)
- LRRK2(25)
- PDGFR(113)
- PTKs/RTKs(10)
- Pyk2(8)
- ROR(41)
- Spleen Tyrosine Kinase (Syk)(33)
- Src(108)
- Tie-2 (4)
- Trk(43)
- VEGFR(200)
- Kinase
- Discoidin Domain Receptor(16)
- DYRK(35)
- Ephrin Receptor(13)
- RET(30)
- ROS(14)
- TAM Receptor(33)
- IGFBR(1)
- Others(55)
Tyrosine Kinase 相关产品(1402)
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10638 | AT9283 | 896466-04-9 | >99.50% | |
A broad spectrum kinase inhibitor | ||||
| GC10644 | Neoruscogenin | 17676-33-4 | - | |
A bioavailable agonist of RORα | ||||
| GC10706 | Rp-8-pCPT-Cyclic GMPS (sodium salt) | 208445-07-2 | - | |
A competitive inhibitor of cGK isoforms | ||||
| GC10720 | NTR 368 | 197230-90-3 | - | |
NTR 368 是衍生自 p75 神经营养因子受体 (p75NTR) 的肽,对应于人类受体的 368-381 位残基。 | ||||
| GC10759 | CH5183284 (Debio-1347) | 1265229-25-1 | >99.00% | |
An inhibitor of FGFR1, 2, and 3 | ||||
| GC10775 | MLR 1023 | 41964-07-2 | >99.50% | |
An allosteric Lyn kinase activator | ||||
| GC10815 | BIBU 1361 dihydrochloride | 793726-84-8 | - | |
EGFR inhibitor | ||||
| GC10833 | BLU9931 | 1538604-68-0 | >99.50% | |
A selective FGFR4 inhibitor | ||||
| GC10915 | GZD824 | 1421783-64-3 | >99.00% | |
A Bcr/Abl inhibitor | ||||
| GC10938 | AAL-993 | 269390-77-4 | - | |
Inhibitor of VEGFR1, 2, and 3 | ||||
| GC10970 | WP1130 | 856243-80-6 | >99.50% | |
A deubiquitinase inhibitor | ||||
| GC11003 | PP121 | 1092788-83-4 | >99.00% | |
A potent dual inhibitor of tyrosine and phosphoinositide kinases | ||||
| GC11024 | AG-213 | 122520-86-9 | >98.00% | |
An inhibitor of EGF receptor kinase | ||||
| GC11057 | LY2801653 | 1206799-15-6 | >98.00% | |
A MET kinase inhibitor | ||||
| GC11140 | Radotinib(IY-5511) | 926037-48-1 | - | |
A selective Bcr-Abl tyrosine kinase inhibitor | ||||
| GC11205 | 5'-Fluoroindirubinoxime | 861214-33-7 | >98.00% | |
An inhibitor of FLT3 kinase | ||||
| GC11209 | Cerdulatinib (PRT062070) | 1198300-79-6 | >99.50% | |
A dual inhibitor of Syk and JAKs | ||||
| GC11250 | WZ8040 | 1214265-57-2 | >98.00% | |
An inhibitor of mutant EGFR | ||||
| GC11264 | CNX-2006 | 1375465-09-0 | >99.50% | |
An irreversible inhibitor of mutant EGFRs | ||||
| GC11312 | EGFR Inhibitor | 879127-07-8 | >99.00% | |
A selective antagonist of the EGFR | ||||
| GC11321 | PRT-060318 | 1194961-19-7 | >99.50% | |
A potent and selective Syk inhibitor | ||||
| GC11336 | Motesanib Diphosphate (AMG-706) | 857876-30-3 | >99.50% | |
A multikinase inhibitor | ||||
| GC11362 | K 252a | 99533-80-9 | >98.00% | |
A non-selective PKC inhibitor | ||||
| GC11417 | SU 4312 | 5812-07-7 | >98.00% | |
A selective dual inhibitor of VEGFR2 and PDGFR | ||||
