Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC35727Coniferyl ferulateCAS: 63644-62-2纯度: >98.50%
A monolignal conjugate with diverse biological activities
- GC35860Dibucaine hydrochlorideCAS: 61-12-1纯度: >99.50%
Dibucaine 盐酸盐 (Cinchocaine hydrochloride) 有局部麻醉活性。
- GC35917Dynorphin A (1-10) TFA纯度: >99.00%
Dynorphin A (1-10) (TFA) 是一种内源性的阿片样神经肽,与 κ 阿片受体 (κ-opioid receptor) 结合。Dynorphin A (1-10) (TFA) 也阻断 NMDA 激活的电流,IC50 为 42.0 μM。
- GC35918Dynorphin A 1-10CAS: 79994-24-4
Dynorphin A (1-10) 是一种内源性的阿片样神经肽,与 κ 阿片受体 (κ-opioid receptor) 结合。Dynorphin A (1-10) 也阻断 NMDA 激活的电流,IC50 为 42.0 μM。
- GC35963Efonidipine hydrochloride monoethanolateCAS: 111011-76-8纯度: >99.00%
An L- and T-type calcium channel inhibitor
- GC35970EIPA hydrochlorideCAS: 1345839-28-2纯度: >99.00%
EIPA hydrochloride (L593754 hydrochloride) 是一种 TRPP3 channel 抑制剂,其 IC50 值为 10.5 μM。EIPA 还抑制 Na+/H+ 交换器 (NHE) 和巨噬细胞。
- GC35975Emamectin BenzoateCAS: 155569-91-8纯度: >98.50%
Emamectin Benzoate (EMB, MK-244) activates gamma-amino butyric acid (GABA) transporter. Emamectin Benzoate induces of reactive oxygen species (ROS)-mediated DNA damage and apoptosis.
- GC35991Endoxifen Z-isomer hydrochlorideCAS: 1032008-74-4纯度: >99.00%
Endoxifen HCl, the active metabolite of Tamoxifen, ia a potent and selective estrogen receptor antagonist. Phase 2.
- GC36027Fanapanel hydrateCAS: 1255517-78-2纯度: >99.50%
Fanapanel hydrate (ZK200775 hydrate) 是高选择性AMPA拮抗剂。
- GC36058Flumazenil acidCAS: 84378-44-9
Flumazenil acid 是 Flumazenil 的一种代谢产物。Flumazenil 是一种 GABAA 受体拮抗剂。
- GC36091Furosemide sodiumCAS: 41733-55-5纯度: >99.50%
A loop diuretic and an inhibitor of NKCC1 and NKCC2
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC35669 | CGP 36742 | 123690-78-8 | >98.00% | |
A GABA B receptor antagonist | ||||
| GC35692 | Chrysosplenetin | 603-56-5 | >99.50% | |
A flavonoid with diverse biological activities | ||||
| GC35713 | CLP290 | 1181083-81-7 | >99.50% | |
A prodrug form of CLP 257 | ||||
| GC35727 | Coniferyl ferulate | 63644-62-2 | >98.50% | |
A monolignal conjugate with diverse biological activities | ||||
| GC35738 | CP-060 | 180090-15-7 | - | |
CP-?060 是一种 Ca2+ 拮抗剂,能够抑制 Ca2+ 过载,具有抗氧化、保护心脏的作用。 | ||||
| GC35858 | Dianicline | 292634-27-6 | - | |
Dianicline是一种α4β2烟碱型乙酰胆碱受体部分激动剂,一类包括伐尼克兰和金雀花碱的戒烟药物。 | ||||
| GC35860 | Dibucaine hydrochloride | 61-12-1 | >99.50% | |
Dibucaine 盐酸盐 (Cinchocaine hydrochloride) 有局部麻醉活性。 | ||||
| GC35892 | Dofequidar | 129716-58-1 | - | |
A quinoline derivative and inhibitor of multidrug resistance | ||||
| GC35903 | DSP-2230 | 1233231-30-5 | >98.00% | |
DSP-2230 是选择性的 Nav1.7/Nav1.8 通道阻断剂。 | ||||
| GC35917 | Dynorphin A (1-10) TFA | - | >99.00% | |
Dynorphin A (1-10) (TFA) 是一种内源性的阿片样神经肽,与 κ 阿片受体 (κ-opioid receptor) 结合。Dynorphin A (1-10) (TFA) 也阻断 NMDA 激活的电流,IC50 为 42.0 μM。 | ||||
| GC35918 | Dynorphin A 1-10 | 79994-24-4 | - | |
Dynorphin A (1-10) 是一种内源性的阿片样神经肽,与 κ 阿片受体 (κ-opioid receptor) 结合。Dynorphin A (1-10) 也阻断 NMDA 激活的电流,IC50 为 42.0 μM。 | ||||
| GC35963 | Efonidipine hydrochloride monoethanolate | 111011-76-8 | >99.00% | |
An L- and T-type calcium channel inhibitor | ||||
| GC35970 | EIPA hydrochloride | 1345839-28-2 | >99.00% | |
EIPA hydrochloride (L593754 hydrochloride) 是一种 TRPP3 channel 抑制剂,其 IC50 值为 10.5 μM。EIPA 还抑制 Na+/H+ 交换器 (NHE) 和巨噬细胞。 | ||||
| GC35975 | Emamectin Benzoate | 155569-91-8 | >98.50% | |
Emamectin Benzoate (EMB, MK-244) activates gamma-amino butyric acid (GABA) transporter. Emamectin Benzoate induces of reactive oxygen species (ROS)-mediated DNA damage and apoptosis. | ||||
| GC35982 | EN6 | 1808714-73-9 | >99.00% | |
An activator of autophagy | ||||
| GC35991 | Endoxifen Z-isomer hydrochloride | 1032008-74-4 | >99.00% | |
Endoxifen HCl, the active metabolite of Tamoxifen, ia a potent and selective estrogen receptor antagonist. Phase 2. | ||||
| GC35993 | Eniporide hydrochloride | 211813-86-4 | >99.00% | |
A NHE-1 inhibitor | ||||
| GC36009 | Esomeprazole magnesium salt | 1198768-91-0 | - | |
An H + /K + -ATPase inhibitor | ||||
| GC36012 | Etifoxine | 21715-46-8 | >98.00% | |
A positive allosteric modulator of GABA A receptors | ||||
| GC36027 | Fanapanel hydrate | 1255517-78-2 | >99.50% | |
Fanapanel hydrate (ZK200775 hydrate) 是高选择性AMPA拮抗剂。 | ||||
| GC36034 | FD 12-9 | 1451741-22-2 | - | |
FD 12-9 是一种类黄酮二聚体,为 P-gp 和 BCRP 的双重抑制剂,EC50 值分别为 285 nM 和 0.9 nM。具有抗胶质细胞瘤活性。 | ||||
| GC36058 | Flumazenil acid | 84378-44-9 | - | |
Flumazenil acid 是 Flumazenil 的一种代谢产物。Flumazenil 是一种 GABAA 受体拮抗剂。 | ||||
| GC36060 | Flupirtine | 56995-20-1 | - | |
An activator of Kv7 channels | ||||
| GC36091 | Furosemide sodium | 41733-55-5 | >99.50% | |
A loop diuretic and an inhibitor of NKCC1 and NKCC2 | ||||
