Sodium Channel
Sodium Channel(钠离子通道)
Sodium channel are integral membrane proteins that form ion channels, conducting sodium ions (Na+) through a cell plasma membrane.
Sodium Channel 相关产品(203)
- GC10500OxcarbazepineCAS: 28721-07-5纯度: >98.50%
A prodrug form of 10,11-dihydro-10-hydroxy carbamazepine
- GC10234GSK1014802(CNV1014802)CAS: 934240-30-9纯度: >99.00%
GSK1014802(CNV1014802) (GSK-1014802)是一种新型的小分子状态依赖性钠通道阻滞剂; Nav1.7 钠通道抑制剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10500 | Oxcarbazepine | 28721-07-5 | >98.50% | |
A prodrug form of 10,11-dihydro-10-hydroxy carbamazepine | ||||
| GC10615 | S0859 | 1019331-10-2 | >99.50% | |
A selective sodium/bicarbonate cotransporter blocker | ||||
| GC10639 | Propafenone HCl | 34183-22-7 | >99.50% | |
A class I antiarrhythmic agent | ||||
| GC12051 | Amiloride HCl dihydrate | 17440-83-4 | >98.00% | |
An Analytical Reference Standard | ||||
| GC12254 | Triamterene | 396-01-0 | >99.50% | |
An ENaC inhibitor | ||||
| GC12410 | Bupivacaine HCl | 18010-40-7 | >98.00% / >99.50% | |
An Analytical Reference Standard | ||||
| GC12858 | Phenytoin sodium | 630-93-3 | >99.50% | |
An anticonvulsant agent | ||||
| GC13397 | Proparacaine HCl | 5875-06-9 | - | |
voltage-gated sodium channels antagonist | ||||
| GC13802 | Riluzole | 1744-22-5 | >98.00% | |
Riluzole 是一种抗惊厥药,属于使用依赖性 Na+ 通道阻滞剂家族,它也可以抑制 GABA 摄取,IC50 为 43 μM。 | ||||
| GC14764 | Lamotrigine | 84057-84-1 | >99.50% | |
An anticonvulsant | ||||
| GC15458 | Ambroxol HCl | 23828-92-4 | >98.00% | |
An expectorant | ||||
| GC15701 | A-803467 | 944261-79-4 | >98.50% | |
A-803467是一种河豚毒素耐受型Na v 1.8钠通道的阻断剂,其阻断人Na v 1.8钠通道的IC 50 为8nM。 | ||||
| GC15823 | Flecainide acetate | 54143-56-5 | >99.50% | |
An inhibitor of cardiac late sodium current | ||||
| GC15860 | Ibutilide Fumarate | 122647-32-9 | >98.00% | |
A class III antiarrhythmic drug | ||||
| GC16086 | Phenytoin | 57-41-0 | >99.50% | |
An anticonvulsant agent | ||||
| GC16173 | Procaine HCl | 51-05-8 | - | |
An Analytical Reference Standard | ||||
| GC16696 | Dibucaine (Cinchocaine) HCl | 61-12-1 | - | |
An Analytical Reference Standard | ||||
| GC17340 | Carbamazepine | 298-46-4 | >99.50% | |
卡马西平是一种钠通道阻滞剂,是一种抗惊厥药。 | ||||
| GC10224 | Mepivacaine HCl | 1722-62-9 | >99.50% | |
An Analytical Reference Standard | ||||
| GC10234 | GSK1014802(CNV1014802) | 934240-30-9 | >99.00% | |
GSK1014802(CNV1014802) (GSK-1014802)是一种新型的小分子状态依赖性钠通道阻滞剂; Nav1.7 钠通道抑制剂。 | ||||
| GC10830 | GS967 | 1262618-39-2 | >99.50% | |
GS967是一种强效、选择性的晚期钠电流抑制剂,在心室肌细胞和离体心脏中的IC 50 值分别为0.13μM和0.21μM。 | ||||
| GC10836 | Jingzhaotoxin III | 925463-91-8 | - | |
NaV1.5 channels blocker | ||||
| GC11041 | Sipatrigine | 130800-90-7 | >99.00% | |
A neuroprotective agent | ||||
| GC11069 | Meticrane | 1084-65-7 | >98.00% | |
Meticrane 是一种利尿剂。 | ||||
