Sodium Channel
Sodium Channel(钠离子通道)
Sodium channel are integral membrane proteins that form ion channels, conducting sodium ions (Na+) through a cell plasma membrane.
Sodium Channel 相关产品(203)
- GC15824Ethyl 3-Aminobenzoate (methanesulfonate)CAS: 886-86-2纯度: >99.50% / >98.00% / >99.00%
A fish anesthetic
- GC25134Benzocaine hydrochlorideCAS: 23239-88-5纯度: >99.00%
Benzocaine hydrochloride (Ethyl 4-aminobenzoate, Ethyl p-aminobenzoate) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.
- GC25812Quinidine sulfateCAS: 6591-63-5
Quinidine (Chinidin, Pitayine, β-quinine, (+)-quinidine) acts as a blocker of voltage-gated sodium channels, also an antimuscarinic and antimalarial.
- GC25936SLC13A5-IN-1CAS: 2227548-95-8
SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5/NaCT). It completely blocks the uptake of 14 C-citrate and has the potential for the treatment of metabolic and/or cardiovascular diseases.
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15824 | Ethyl 3-Aminobenzoate (methanesulfonate) | 886-86-2 | >99.50% / >98.00% / >99.00% | |
A fish anesthetic | ||||
| GC15893 | EIPA | 1154-25-2 | >98.00% / >99.00% | |
EIPA 抑制 TRPP3 介导的 Ca2+- 激活电流,IC50 值为 10.5 μM 。 | ||||
| GC15915 | Dibucaine | 85-79-0 | >99.50% | |
An Analytical Reference Standard | ||||
| GC15978 | Levobupivacaine HCl | 27262-48-2 | >99.00% | |
A sodium channel blocker and local anesthetic | ||||
| GC16149 | Topiramate | 97240-79-4 | >98.00% | |
Topiramate是一种口服有效的磺胺衍生单糖,具有广谱抗癫痫活性。 | ||||
| GC16182 | Co 102862 | 181144-66-1 | - | |
Co 102862 (V 102862) 是一种强效、广谱、依赖于状态的 Na+ 通道阻滞剂。 | ||||
| GC16390 | Ropivacaine hydrochloride monohydrate | 132112-35-7 | >99.50% | |
A sodium channel blocker | ||||
| GC16658 | Vinpocetine | 42971-09-5 | >99.50% | |
An inhibitor of PDE1 | ||||
| GC16786 | KC 12291 hydrochloride | 181936-98-1 | - | |
voltage-gated sodium channel blocker | ||||
| GC17395 | ICA 121431 | 313254-51-2 | >98.00% | |
A selective Na v 1.1 and Na v 1.3 channel blocker | ||||
| GC17495 | QX 314 chloride | 5369-03-9 | >99.50% | |
A selective sodium channel blocker | ||||
| GC17608 | Lidocaine | 137-58-6 | >99.50% | |
An Analytical Reference Standard | ||||
| GC17842 | CARIPORIDE | 159138-80-4 | >98.50% | |
An NHE-1 inhibitor | ||||
| GC17853 | Amiloride HCl | 2016-88-8 | >98.00% | |
An Analytical Reference Standard | ||||
| GC17952 | Zonisamide sodium | 68291-98-5 | - | |
A broad-spectrum sulfonamide antiepileptic agent | ||||
| GC18203 | Annonacin | 111035-65-5 | >98.00% | |
A mitochondrial complex I inhibitor | ||||
| GC18947 | PF-05089771 (tosylate) | 1430806-04-4 | - | |
An Na v 1.7 channel blocker | ||||
| GC19281 | PF-01247324 | 875051-72-2 | >99.50% | |
An inhibitor of Na v 1.8 channels | ||||
| GC19289 | PF-06869206 | 2227425-05-8 | >99.50% | |
An NaPi2a inhibitor | ||||
| GC19352 | Tenapanor | 1234423-95-0 | - | |
A NHE-3 inhibitor | ||||
| GC25134 | Benzocaine hydrochloride | 23239-88-5 | >99.00% | |
Benzocaine hydrochloride (Ethyl 4-aminobenzoate, Ethyl p-aminobenzoate) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings. | ||||
| GC25812 | Quinidine sulfate | 6591-63-5 | - | |
Quinidine (Chinidin, Pitayine, β-quinine, (+)-quinidine) acts as a blocker of voltage-gated sodium channels, also an antimuscarinic and antimalarial. | ||||
| GC25936 | SLC13A5-IN-1 | 2227548-95-8 | - | |
SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5/NaCT). It completely blocks the uptake of 14 C-citrate and has the potential for the treatment of metabolic and/or cardiovascular diseases. | ||||
| GC26033 | Veratrine | 62-59-9 | - | |
Veratridine (Cevadine, Cevadin, Cevadene), a steroidal alkaloid found in plants of the lily family, is a voltage-gated sodium channel activator. Veratridine induces anxiogenic-like behaviors in rats. | ||||
