Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC10038Vernakalant HydrochlorideCAS: 748810-28-8纯度: >99.00%
Vernakalant hydrochloride 是一种混合的电压和频率依赖性 Na+ 和心房首选的 K+ 通道阻滞剂。
- GC10500OxcarbazepineCAS: 28721-07-5纯度: >98.50%
A prodrug form of 10,11-dihydro-10-hydroxy carbamazepine
- GC10680AR-C155858CAS: 496791-37-8纯度: >98.00%
AR-C155858是一种强效的单羧酸转运蛋白1(MCT1)抑制剂,K i 值为2.3nM,也能抑制MCT2,K i 值>10nM。
- GC10772FlumazenilCAS: 78755-81-4纯度: >99.50% / >98.00%
A GABA A receptor antagonist and partial agonist
- GC11058Scrambled 10PanxCAS: 1315378-72-3
Panx-1 mimetic inhibitory peptide, blocks pannexin-1 gap junctions
- GC11070Dehydroepiandrosterone (DHEA)CAS: 53-43-0纯度: >99.00%
脱氢表雄酮 (DHEA) 及其硫酸酯 DHEAS 共同代表了人体内最丰富的类固醇激素。
- GC11411ML-7 hydrochlorideCAS: 110448-33-4纯度: >99.50% / >98.00%
ML-7 hydrochloride是一种选择性肌球蛋白轻链激酶(IC 50 = 300nM)。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10038 | Vernakalant Hydrochloride | 748810-28-8 | >99.00% | |
Vernakalant hydrochloride 是一种混合的电压和频率依赖性 Na+ 和心房首选的 K+ 通道阻滞剂。 | ||||
| GC10091 | Nateglinide | 105816-04-4 | >99.50% | |
A hypoglycemic agent | ||||
| GC10206 | Bitopertin | 845614-11-1 | >99.50% | |
An inhibitor of GlyT1 | ||||
| GC10270 | Noopept | 157115-85-0 | >99.50% | |
An Analytical Reference Standard | ||||
| GC10415 | Tezampanel | 154652-83-2 | - | |
AMPA receptor antagonist | ||||
| GC10424 | Tolbutamide | 64-77-7 | >99.50% | |
A SUR1/K ir 6.2 channel inhibitor | ||||
| GC10447 | Isradipine (Dynacirc) | 75695-93-1 | >99.00% | |
An L-type calcium channel blocker | ||||
| GC10500 | Oxcarbazepine | 28721-07-5 | >98.50% | |
A prodrug form of 10,11-dihydro-10-hydroxy carbamazepine | ||||
| GC10522 | Felbamate | 25451-15-4 | >98.00% | |
An inhibitor of NMDA receptors and a modulator of GABA A receptors | ||||
| GC10599 | Esomeprazole Sodium | 161796-78-7 | >99.50% | |
Esomeprazole Sodium是一种强效、具有口服活性的质子泵抑制剂。 | ||||
| GC10615 | S0859 | 1019331-10-2 | >99.50% | |
A selective sodium/bicarbonate cotransporter blocker | ||||
| GC10639 | Propafenone HCl | 34183-22-7 | >99.50% | |
A class I antiarrhythmic agent | ||||
| GC10680 | AR-C155858 | 496791-37-8 | >98.00% | |
AR-C155858是一种强效的单羧酸转运蛋白1(MCT1)抑制剂,K i 值为2.3nM,也能抑制MCT2,K i 值>10nM。 | ||||
| GC10772 | Flumazenil | 78755-81-4 | >99.50% / >98.00% | |
A GABA A receptor antagonist and partial agonist | ||||
| GC10928 | Tariquidar methanesulfonate, hydrate | 625375-83-9 | >98.00% | |
A P-glycoprotein inhibitor | ||||
| GC10974 | AWD 131-138 | 188116-07-6 | >99.00% | |
A partial agonist of the GABA A receptor | ||||
| GC11058 | Scrambled 10Panx | 1315378-72-3 | - | |
Panx-1 mimetic inhibitory peptide, blocks pannexin-1 gap junctions | ||||
| GC11070 | Dehydroepiandrosterone (DHEA) | 53-43-0 | >99.00% | |
脱氢表雄酮 (DHEA) 及其硫酸酯 DHEAS 共同代表了人体内最丰富的类固醇激素。 | ||||
| GC11195 | Sarcosine | 107-97-1 | >98.00% | |
An intermediate in the biosynthesis of glycine | ||||
| GC11229 | IOWH-032 | 1191252-49-9 | >99.50% | |
A modulator of CFTR | ||||
| GC11299 | Mitiglinide Calcium | 145525-41-3 | >98.50% | |
A SUR1/K ir 6.2 inhibitor | ||||
| GC11341 | LY 2365109 hydrochloride | 868265-28-5 | >99.00% | |
glycine transporter 1 (GlyT1) inhibitor | ||||
| GC11411 | ML-7 hydrochloride | 110448-33-4 | >99.50% / >98.00% | |
ML-7 hydrochloride是一种选择性肌球蛋白轻链激酶(IC 50 = 300nM)。 | ||||
| GC11432 | Amiodarone HCl | 19774-82-4 | >99.50% / >98.00% | |
An antiarrhythmic agent | ||||
