Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC12268MibefradilCAS: 116644-53-2纯度: >98.00%
Mibefradil是一种钙通道阻断剂,可以阻断T型和L型钙通道,Mibefradil对T型和L型钙电流的IC 50 分别为0.7μM和2μM。
- GC12970FurosemideCAS: 54-31-9纯度: >99.50% / >98.00%
A loop diuretic and an inhibitor of NKCC1 and NKCC2
- GC13016SafinamideCAS: 133865-89-1纯度: >99.50%
Safinamide 是一种强效、选择性和可逆的单胺氧化酶 B (MAO-B) 抑制剂 (IC50=0.098 μM),优于 MAO-A (IC50=580 μM)。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11470 | Flupirtine maleate | 75507-68-5 | >99.50% | |
An activator of Kv7 channels | ||||
| GC11735 | Zonisamide | 68291-97-4 | >99.50% | |
A broad-spectrum sulfonamide antiepileptic agent | ||||
| GC11819 | Strontium Ranelate | 135459-87-9 | >99.50% | |
An antiosteoporotic agent | ||||
| GC11865 | UK-5099 | 56396-35-1 | >99.50% | |
UK-5099是一种线粒体丙酮酸载体(MPC)抑制剂,抑制丙酮酸依赖性O 2 消耗的IC 50 值为50nM。 | ||||
| GC11901 | Nefiracetam | 77191-36-7 | >99.00% | |
An Analytical Reference Standard | ||||
| GC12032 | NFPS | 405225-21-0 | - | |
NFPS 是一种选择性、非竞争性甘氨酸转运蛋白-1 (GlyT1) 抑制剂,对 hGlyT1 和 rGlyT1 的 IC50 分别为 2.8 nM 和 9.8 nM。 | ||||
| GC12051 | Amiloride HCl dihydrate | 17440-83-4 | >98.00% | |
An Analytical Reference Standard | ||||
| GC12112 | Lansoprazole sodium | 226904-00-3 | - | |
Proton pump inhibitor | ||||
| GC12234 | Dronedarone HCl | 141625-93-6 | >99.50% | |
An antiarrhythmic agent | ||||
| GC12254 | Triamterene | 396-01-0 | >99.50% | |
An ENaC inhibitor | ||||
| GC12268 | Mibefradil | 116644-53-2 | >98.00% | |
Mibefradil是一种钙通道阻断剂,可以阻断T型和L型钙通道,Mibefradil对T型和L型钙电流的IC 50 分别为0.7μM和2μM。 | ||||
| GC12312 | Cilnidipine | 132203-70-4 | >99.50% | |
An L- and N-type calcium channel blocker | ||||
| GC12339 | Ivermectin | 70288-86-7 | >98.00% | |
Ivermectin是一种大环内酯类内外抗寄生虫药,对体内和体外寄生虫均有活性。 | ||||
| GC12410 | Bupivacaine HCl | 18010-40-7 | >98.00% / >99.50% | |
An Analytical Reference Standard | ||||
| GC12436 | Org 25543 hydrochloride | 495076-64-7 | - | |
GlyT2抑制剂 | ||||
| GC12489 | Ivacaftor benzenesulfonate | 1134822-09-5 | - | |
A CFTR potentiator | ||||
| GC12528 | NS309 | 18711-16-5 | >98.00% | |
NS309是中电导Ca 2+ 激活K + 通道KCa3.1最有效的正门控调制剂,EC 50 为75nmol/L。 | ||||
| GC12714 | Gabapentin | 60142-96-3 | >98.00% | |
An approved antiepileptic drug | ||||
| GC12858 | Phenytoin sodium | 630-93-3 | >99.50% | |
An anticonvulsant agent | ||||
| GC12911 | Tetracaine HCl | 136-47-0 | >99.50% / >99.00% | |
An Analytical Reference Standard | ||||
| GC12970 | Furosemide | 54-31-9 | >99.50% / >98.00% | |
A loop diuretic and an inhibitor of NKCC1 and NKCC2 | ||||
| GC13003 | AMG-517 | 659730-32-2 | >99.50% | |
A TRPV1 antagonist | ||||
| GC13016 | Safinamide | 133865-89-1 | >99.50% | |
Safinamide 是一种强效、选择性和可逆的单胺氧化酶 B (MAO-B) 抑制剂 (IC50=0.098 μM),优于 MAO-A (IC50=580 μM)。 | ||||
| GC13022 | Esomeprazole Magnesium trihydrate | 217087-09-7 | - | |
An H + /K + -ATPase inhibitor | ||||
