Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC13733A 438079 hydrochlorideCAS: 899431-18-6纯度: >99.50%
An antagonist of the nucleotide receptor P2X7
- GC13882Ranolazine 2HClCAS: 95635-56-6纯度: >99.50%
A piperazine derivative with cardioprotective activity
- GC13888Benidipine HClCAS: 91599-74-5纯度: >99.50% / >98.00%
An L-, T-, and N-type calcium channel blocker
- GC14313Esomeprazole MagnesiumCAS: 161973-10-0纯度: >98.00%
A form of esomeprazole in complex with magnesium
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13040 | TRAM-34 | 289905-88-0 | >99.50% | |
An IKCa1/K Ca 3.1 channel blocker | ||||
| GC13146 | Amlodipine Besylate | 111470-99-6 | >99.50% | |
An L-type calcium channel blocker | ||||
| GC13164 | Ampalex | 154235-83-3 | >99.50% | |
An AMPA receptor modulator | ||||
| GC13218 | TRPC6 inhibitor | 1333207-63-8 | - | |
A TRPC6 channel blocker | ||||
| GC13316 | Ivacaftor hydrate | 1134822-07-3 | >99.00% | |
A CFTR potentiator | ||||
| GC13397 | Proparacaine HCl | 5875-06-9 | - | |
voltage-gated sodium channels antagonist | ||||
| GC13523 | Amlodipine | 88150-42-9 | >99.50% | |
An L-type calcium channel blocker | ||||
| GC13527 | Gliclazide | 21187-98-4 | >99.50% | |
An inhibitor of pancreatic β-cell K ATP channels | ||||
| GC13698 | Nilvadipine | 75530-68-6 | >99.50% | |
An L-type calcium channel blocker | ||||
| GC13733 | A 438079 hydrochloride | 899431-18-6 | >99.50% | |
An antagonist of the nucleotide receptor P2X7 | ||||
| GC13792 | Rufinamide | 106308-44-5 | >99.50% | |
An anticonvulsant | ||||
| GC13802 | Riluzole | 1744-22-5 | >98.00% | |
Riluzole 是一种抗惊厥药,属于使用依赖性 Na+ 通道阻滞剂家族,它也可以抑制 GABA 摄取,IC50 为 43 μM。 | ||||
| GC13824 | Indapamide | 26807-65-8 | >99.50% / >98.00% | |
An Analytical Reference Standard | ||||
| GC13863 | 10Panx | 955091-53-9 | >98.00% | |
10Panx是一种强效的Panx1通道抑制剂,靶向Panx1蛋白ECL1结构域中的W74至Y83片段。 | ||||
| GC13882 | Ranolazine 2HCl | 95635-56-6 | >99.50% | |
A piperazine derivative with cardioprotective activity | ||||
| GC13888 | Benidipine HCl | 91599-74-5 | >99.50% / >98.00% | |
An L-, T-, and N-type calcium channel blocker | ||||
| GC14039 | MDL-29951 | 130798-51-5 | >99.50% | |
An NMDA receptor antagonist and GPR17 agonist | ||||
| GC14111 | (R)-baclofen | 69308-37-8 | >99.00% / >98.00% | |
(R)-巴氯芬 (Arbaclofen) 是一种选择性 GABAB 受体激动剂。 | ||||
| GC14313 | Esomeprazole Magnesium | 161973-10-0 | >98.00% | |
A form of esomeprazole in complex with magnesium | ||||
| GC14417 | NNC 55-0396 | 357400-13-6 | >99.00% | |
A selective T-type calcium channel inhibitor | ||||
| GC14580 | SB705498 | 501951-42-4 | >99.50% | |
SB705498是一种口服生物可利用的、竞争性的辣椒素介导的 TRPV1 受体拮抗剂(人类、大鼠和豚鼠的pKis分别为7.6、7.5和7.3)。SB705498能够快速、可逆地抑制辣椒素、酸或热介导的人类TRPV1激活。 | ||||
| GC14764 | Lamotrigine | 84057-84-1 | >99.50% | |
An anticonvulsant | ||||
| GC14792 | Reserpine hydrochloride | 16994-56-2 | >99.50% | |
Irreversible inhibitor of VMAT1 and VMAT2 | ||||
| GC14916 | Acamprosate calcium | 77337-73-6 | >98.00% | |
An NMDA modulator | ||||
