GABA Receptor
GABA Receptor(γ-氨基丁酸受体)
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
GABA Receptor 相关产品(219)
- GC10772FlumazenilCAS: 78755-81-4纯度: >99.50% / >98.00%
A GABA A receptor antagonist and partial agonist
- GA10004H-D-Met-OHCAS: 348-67-4纯度: >98.00%
H-D-Met-OH (MRX-1024; D-H-D-Met-OH) 是一种有效的化学保护剂,还可以通过 GABAA 受体激活抑制神经元活性。
- GC10101SR 95531 hydrobromideCAS: 104104-50-9纯度: >98.00% / >97.00%
SR 95531 氢溴酸盐 (Gabazine) 是 GABAA 受体上 GABA 结合位点的选择性拮抗剂 。
- GC10262Tracazolate hydrochlorideCAS: 1135210-68-2
Tracazolate (ICI 136753) hydrochloride 是一种有效的 GABAA 受体调节剂。
- GC10530Dihydroergotoxine mesylateCAS: 8067-24-1纯度: >98.00%
A mixture of alkaloids with diverse biological activities
- GC10856THIP hydrochlorideCAS: 85118-33-8纯度: >99.00%
A GABA A receptor agonist and GABA C receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10772 | Flumazenil | 78755-81-4 | >99.50% / >98.00% | |
A GABA A receptor antagonist and partial agonist | ||||
| GC10974 | AWD 131-138 | 188116-07-6 | >99.00% | |
A partial agonist of the GABA A receptor | ||||
| GC11901 | Nefiracetam | 77191-36-7 | >99.00% | |
An Analytical Reference Standard | ||||
| GC12714 | Gabapentin | 60142-96-3 | >98.00% | |
An approved antiepileptic drug | ||||
| GC13792 | Rufinamide | 106308-44-5 | >99.50% | |
An anticonvulsant | ||||
| GC14111 | (R)-baclofen | 69308-37-8 | >99.00% / >98.00% | |
(R)-巴氯芬 (Arbaclofen) 是一种选择性 GABAB 受体激动剂。 | ||||
| GC14916 | Acamprosate calcium | 77337-73-6 | >98.00% | |
An NMDA modulator | ||||
| GC16564 | Niflumic acid | 4394-00-7 | >99.50% | |
A selective COX-2 inhibitor | ||||
| GA10004 | H-D-Met-OH | 348-67-4 | >98.00% | |
H-D-Met-OH (MRX-1024; D-H-D-Met-OH) 是一种有效的化学保护剂,还可以通过 GABAA 受体激活抑制神经元活性。 | ||||
| GA10664 | H-Dab•HBr | 1758-80-1 | >98.00% | |
H-Dab•HBr (L-2,4-Diaminobutyric acid) 是一周 GABA 转氨酶抑制剂,IC50 大于 500 μM;在体内和体外均表现出抗肿瘤活性。 | ||||
| GC10065 | (-)-Bicuculline methiodide | 40709-69-1 | - | |
GABAA受体拮抗剂 | ||||
| GC10101 | SR 95531 hydrobromide | 104104-50-9 | >98.00% / >97.00% | |
SR 95531 氢溴酸盐 (Gabazine) 是 GABAA 受体上 GABA 结合位点的选择性拮抗剂 。 | ||||
| GC10183 | TPMPA | 182485-36-5 | >95.00% | |
A selective GABA A -ρ1 (ρ1 GABA C ) receptor antagonist | ||||
| GC10186 | Tiagabine | 115103-54-3 | 99.98% | |
A GAT-1 inhibitor | ||||
| GC10262 | Tracazolate hydrochloride | 1135210-68-2 | - | |
Tracazolate (ICI 136753) hydrochloride 是一种有效的 GABAA 受体调节剂。 | ||||
| GC10313 | ZAPA sulfate | 371962-01-5 | - | |
GABAA receptors agonist | ||||
| GC10489 | CGP 54626 hydrochloride | 149184-21-4 | ≥95.00% | |
A selective GABA B receptor antagonist | ||||
| GC10530 | Dihydroergotoxine mesylate | 8067-24-1 | >98.00% | |
A mixture of alkaloids with diverse biological activities | ||||
| GC10641 | AA 29504 | 945828-50-2 | - | |
GABAA receptor modulator | ||||
| GC10741 | TCS 1205 | 355022-97-8 | - | |
TCS 1205 (compound 2b) 是一种有效的选择性 GABAA 激动剂。 | ||||
| GC10844 | SCS | 3232-36-8 | - | |
GABAA receptor antagonist | ||||
| GC10856 | THIP hydrochloride | 85118-33-8 | >99.00% | |
A GABA A receptor agonist and GABA C receptor antagonist | ||||
| GC10888 | SCH 50911 | 733717-87-8 | - | |
SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-乙酸,一种选择性、口服活性和竞争性 γ-氨基丁酸 B GABA(B) 受体拮抗剂,与 GABA(B ) 受体,IC50 为 1.1 μM。 | ||||
| GC10967 | TACA | 38090-53-8 | - | |
An agonist of homomeric GABA A receptors | ||||
