GlpBio

GABA Receptor

GABA Receptor(γ-氨基丁酸受体)

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

GABA Receptor 相关产品(219)

  • GC17223 structure
    GC1722317-PA
    CAS: 694438-95-4

    17-PA 是神经类固醇增强和 GABAA 受体直接门控的选择性拮抗剂。

  • GC17257 structure
    GC17257Saclofen
    CAS: 125464-42-8
    纯度: >98.00% / >99.00%

    Saclofen是一种口服竞争性GABAB受体拮抗剂，IC 50 值为7.8μM。

  • GC17321 structure
    GC17321RuBi-GABA
    CAS: 1028141-88-9

    RuBi-GABA 是一种新型的钌基笼状 GABA 化合物。

  • GC17350 structure
    GC17350L-655,708
    CAS: 130477-52-0
    纯度: >99.00% / >98.00% / >98.50%

    A ligand for α 5 subunit-containing GABA A receptors with nootropic activity

  • GC17381 structure
    GC17381trans-4-Hydroxycrotonic acid
    CAS: 24587-49-3

    ligand of γ-hydroxybutyric acid (GHB) receptor

  • GC17399 structure
    GC17399Pregnanolone
    CAS: 128-20-1

    GABAA receptor positive allosteric modulator

  • GC17402 structure
    GC17402Tiagabine hydrochloride
    CAS: 145821-59-6
    纯度: >99.50%

    A GAT-1 inhibitor

  • GC17934 structure
    GC17934TB 21007
    CAS: 207306-50-1

    An inverse agonist of α 5 β 3 γ 2 subunit-containing GABA A receptors

  • GC18299 structure
    GC18299Lorediplon
    CAS: 917393-39-6
    纯度: >99.50%

    A ligand for α 1 subunit-containing GABA A receptors

  • GC19057 structure
    GC19057Basmisanil
    CAS: 1159600-41-5
    纯度: >99.50%

    A negative allosteric modulator of α 5 subunit-containing GABA A receptors

  • GC19271 structure
    GC19271ONO-8590580
    CAS: 1802661-73-9
    纯度: >99.00%

    A negative allosteric modulator of α 5 subunit-containing GABA A receptors

  • GC25531 structure
    GC25531Isonipecotic acid
    CAS: 498-94-2

    Isonipecotic acid (4-Piperidinecarboxylic acid, 4-Carboxypiperidine, Hexahydroisonicotinic acid) is a heterocyclic compound that mainly acts as a GABAA receptor partial agonist.

  • GC25566 structure
    GC25566L-DAB HBR
    CAS: 73143-97-2

    L-DAB HBR (L-Dab Hydrobromide, L-2,4-Diaminobutyric acid hydrobromide) is an inhibitor of GABA (Gamma-aminobutyric acid) transaminase with IC50 of >500 μM

  • GC30088 structure
    GC30088Fluxametamide
    CAS: 928783-29-3
    纯度: >98.50% / >98.00%

    Fluxametamide是一种GABA和谷氨酸门控氯离子通道的拮抗剂，对GABACls和GluCls的IC 50 值分别为1.95nM和225nM。

  • GC30433 structure
    GC30433Ru-32514
    CAS: 90807-98-0

    Ru-32514是一种苯二氮受体(benzodiazepinereceptor)激动剂。

  • GC30521 structure
    GC30521Broflanilide
    CAS: 1207727-04-5
    纯度: >98.00%

    Broflanilide是一种杀虫剂，可以分解成desmethyl-broflanilide，为特异性的昆虫耐狄氏剂的GABAreceptor拮抗剂，抑制斜纹夜蛾RDLGABAR，IC50值为1.3nM。

  • GC30827 structure
    GC30827Pipequaline (PK-8165)
    CAS: 77472-98-1
    纯度: >99.50%

    A partial agonist of central benzodiazepine receptors

  • GC30844 structure
    GC30844Afloqualone
    CAS: 56287-74-2
    纯度: >98.00%

    An Analytical Reference Standard

  • GC30862 structure
    GC30862L-Cycloserine ((S)-4-Amino-3-isoxazolidone)
    CAS: 339-72-0
    纯度: >99.00%

    An inhibitor of sphingolipid synthesis and aminotransferases

  • GC30865 structure
    GC30865TPA 023
    CAS: 252977-51-8
    纯度: >99.50%

    TPA023是GABAAα2/α3的选择性的激动剂，Ki值为0.19-0.41nM。

  • GC30889 structure
    GC30889(-)-Securinine
    CAS: 5610-40-2
    纯度: >98.00%

    An alkaloid

  • GC30898 structure
    GC308986-Methylflavone
    CAS: 29976-75-8
    纯度: >98.00%

    6-methylflavone是α1β2γ2L和α1β2GABAA受体的激活剂。

  • GC30930 structure
    GC30930DAA-1106
    CAS: 220551-92-8
    纯度: >99.50%

    A TSPO agonist

  • GC30933 structure
    GC30933(+)-Kavain
    CAS: 500-64-1
    纯度: >98.00%

    A kavalactone with diverse biological activities