GABA Receptor
GABA Receptor(γ-氨基丁酸受体)
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
GABA Receptor 相关产品(219)
- GC309436,2'-DihydroxyflavoneCAS: 92439-20-8纯度: >99.50% / >98.00%
6,2'-Dihydroxyflavone是一个新型的GABAA受体拮抗剂。
- GC30983alpha-Asarone (α-Asarone)CAS: 2883-98-9纯度: >99.50%
An inhibitor of HMG- CoA reductase and CYP450 isoforms
- GC31120CirsimaritinCAS: 6601-62-3纯度: >98.00%
Cirsimaritin是一种存在于植物中的二甲氧基黄酮，具有抗癌潜力，并显示出显著的抗菌、抗氧化、解痉作用，同时还可抑制环氧合酶-1。
- GC31121S-8510 phosphate (SB-737552 phosphate)CAS: 151466-23-8
S-8510 (phosphate) 是一种反向苯二氮卓 (BDZ) 受体激动剂，对 -GABA 和 +GABA 的 Kis 分别为 34.6 nM、36.2 nM。
- GC31257Rilmazafone hydrochloride (450191S)CAS: 85815-37-8纯度: >99.50%
Rilmazafone hydrochloride (450191S) (450191S) 是苯二氮卓 (omega) 配体。
- GC31282p-HydroxybenzaldehydeCAS: 123-08-0
p-Hydroxybenzaldehyde (4-Hydroxybenzaldehyde, 4-Formylphenol, p-Formylphenol), which can be found in the orchids Gastrodia elata, Galeola faberi and vanilla, is a hydroxybenzaldehyde that reacts with NAD+ and H2O to produce 4-hydroxybenzoate, NADH, and 2 protons. p-Hydroxybenzaldehyde at 101.7 μM can significantly reduce the GABA-induced chloride current of GABAA receptors(α1β2γ2S subtype) expressed.
- GC337033,4,5-Trimethoxycinnamic acidCAS: 90-50-6 ; 20329-98-0纯度: >99.00%
3,4,5-Trimethoxycinnamic acid (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the GABAA/BZ receptor complex.
- GC34064Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)CAS: 2921-14-4纯度: >98.00%
Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)是一种苹果酸-天冬氨酸穿梭（MAS）抑制剂和γ-氨基丁酸转氨酶（GABA-T）抑制剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC30943 | 6,2'-Dihydroxyflavone | 92439-20-8 | >99.50% / >98.00% | |
6,2'-Dihydroxyflavone是一个新型的GABAA受体拮抗剂。 | ||||
| GC30983 | alpha-Asarone (α-Asarone) | 2883-98-9 | >99.50% | |
An inhibitor of HMG- CoA reductase and CYP450 isoforms | ||||
| GC31010 | AZD-6280 | 942436-93-3 | >99.00% | |
AZD-6280 is a selective GABAA (α2/3) receptor modulator, used for treatment of generalized anxiety disorder. | ||||
| GC31013 | U-101017 (PNU 101017) | 170568-47-5 | - | |
U-101017 (PNU 101017) 是苯二氮卓受体和 GABAA 受体的部分激动剂，具有抗焦虑作用。 | ||||
| GC31018 | NEO 376 (SPI-376) | 496921-73-4 | - | |
NEO 376 (SPI-376) 是 5-HT1 受体、GABA 受体和多巴胺受体的选择性调节剂，具有抗精神病活性。 | ||||
| GC31023 | Ethyl dirazepate | 23980-14-5 | - | |
Ethyldirazepate是一种苯并二氮杂(benzodiazepine)衍生物。具有抗焦虑和催眠特性。 | ||||
| GC31049 | RWJ-51204 | 205701-85-5 | - | |
RWJ-51204是GABA(A)receptor的部分激动剂，Ki值为0.2-2nM。 | ||||
| GC31052 | CP-409092 | 194098-25-4 | - | |
CP-409092是GABA(A)的部分激动剂，主要用于抗焦虑研究。 | ||||
| GC31112 | Sarmazenil (Ro 15-3505) | 78771-13-8 | - | |
Sarmazenil (Ro 15-3505) 是一种苯二氮卓受体拮抗剂。 | ||||
| GC31120 | Cirsimaritin | 6601-62-3 | >98.00% | |
Cirsimaritin是一种存在于植物中的二甲氧基黄酮，具有抗癌潜力，并显示出显著的抗菌、抗氧化、解痉作用，同时还可抑制环氧合酶-1。 | ||||
| GC31121 | S-8510 phosphate (SB-737552 phosphate) | 151466-23-8 | - | |
S-8510 (phosphate) 是一种反向苯二氮卓 (BDZ) 受体激动剂，对 -GABA 和 +GABA 的 Kis 分别为 34.6 nM、36.2 nM。 | ||||
| GC31142 | Uldazepam (U31920) | 28546-58-9 | - | |
Uldazepam (U31920) 是一种苯二氮卓类衍生物，具有治疗焦虑症的潜力。 | ||||
| GC31196 | SX-3228 | 156364-04-4 | - | |
SX-3228是一种选择性苯二氮卓类(benzodiazepine1，BZ1)受体激动剂，IC50为17nM。 | ||||
| GC31224 | Carburazepam (RGH 3331) | 59009-93-7 | - | |
Carburazepam (RGH 3331) 是一种衍生自苯二氮卓类药物的药物。 | ||||
| GC31257 | Rilmazafone hydrochloride (450191S) | 85815-37-8 | >99.50% | |
Rilmazafone hydrochloride (450191S) (450191S) 是苯二氮卓 (omega) 配体。 | ||||
| GC31282 | p-Hydroxybenzaldehyde | 123-08-0 | - | |
p-Hydroxybenzaldehyde (4-Hydroxybenzaldehyde, 4-Formylphenol, p-Formylphenol), which can be found in the orchids Gastrodia elata, Galeola faberi and vanilla, is a hydroxybenzaldehyde that reacts with NAD+ and H2O to produce 4-hydroxybenzoate, NADH, and 2 protons. p-Hydroxybenzaldehyde at 101.7 μM can significantly reduce the GABA-induced chloride current of GABAA receptors(α1β2γ2S subtype) expressed. | ||||
| GC31990 | Bamaluzole | 87034-87-5 | - | |
Bamaluzole是一个GABA受体激动剂，来自专利WO2012064642A1。 | ||||
| GC33504 | 4-Acetamidobutanoic acid (N-acetyl GABA) | 3025-96-5 | >98.00% | |
A GABA derivative | ||||
| GC33703 | 3,4,5-Trimethoxycinnamic acid | 90-50-6 ; 20329-98-0 | >99.00% | |
3,4,5-Trimethoxycinnamic acid (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the GABAA/BZ receptor complex. | ||||
| GC33751 | CGP11952 | 64078-09-7 | - | |
CGP11952是一种三唑基Benzaphenon。CGP11952是一种苯二氮卓类(benzodiazepine)衍生物。 | ||||
| GC33754 | FG8119 (NNC13-8119) | 106447-61-4 | - | |
FG8119 (NNC13-8119) 是一种从美国专利 4745112 A 中提取的新型苯二氮卓类激动剂。 | ||||
| GC34064 | Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) | 2921-14-4 | >98.00% | |
Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)是一种苹果酸-天冬氨酸穿梭（MAS）抑制剂和γ-氨基丁酸转氨酶（GABA-T）抑制剂。 | ||||
| GC34362 | SSD114 hydrochloride | 2319790-02-6 | >99.00% | |
SSD114hydrochloride是一种新型GABAB受体正变构调节剂。 | ||||
| GC34494 | Bifenazate | 149877-41-8 | >99.50% | |
An acaricide | ||||