GlpBio

Monoamine transporter

Monoamine transporter(单胺转运蛋白)

Monoamine transporters are a family of plasma membrane transporter that regulates the reuptake of neurotransmitters into nerve terminals. It divided into DAT (dopamine transporter), NET (norepinephrine transporter) and SERT (serotonin transporter).

Monoamine transporter 相关产品(15)

  • GC14792 structure
    GC14792Reserpine hydrochloride
    CAS: 16994-56-2
    纯度: >99.50%

    Irreversible inhibitor of VMAT1 and VMAT2

  • GC13672 structure
    GC13672Tetrabenazine
    CAS: 58-46-8
    纯度: >99.50%

    丁苯那嗪是美国食品和药物管理局唯一批准的亨廷顿舞蹈病药物，适用于治疗与亨廷顿舞蹈病相关的舞蹈症。

  • GC19370 structure
    GC19370Valbenazine
    CAS: 1025504-45-3
    纯度: >99.00%

    An inhibitor of VMAT2

  • GC26029 structure
    GC26029Valbenazine tosylate
    CAS: 1639208-54-0

    Valbenazine tosylate (NBI-98854) is the tosylate salt of valbenazine, a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).

  • GC30994 structure
    GC30994Vanilpyruvic acid (Vanylpyruvic acid)
    CAS: 1081-71-6
    纯度: >98.00%

    香草丙酮酸 (Vanylpyruvic acid) 是儿茶酚胺代谢物和香草乳酸的前体。

  • GC31060 structure
    GC31060Radafaxine hydrochloride (GW-353162A)
    CAS: 106083-71-0
    纯度: >99.50%

    An active metabolite of bupropion

  • GC36705 structure
    GC36705NBI-98782
    CAS: 85081-18-1
    纯度: >98.50%

    NBI-98782是一种强效且选择性的vesicular monoamine transporter 2 (VMAT2)抑制剂，K i 值为3nM。

  • GC37768 structure
    GC37768Tetrabenazine Racemate
    CAS: 718635-93-9
    纯度: >98.00%

    Tetrabenazine (Racemate)是一个有选择性和可逆转的VMAT-2抑制剂。

  • GC37820 structure
    GC37820Trans (2,3)-Dihydrotetrabenazine
    CAS: 171598-74-6

    Trans (2,3)-Dihydrotetrabenazine， 是抗精神病药物Tetrabenazine的体内代谢物，能够抑制囊泡单胺转运体 2 (VMAT2)。

  • GC40180 structure
    GC40180Tetrabenazine-d6
    CAS: 1392826-25-3
    纯度: >99.00%

    An internal standard for the quantification of tetrabenazine

  • GC50649 structure
    GC50649FFN 200 dihydrochloride
    CAS: 2080306-27-8
    纯度: >98.00%

    Selective fluorescent VMAT2 substrate

  • GC69565 structure
    GC69565Nisoxetine
    CAS: 53179-07-0
    纯度: >98.00%

    Nisoxetine 是一种有效的和选择性的去甲肾上腺素转运蛋白 (NET) 抑制剂，Kd 值为 0.76 nM。Nisoxetine 是一种抗抑郁试剂和局部麻药，它可以阻断电压门控性钠通道。

  • GC70443 structure
    GC70443GZ-793A
    CAS: 1356447-90-9
    纯度: >99.00%

    GZ-793A是一种口服活性和选择性囊泡单胺转运蛋白-2（VMAT2）抑制剂，Ki为0.029µM。

  • GC73217 structure
    GC73217FFN246
    CAS: 2210244-83-8
    纯度: >99.00%

    FFN246是血清素转运蛋白（SERT）探针和水疱单胺转运蛋白2 （VMAT2）的荧光双底物，激发和发射光谱为392/427 nm。

  • GN10779 structure
    GN10779Reserpine
    CAS: 50-55-5
    纯度: >98.50%

    Irreversible inhibitor of VMAT1 and VMAT2