Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC16986SDZ 220-581 hydrochlorideCAS: 179411-93-9纯度: >99.50%
SDZ 220-581 hydrochloride 是一种口服有效的竞争性 NMDA 受体拮抗剂,pKi 值为 7.7。
- GC17106Verapamil HClCAS: 152-11-4纯度: >99.50% / >99.00%
Verapamil HCl是 L 型钙通道阻滞剂和肾上腺素能受体拮抗剂,常用于高血压、心律失常和心绞痛的研究。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16561 | Gliquidone | 33342-05-1 | >99.00% | |
A second generation sulfonylurea | ||||
| GC16564 | Niflumic acid | 4394-00-7 | >99.50% | |
A selective COX-2 inhibitor | ||||
| GC16570 | Lansoprazole | 103577-45-3 | >98.00% | |
Proton pump inhibitor | ||||
| GC16616 | (+)-MK 801 | 70449-94-4 | >98.00% | |
强效 NMDA 拮抗剂 | ||||
| GC16672 | Zosuquidar | 167354-41-8 | >98.00% | |
A modulator of P-gp | ||||
| GC16696 | Dibucaine (Cinchocaine) HCl | 61-12-1 | - | |
An Analytical Reference Standard | ||||
| GC16882 | Icilin | 36945-98-9 | - | |
An agonist of CMR1/TRPM8 | ||||
| GC16889 | Nisoldipine | 63675-72-9 | >99.00% | |
A calcium channel inhibitor | ||||
| GC16986 | SDZ 220-581 hydrochloride | 179411-93-9 | >99.50% | |
SDZ 220-581 hydrochloride 是一种口服有效的竞争性 NMDA 受体拮抗剂,pKi 值为 7.7。 | ||||
| GC16999 | Nitrendipine | 39562-70-4 | >99.00% | |
An L-type calcium channel blocker | ||||
| GC17106 | Verapamil HCl | 152-11-4 | >99.50% / >99.00% | |
Verapamil HCl是 L 型钙通道阻滞剂和肾上腺素能受体拮抗剂,常用于高血压、心律失常和心绞痛的研究。 | ||||
| GC17152 | Dofetilide | 115256-11-6 | >98.00% | |
An antiarrythmic agent that inhibits potassium channels | ||||
| GC17173 | Felodipine | 72509-76-3 | >98.50% | |
An L-type calcium channel inhibitor | ||||
| GC17212 | A 438079 | 899507-36-9 | >99.50% | |
A 438079是一种高选择性P2X7受体(P2X7R)拮抗剂,对大鼠P2X7R的IC 50 值为0.1μM。 | ||||
| GC17316 | Gabapentin HCl | 60142-95-2 | >98.00% | |
An approved antiepileptic drug | ||||
| GC17340 | Carbamazepine | 298-46-4 | >99.50% | |
卡马西平是一种钠通道阻滞剂,是一种抗惊厥药。 | ||||
| GC17587 | Manidipine | 89226-50-6 | - | |
An L- and T-type calcium channel blocker | ||||
| GC17710 | A-317491 | 475205-49-3 | >99.00% | |
A-317491是一种高亲和力、选择性的P2X3和P2X2/3受体激活拮抗剂,其对大鼠P2X3和P2X2/3的K i 值分别为22nM和92nM。 | ||||
| GC17804 | GlyH-101 | 328541-79-3 | >98.00% | |
A reversible CFTR channel blocker | ||||
| GC17852 | Gue 1654 | 397290-30-1 | - | |
Gue 1654 是 OXE-R 的调节剂。 | ||||
| GC17918 | Capsazepine | 138977-28-3 | >99.00% | |
Capsazepine是瞬时受体电位香草素1(TRPV1)受体的特异性拮抗剂,IC 50 值为562 nM。 | ||||
| GC17952 | Zonisamide sodium | 68291-98-5 | - | |
A broad-spectrum sulfonamide antiepileptic agent | ||||
| GC18118 | SDZ 220-581 | 174575-17-8 | >99.00% | |
SDZ 220-581 是一种具有口服活性、强效、竞争性 NMDA 受体拮抗剂,pKi 值为 7.7。 | ||||
| GC38465 | GsMTx4 | 1209500-46-8 | >98.00% | |
GsMTx4是一种由34个氨基酸组成的蜘蛛毒素肽,属于huwentoxin-1家族。 | ||||
