Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
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- MCT(3)
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- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC15270(-)-MK-801 maleateCAS: 121917-57-5纯度: >98.00%
(-)-MK 801是一种选择性、非竞争性N-甲基-D-天冬氨酸(NMDA)受体拮抗剂(K i = 211.7nM)。
- GC15363Felbamate hydrateCAS: 1177501-39-1
An inhibitor of NMDA receptors and a modulator of GABA A receptors
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC14977 | Minoxidil | 38304-91-5 | >99.00% | |
An anti-hypertensive vasodilator | ||||
| GC14991 | ML133 HCl | 1222781-70-5 | >98.00% | |
A K ir 2 channel inhibitor | ||||
| GC15101 | Azelnidipine | 123524-52-7 | >99.50% | |
A calcium channel blocker | ||||
| GC15270 | (-)-MK-801 maleate | 121917-57-5 | >98.00% | |
(-)-MK 801是一种选择性、非竞争性N-甲基-D-天冬氨酸(NMDA)受体拮抗剂(K i = 211.7nM)。 | ||||
| GC15293 | Manidipine 2HCl | 89226-75-5 | >98.50% | |
An L- and T-type calcium channel blocker | ||||
| GC15363 | Felbamate hydrate | 1177501-39-1 | - | |
An inhibitor of NMDA receptors and a modulator of GABA A receptors | ||||
| GC15419 | Glipizide | 29094-61-9 | >99.50% | |
A hypoglycemic agent | ||||
| GC15458 | Ambroxol HCl | 23828-92-4 | >98.00% | |
An expectorant | ||||
| GC15467 | ALX 5407 hydrochloride | 200006-08-2 | - | |
An inhibitor of GlyT1 | ||||
| GC15524 | Bumetanide | 28395-03-1 | >99.50% | |
An NKCC1 inhibitor | ||||
| GC15550 | Lacidipine | 103890-78-4 | >99.50% | |
An L-type calcium channel blocker | ||||
| GC15552 | Nicorandil | 65141-46-0 | >99.50% | |
A SUR2B/K ir 6.2 activator and nitric oxide donor | ||||
| GC15570 | Tariquidar | 206873-63-4 | >98.50% | |
Tariquidar是一种高效、选择性的P-糖蛋白抑制剂,K D 值为5.1nM。 | ||||
| GC15701 | A-803467 | 944261-79-4 | >98.50% | |
A-803467是一种河豚毒素耐受型Na v 1.8钠通道的阻断剂,其阻断人Na v 1.8钠通道的IC 50 为8nM。 | ||||
| GC15823 | Flecainide acetate | 54143-56-5 | >99.50% | |
An inhibitor of cardiac late sodium current | ||||
| GC15860 | Ibutilide Fumarate | 122647-32-9 | >98.00% | |
A class III antiarrhythmic drug | ||||
| GC15947 | HC-030031 | 349085-38-7 | >98.00% | |
HC-030031是瞬时受体电位锚蛋白亚家族成员1(TRPA1)的选择性抑制剂。HC-030031可阻断细胞的钙流入,对肉桂醛和异硫氰酸烯丙酯(AITC)诱导的钙内流的IC 50 值分别为4.9±0.1和7.5±0.2μM。 | ||||
| GC16036 | Repaglinide | 135062-02-1 | >99.50% | |
An ATP-dependent potassium channel blocker | ||||
| GC16086 | Phenytoin | 57-41-0 | >99.50% | |
An anticonvulsant agent | ||||
| GC16128 | Clevidipine Butyrate | 167221-71-8 | >99.50% | |
An inhibitor of L-type calcium channels | ||||
| GC16173 | Procaine HCl | 51-05-8 | - | |
An Analytical Reference Standard | ||||
| GC16402 | Org 24598 lithium salt | 722456-08-8 | - | |
glial glycine transporter (GlyT1) inhibitor | ||||
| GC16453 | Zinc Pyrithione | 13463-41-7 | >98.00% | |
A coordination complex of zinc and pyrithione | ||||
| GC16532 | Flunarizine 2HCl | 30484-77-6 | >99.50% | |
A calcium antagonist | ||||
