GlpBio

Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel(跨膜转运)

研究方向

Membrane Transporter/Ion Channel 相关产品(2265)

  • GC34998 structure
    GC34998(S)-(-)-5-Fluorowillardiine hydrochloride
    CAS: 1321546-70-6
    纯度: >99.50%

    (S)-(-)-5-Fluorowillardiine hydrochloride 是AMPAR高效选择性激动剂。

  • GC35010 structure
    GC35010(Z)-Capsaicin
    CAS: 25775-90-0
    纯度: >99.50%

    Zucapsaicin, the cis-isomer of capsaicin, is a topical analgesic used to treat osteoarthritis of the knee and other neuropathic pain. It is also a TRPV-1 modulator.

  • GC35075 structure
    GC3507520-HETE
    CAS: 79551-86-3
    纯度: >98.00%

    A cytochrome P450 (CYP450) metabolite of arachidonic acid

  • GC35108 structure
    GC351083-Deoxyaconitine
    CAS: 3175-95-9
    纯度: >98.50%

    3-Deoxyaconitine is a diterpenoid alkaloid isolated from the root of Aconitum Carmichaeli Debx.

  • GC35147 structure
    GC351475-(N,N-Hexamethylene)-amiloride
    CAS: 1428-95-1
    纯度: >98.00%

    5-(N,N-Hexamethylene)-amiloride是一种强效的Na + /H + 交换体抑制剂，对肿瘤细胞具有毒性。

  • GC35211 structure
    GC35211A-317491 sodium salt hydrate
    纯度: >99.50%

    A P2X 3 and P2X 2/3 receptor antagonist

  • GC35222 structure
    GC35222ABT-239
    CAS: 460746-46-7
    纯度: >99.00%

    ABT-239 是一种新颖的，高效的，非咪唑类的 H3R 拮抗剂，也是 TRPV1 的拮抗剂。

  • GC35273 structure
    GC35273Ajmaline
    CAS: 4360-12-7
    纯度: >99.50%

    Ajmaline是一种生物碱, 是一种Ia类的抗心律失常药。

  • GC35293 structure
    GC35293Allocryptopine
    CAS: 485-91-6
    纯度: >98.00%

    An isoquinoline alkaloid with antimicrobial activity

  • GC35316 structure
    GC35316AMG2850
    CAS: 1470018-52-0

    AMG2850 是一个有效的、有口服活性的TRPM8 的选择性拮抗剂。

  • GC35322 structure
    GC35322Amiodarone
    CAS: 1951-25-3

    Amiodarone (NSC 85442,Amiodar,Amiodarone hydrochloride,Nexterone) HCl is a sodium/potassium-ATPase inhibitor and an autophagy activator, used to treat various types of cardiac dysrhythmias.

  • GC35325 structure
    GC35325Amlodipine maleate
    CAS: 88150-47-4
    纯度: >99.50%

    Amlodipine (Amvaz, UK-48340) maleate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.

  • GC35407 structure
    GC35407Asivatrep
    CAS: 1005168-10-4
    纯度: >95.00%

    Asivatrep是一种强效、选择性、非甾体类的transient receptor potential vanilloid subfamily V member 1 (TRPV1)拮抗剂。

  • GC35421 structure
    GC35421ATP synthase inhibitor 1
    CAS: 1023043-30-2
    纯度: >99.50%

    ATP synthase inhibitor 1 是一种 F1/FO-ATP 合酶复合物 c 亚基的有效抑制剂，抑制线粒体通透性转换孔的开放，但不影响 ATP 的水平。

  • GC35451 structure
    GC35451Azelnidipine D7

    Azelnidipine D7是Azelnidipine氘代化合物标准品。

  • GC35453 structure
    GC35453Azimilide Dihydrochloride
    CAS: 149888-94-8
    纯度: >98.00% / >97.50%

    A class III antiarrhythmic agent

  • GC35469 structure
    GC35469Barnidipine
    CAS: 104713-75-9

    A calcium channel blocker

  • GC35501 structure
    GC35501Beta-Eudesmol
    CAS: 473-15-4
    纯度: >98.00%

    A sesquiterpene with diverse biological activities

  • GC35527 structure
    GC35527Bitopertin R enantiomer
    CAS: 845614-12-2

    Bitopertin R enantiomer (RG1678 R enantiomer; RO4917838 R enantiomer) 是 Bitopertin 的R型对映体。Bitopertin是非竞争性甘氨酸重吸收 (GlyT1) 抑制剂。

  • GC35538 structure
    GC35538BNC375
    CAS: 1557240-80-8
    纯度: >99.50%

    BNC375 是一种口服有效的选择性 α7nAChRs I 型正向变构调节剂，EC50 为 1.9 μM。

  • GC35567 structure
    GC35567Bullatine A
    CAS: 1354-84-3

    Bullatine A (BLA) 雪上一枝蒿甲素是乌头属 genus Aconitum 的二萜类生物碱，具有抗风湿，抗炎和抗伤害感受作用。 Bullatine A 是一种有效的 P2X7 拮抗剂，可抑制 ATP 诱导的细胞凋亡和 P2X 受体介导的炎症反应。Bullatine A 能缓解过敏反应。

  • GC35568 structure
    GC35568Bulleyaconitine A
    CAS: 107668-79-1
    纯度: >99.00%

    Bulleyaconi cine A (Bulleyaconitine A, BLA) is an active ingredient of Aconitum bulleyanum plants and classified as an "aconitine-like" alkaloid. It is a potent use-dependent blocker for both Nav1.7 and Nav1.8 Na+ currents.

  • GC35619 structure
    GC35619Cav 2.2 blocker 1
    CAS: 1567335-29-8
    纯度: >99.00%

    Cav 2.2 blocker 1 (compound 9) is a N-type calcium channel (Cav 2.2) blocker for the treatment of pain with IC50 of 0.001 μM.

  • GC35667 structure
    GC35667CFTR corrector 1
    CAS: 2216712-66-0
    纯度: >99.50%

    An F508del-CFTR corrector and potentiator